Page last updated: 2024-09-05

dapivirine and uc-781

dapivirine has been researched along with uc-781 in 7 studies

Compound Research Comparison

Studies
(dapivirine)
Trials
(dapivirine)
Recent Studies (post-2010)
(dapivirine)
Studies
(uc-781)
Trials
(uc-781)
Recent Studies (post-2010) (uc-781)
1966416070621

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (42.86)29.6817
2010's4 (57.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anton, P; Cranage, M; Herrera, C; McGowan, I; Shattock, RJ1
Anderson, KS; Bollini, M; Cisneros, JA; Jorgensen, WL; Spasov, KA1
Ariën, KK; Augustyns, K; Cos, P; Dirié, B; Heeres, J; Joossens, J; Lewi, PJ; Lyssens, S; Maes, L; Michiels, J; Van der Veken, P; Vanham, G; Venkatraj, M1
Balzarini, J; Fransen, K; Janssen, P; Kestens, L; Lewi, P; Michiels, J; Van Herrewege, Y; Van Roey, J; Vanham, G1
Cara, A; Costi, R; Di Santo, R; Hazuda, D; Lewi, P; Terrazas-Aranda, K; Van Herrewege, Y; Vanham, G1
Moncla, BJ; Pryke, K; Rohan, LC; Yang, H1
Szpir, M; Van Damme, L1

Reviews

1 review(s) available for dapivirine and uc-781

ArticleYear
Current status of topical antiretroviral chemoprophylaxis.
    Current opinion in HIV and AIDS, 2012, Volume: 7, Issue:6

    Topics: Adenine; Administration, Intravaginal; Administration, Topical; Anilides; Anti-HIV Agents; Chemoprevention; Clinical Trials, Phase II as Topic; Female; Furans; HIV Infections; Humans; Organophosphonates; Pyrimidines; Tenofovir; Thioamides; Treatment Outcome

2012

Other Studies

6 other study(ies) available for dapivirine and uc-781

ArticleYear
Reverse transcriptase inhibitors as potential colorectal microbicides.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:5

    Topics: Adenine; Anilides; Anti-HIV Agents; Anti-Infective Agents, Local; Colon; Drug Resistance, Viral; Furans; HIV Infections; HIV-1; Humans; Leukocytes, Mononuclear; Organophosphonates; Pyrimidines; Rectum; Reverse Transcriptase Inhibitors; Tenofovir; Thioamides; Tissue Culture Techniques; Virus Replication

2009
Optimization of diarylazines as anti-HIV agents with dramatically enhanced solubility.
    Bioorganic & medicinal chemistry letters, 2013, Sep-15, Volume: 23, Issue:18

    Topics: Anti-HIV Agents; Cell Line, Transformed; Cell Proliferation; Dose-Response Relationship, Drug; HIV-1; Humans; Hydrazines; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Solubility; Structure-Activity Relationship

2013
From human immunodeficiency virus non-nucleoside reverse transcriptase inhibitors to potent and selective antitrypanosomal compounds.
    Bioorganic & medicinal chemistry, 2014, Oct-01, Volume: 22, Issue:19

    Topics: Anti-HIV Agents; Cell Line; Cell Survival; Dose-Response Relationship, Drug; HIV Reverse Transcriptase; HIV-1; Humans; Microbial Sensitivity Tests; Molecular Structure; Parasitic Sensitivity Tests; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense

2014
In vitro evaluation of nonnucleoside reverse transcriptase inhibitors UC-781 and TMC120-R147681 as human immunodeficiency virus microbicides.
    Antimicrobial agents and chemotherapy, 2004, Volume: 48, Issue:1

    Topics: Anilides; Anti-HIV Agents; CD4-Positive T-Lymphocytes; Cell-Free System; Cells, Cultured; Coculture Techniques; Dendritic Cells; Enzyme-Linked Immunosorbent Assay; Furans; HIV Infections; HIV-1; Humans; Pyrimidines; Reverse Transcriptase Inhibitors; Thioamides

2004
Human immunodeficiency virus type 1 (HIV-1) integration: a potential target for microbicides to prevent cell-free or cell-associated HIV-1 infection.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:7

    Topics: Anilides; Anti-HIV Agents; CD4-Positive T-Lymphocytes; Cell Line; Cells, Cultured; Coculture Techniques; Dendritic Cells; Female; Furans; HIV Infections; HIV Integrase Inhibitors; HIV-1; Humans; Male; Naphthyridines; Pyrimidines; Reverse Transcriptase Inhibitors; Thioamides; Virus Integration

2008
Testing of viscous anti-HIV microbicides using Lactobacillus.
    Journal of microbiological methods, 2012, Volume: 88, Issue:2

    Topics: Adenine; Anilides; Animals; Anti-HIV Agents; Anti-Infective Agents, Local; Cattle; Chemokine CCL5; Colony Count, Microbial; Excipients; Female; Furans; Humans; Lactobacillus; Microbial Sensitivity Tests; Microbial Viability; Organophosphonates; Pyrimidines; Serum Albumin, Bovine; Tenofovir; Thioamides; Vagina; Viscosity

2012