Page last updated: 2024-09-03

es 242-1 and ketamine

es 242-1 has been researched along with ketamine in 1 studies

*Ketamine: A cyclohexanone derivative used for induction of anesthesia. Its mechanism of action is not well understood, but ketamine can block NMDA receptors (RECEPTORS, N-METHYL-D-ASPARTATE) and may interact with sigma receptors. [MeSH]

*Ketamine: A cyclohexanone derivative used for induction of anesthesia. Its mechanism of action is not well understood, but ketamine can block NMDA receptors (RECEPTORS, N-METHYL-D-ASPARTATE) and may interact with sigma receptors. [MeSH]

Compound Research Comparison

Studies
(es 242-1)
Trials
(es 242-1)
Recent Studies (post-2010)
(es 242-1)
Studies
(ketamine)
Trials
(ketamine)
Recent Studies (post-2010) (ketamine)
50015,0292,3216,678

Protein Interaction Comparison

ProteinTaxonomyes 242-1 (IC50)ketamine (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)4.216
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)4.216
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)5.02
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)5.02
Glutamate receptor ionotropic, NMDA 1Homo sapiens (human)3.7762
Glutamate receptor ionotropic, NMDA 2AHomo sapiens (human)3.5563
Glutamate receptor ionotropic, NMDA 2BHomo sapiens (human)4.1059
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)5.02
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)5.02
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)5.02

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ando, K; Kawamoto, I; Matsuda, Y; Sano, H; Toki, S; Yoshida, M1

Other Studies

1 other study(ies) available for es 242-1 and ketamine

ArticleYear
ES-242-1, a novel compound from Verticillium sp., binds to a site on N-methyl-D-aspartate receptor that is coupled to the channel domain.
    The Journal of antibiotics, 1992, Volume: 45, Issue:1

    Topics: Animals; Bacteria; Binding, Competitive; Centrifugation; Chromatography, High Pressure Liquid; Chromatography, Thin Layer; Culture Techniques; Dizocilpine Maleate; Dose-Response Relationship, Drug; Fermentation; Kainic Acid; Ketamine; Mitosporic Fungi; Molecular Structure; Phencyclidine; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Soil Microbiology; Solubility; Synaptic Membranes

1992