Page last updated: 2024-09-03

l 687414 and ro 25-6981

l 687414 has been researched along with ro 25-6981 in 2 studies

Compound Research Comparison

Studies
(l 687414)
Trials
(l 687414)
Recent Studies (post-2010)
(l 687414)
Studies
(ro 25-6981)
Trials
(ro 25-6981)
Recent Studies (post-2010) (ro 25-6981)
13042210137

Protein Interaction Comparison

ProteinTaxonomyl 687414 (IC50)ro 25-6981 (IC50)
Glutamate receptor ionotropic, NMDA 2DHomo sapiens (human)0.006
Glutamate receptor ionotropic, NMDA 3BHomo sapiens (human)0.006
Prolyl endopeptidaseSus scrofa (pig)0.006
Delta-type opioid receptorMus musculus (house mouse)0.006
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.0311
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.058
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.0426
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.058
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)0.0315
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)0.006
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)0.024
Glutamate receptor ionotropic, NMDA 2CHomo sapiens (human)0.006
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.058
Glutamate receptor ionotropic, NMDA 3AHomo sapiens (human)0.006
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.058
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.058

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boyce, S; Hill, RG; Mason, G; O'Donnell, R; Rigby, M; Rupniak, NM; Sirinathsinghji, D; Webb, JK; Wyatt, A1
Elliot, J; Grimwood, S; Huscroft, I; Hutson, PH; Kennedy, J; Mohnen, K; Murray, F; Russell, MG1

Other Studies

2 other study(ies) available for l 687414 and ro 25-6981

ArticleYear
Selective NMDA NR2B antagonists induce antinociception without motor dysfunction: correlation with restricted localisation of NR2B subunit in dorsal horn.
    Neuropharmacology, 1999, Volume: 38, Issue:5

    Topics: Acetates; Amines; Animals; Anticonvulsants; Cyclohexanecarboxylic Acids; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Gabapentin; gamma-Aminobutyric Acid; Hyperalgesia; Lamotrigine; Male; Motor Activity; Pain Measurement; Phenols; Piperidines; Pyrrolidinones; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Triazines

1999
Modulation of [3H]MK-801 binding to NMDA receptors in vivo and in vitro.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Chromans; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Ketamine; Kinetics; Male; Membranes; Mice; Phencyclidine; Phenols; Piperazines; Piperidines; Pyrrolidinones; Quinolones; Radioligand Assay; Rats; Receptors, N-Methyl-D-Aspartate; Tritium

2000