Page last updated: 2024-08-21

indazoles and mln 8237

indazoles has been researched along with mln 8237 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Christian, S; Danciu, OC; Dudek, AZ; Fischer, JH; Liu, LC; Russell, MJ; Shah, HA; Venepalli, NK; Zacny, JP1
Khan, T; Prabhu, A; Sankhe, K1

Reviews

1 review(s) available for indazoles and mln 8237

ArticleYear
Design strategies, SAR, and mechanistic insight of Aurora kinase inhibitors in cancer.
    Chemical biology & drug design, 2021, Volume: 98, Issue:1

    Topics: Animals; Antineoplastic Agents; Aurora Kinase A; Azepines; Benzamides; Drug Approval; Drug Resistance; Drug Screening Assays, Antitumor; Flavones; Gene Expression Regulation; Humans; Indazoles; Neoplasms; Organophosphates; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Quinazolines; Structure-Activity Relationship

2021

Trials

1 trial(s) available for indazoles and mln 8237

ArticleYear
Phase I Study of Aurora A Kinase Inhibitor Alisertib (MLN8237) in Combination With Selective VEGFR Inhibitor Pazopanib for Therapy of Advanced Solid Tumors.
    American journal of clinical oncology, 2019, Volume: 42, Issue:5

    Topics: Adult; Age Factors; Aged; Azepines; Cohort Studies; Disease-Free Survival; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Female; Humans; Indazoles; Kaplan-Meier Estimate; Male; Maximum Tolerated Dose; Middle Aged; Neoplasm Invasiveness; Neoplasm Staging; Neoplasms; Patient Safety; Pyrimidines; Response Evaluation Criteria in Solid Tumors; Retrospective Studies; Risk Assessment; Sex Factors; Sulfonamides; Survival Analysis; Treatment Outcome

2019