Page last updated: 2024-09-03

gr 73632 and cp 96345

gr 73632 has been researched along with cp 96345 in 5 studies

Compound Research Comparison

Studies
(gr 73632)
Trials
(gr 73632)
Recent Studies (post-2010)
(gr 73632)
Studies
(cp 96345)
Trials
(cp 96345)
Recent Studies (post-2010) (cp 96345)
7719403116

Protein Interaction Comparison

ProteinTaxonomygr 73632 (IC50)cp 96345 (IC50)
Substance-P receptorHomo sapiens (human)0.0028
Substance-P receptorCavia porcellus (domestic guinea pig)0.0004

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buéno, L; Julia, V; Morteau, O1
Dray, A; Maggi, CA; Nagy, I; Urban, L; Woolf, CJ1
Honda, K; Kamiya, H; Nakayama, Y; Saigo, A; Saito, R; Takano, Y1
Ando, R; Inoue, M; Kisara, K; Sakurada, C; Sakurada, T; Tan-No, K; Watanabe, C1
Li, YS; Miyano, K; Nakata, Y; Tang, HB1

Other Studies

5 other study(ies) available for gr 73632 and cp 96345

ArticleYear
Involvement of neurokinin 1 and 2 receptors in viscerosensitive response to rectal distension in rats.
    Gastroenterology, 1994, Volume: 107, Issue:1

    Topics: Abdomen; Animals; Benzamides; Biphenyl Compounds; Colon; Colonic Diseases, Functional; Gastrointestinal Motility; Hypnotics and Sedatives; Indoles; Isoindoles; Male; Neurokinin A; Peptide Fragments; Piperidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Tachykinin; Rectum; Substance P; Tachykinins

1994
The role of neurokinin and N-methyl-D-aspartate receptors in synaptic transmission from capsaicin-sensitive primary afferents in the rat spinal cord in vitro.
    Neuroscience, 1993, Volume: 52, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Afferent Pathways; Animals; Biphenyl Compounds; Capsaicin; Ganglia, Spinal; In Vitro Techniques; Membrane Potentials; N-Methylaspartate; Neurokinin A; Neurons; Peptide Fragments; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Spinal Cord; Substance P; Synapses; Synaptic Transmission

1993
Role of NK-1 receptor in central cardiovascular regulation in rats: studies on a novel non-peptide antagonist, CP-96,345, of substance P NK-1 receptor.
    Regulatory peptides, 1993, Jul-02, Volume: 46, Issue:1-2

    Topics: Animals; Biphenyl Compounds; Blood Pressure; Cerebral Ventricles; Heart Rate; Hypnotics and Sedatives; Injections, Intraventricular; Male; Muscle Contraction; Neurokinin A; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Rats; Receptors, Neurokinin-1; Substance P; Tachykinins; Vas Deferens

1993
Spinal actions of GR73632, a novel tachykinin NK1 receptor agonist.
    Peptides, 1999, Volume: 20, Issue:2

    Topics: Animals; Behavior, Animal; Biphenyl Compounds; Drug Interactions; Injections, Spinal; Male; Mice; Peptide Fragments; Receptors, Neurokinin-1; Spinal Cord; Substance P

1999
Phosphorylation of TRPV1 by neurokinin-1 receptor agonist exaggerates the capsaicin-mediated substance P release from cultured rat dorsal root ganglion neurons.
    Neuropharmacology, 2008, Volume: 55, Issue:8

    Topics: Analysis of Variance; Animals; Biphenyl Compounds; Capsaicin; Cells, Cultured; Enzyme Inhibitors; Ganglia, Spinal; Neurons; Peptide Fragments; Phosphorylation; Rats; Rats, Wistar; Receptors, Neurokinin-1; Substance P; Time Factors; TRPV Cation Channels

2008