Page last updated: 2024-08-21

phenazocine and u-50488

phenazocine has been researched along with u-50488 in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19906 (46.15)18.7374
1990's4 (30.77)18.2507
2000's0 (0.00)29.6817
2010's3 (23.08)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bridges, RS; Kinsley, CH; Mann, PE1
Cone, EJ; Johnson, RE; Su, TP; Vaupel, DB1
France, CP; Snyder, AM; Woods, JH1
Cowan, A; Jacoby, HI; Vaught, JL1
Cooper, SJ; Jackson, A; Kirkham, TC1
Burks, TF; Hirning, LD; Porreca, F1
Dykstra, LA; Picker, M1
Dykstra, LA; Heise, JW; Picker, M1
Brusa, L; D'Amore, A; Lorenzini, P; Massotti, M1
Chiou, GC; el Messiry, S; Rohde, BH; Zhu, M1
Isotani, K; Mori, T; Narita, M; Nomura, M; Suzuki, T; Torigoe, K; Tsukiyama, Y; Yoshizawa, K1
Hall, FS; Kitanaka, J; Kitanaka, N; Nishiyama, N; Takemura, M; Tanaka, K; Uhl, GR1
Halberstadt, AL; Hyun, J; Powell, SB; Ruderman, MA1

Reviews

1 review(s) available for phenazocine and u-50488

ArticleYear
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response

1985

Other Studies

12 other study(ies) available for phenazocine and u-50488

ArticleYear
Opioid receptor subtype involvement in maternal behavior in lactating rats.
    Neuroendocrinology, 1991, Volume: 53, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; beta-Endorphin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Lactation; Maternal Behavior; Morphine; Phenazocine; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu

1991
Kappa opioid partial agonist activity of the enkephalin-like pentapeptide BW942C based on urination and in vitro studies in humans and animals.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adult; Amino Acid Sequence; Animals; Diuresis; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Methionine; Enkephalins; Humans; In Vitro Techniques; Male; Molecular Sequence Data; Morphine; Naltrexone; Oligopeptides; Phenazocine; Pyrrolidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Urination; Vas Deferens

1990
Analgesic effects of phencyclidine-like drugs in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Alfentanil; Analgesia; Analgesics; Anesthetics; Animals; Anticonvulsants; Dextrorphan; Dibenzocycloheptenes; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Fentanyl; Ketamine; Macaca mulatta; Phenazocine; Phencyclidine; Pyrrolidines

1989
Mu and delta, but not kappa, opioid agonists induce contractions of the canine small intestine in vivo.
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dogs; Duodenum; Dynorphins; Electric Stimulation; Enkephalin, Methionine; Female; Gastrointestinal Motility; Male; Morphine; Morphine Derivatives; Naloxone; Peptide Fragments; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Mu, but not kappa, opioid agonists induce contractions of the canine small intestine ex vivo.
    European journal of pharmacology, 1985, Feb-12, Volume: 109, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzomorphans; Cyclazocine; Dimethylphenylpiperazinium Iodide; Dogs; Ethylketocyclazocine; Gastrointestinal Motility; In Vitro Techniques; Intestine, Small; Morphine; Nalorphine; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors

1987
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule

1987
Area tempestas modulates the behavioural responses to nociceptive stimuli in rats.
    Annali dell'Istituto superiore di sanita, 1993, Volume: 29, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anticonvulsants; Azocines; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Escape Reaction; Foot; Hot Temperature; Male; Morphine; Naltrexone; Narcotic Antagonists; Olfactory Pathways; Pain; Phenazocine; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Seizures; Tail

1993
Effects of some opiates and opioid peptide eyedrops on ocular melatonin regulation in rabbits.
    Ophthalmic research, 1993, Volume: 25, Issue:6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Binding Sites; Endorphins; Female; Melatonin; Ophthalmic Solutions; Phenazocine; Pyrrolidines; Rabbits; Radioimmunoassay; Receptors, Opioid; Retina; Uvea

1993
Sigma-1 receptor function is critical for both the discriminative stimulus and aversive effects of the kappa-opioid receptor agonist U-50488H.
    Addiction biology, 2012, Volume: 17, Issue:4

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Avoidance Learning; Conditioning, Psychological; Discrimination Learning; Discrimination, Psychological; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Narcotic Antagonists; Pentazocine; Phenazocine; Phencyclidine; Propylamines; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, sigma; Sigma-1 Receptor

2012
Straub tail reaction in mice treated with σ(1) receptor antagonist in combination with methamphetamine.
    Brain research, 2012, Oct-30, Volume: 1482

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Non-Narcotic; Animals; Antipsychotic Agents; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Male; Methamphetamine; Mice; Mice, Inbred Strains; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Phenazocine; Pyrimidines; Receptors, Opioid, delta; Reflex; Tail; Time Factors

2012
Effects of the psychotomimetic benzomorphan N-allylnormetazocine (SKF 10,047) on prepulse inhibition of startle in mice.
    Pharmacology, biochemistry, and behavior, 2016, Volume: 148

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anisoles; Dose-Response Relationship, Drug; Hallucinogens; Male; Mice; Mice, Inbred C57BL; Naltrexone; Phenazocine; Prepulse Inhibition; Propylamines; Receptors, Opioid, kappa; Receptors, Phencyclidine; Receptors, sigma; Reflex, Startle; Sigma-1 Receptor; Stereoisomerism

2016