Page last updated: 2024-09-03

gr 73632 and aprepitant

gr 73632 has been researched along with aprepitant in 3 studies

Compound Research Comparison

Studies
(gr 73632)
Trials
(gr 73632)
Recent Studies (post-2010)
(gr 73632)
Studies
(aprepitant)
Trials
(aprepitant)
Recent Studies (post-2010) (aprepitant)
7719769229521

Protein Interaction Comparison

ProteinTaxonomygr 73632 (IC50)aprepitant (IC50)
Cytochrome P450 3A4Homo sapiens (human)0.046
Substance-P receptorHomo sapiens (human)0.0002
Substance-P receptorMeriones unguiculatus (Mongolian gerbil)0.0001

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ballard, TM; Haman, M; Higgins, GA; Woolley, ML1
Asai, H; Ishii, T; Kiuchi, S; Nagasaki, M; Okamoto, M; Saito, A; Taniguchi, H; Watanabe, Y1
Bettelini, L; Corsi, M; Costantini, VJ; Dünstl, G; Gerrard, P; Zonzini, L1

Other Studies

3 other study(ies) available for gr 73632 and aprepitant

ArticleYear
Investigating the effect of bilateral amygdala lesions on fear conditioning and social interaction in the male Mongolian gerbil.
    Brain research, 2006, Mar-17, Volume: 1078, Issue:1

    Topics: Amygdala; Analysis of Variance; Animals; Aprepitant; Behavior, Animal; Conditioning, Classical; Dose-Response Relationship, Drug; Drug Interactions; Fear; Gerbillinae; Ibotenic Acid; Immobility Response, Tonic; Interpersonal Relations; Male; Morpholines; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Substance P

2006
Pharmacological characterization of T-2328, 2-fluoro-4'-methoxy-3'-[[[(2S,3S)-2-phenyl-3-piperidinyl]amino]methyl]-[1,1'-biphenyl]-4-carbonitrile dihydrochloride, as a brain-penetrating antagonist of tachykinin NK1 receptor.
    Journal of pharmacological sciences, 2008, Volume: 106, Issue:1

    Topics: Animals; Antiemetics; Antineoplastic Agents; Aprepitant; Binding Sites; Brain; Cell Line, Tumor; CHO Cells; Cisplatin; Cricetinae; Cricetulus; Disease Models, Animal; Dose-Response Relationship, Drug; Ferrets; Gerbillinae; Humans; Kinetics; Male; Morpholines; Motor Activity; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Receptors, Neurokinin-1; Substance P; Transfection; Vomiting

2008
The NK1 receptor antagonist aprepitant attenuates NK1 agonist-induced scratching behaviour in the gerbil after intra-dermal, topical or oral administration.
    Experimental dermatology, 2015, Volume: 24, Issue:4

    Topics: Administration, Oral; Administration, Topical; Animals; Antipruritics; Aprepitant; Disease Models, Animal; Drug Evaluation, Preclinical; Gerbillinae; Humans; Injections, Intradermal; Morpholines; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Pruritus; Receptors, Neurokinin-1; Substance P

2015