dapi and diminazene

dapi has been researched along with diminazene in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.11)18.7374
1990's8 (44.44)18.2507
2000's5 (27.78)29.6817
2010's3 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clercq, ED; Dann, O1
Huang, TL; Mayence, A; Vanden Eynde, JJ1
Kawanishi, S; Yamamoto, K1
Arakawa, A; Chitambo, H1
Balber, AE; Frommel, TO1
Breslauer, KJ; Pilch, DS1
Chen, AY; Gatto, B; Liu, LF; Yu, C1
Alvarez Bujidos, ML; Balaña Fouce, R; Cubria, JC; Ordoñez, D; Reguera, R1
Bailly, C; Colson, P; Houssier, C1
Bailly, C; Colson, P; Hamy, F; Houssier, C1
Brazil-Zison, M; Dickerson, RE; Filipowsky, ME; Kopka, ML; Lown, JW1
Cho, A; Eliseev, AV; Ochoa Lara, KL; Yatsimirsky, AK1
Neidle, S1
De Pauw, E; Gabelica, V; Houssier, C; Rosu, F1
Edwards, TE; Sigurdsson, ST1
Nguyen, B; Wilson, WD1
Chen, X; Dürrnagel, S; Li, M; MacDonald, JF; Orser, BA; Qiu, L; Xiong, ZG1
Blair, SD; Chamot, D; Dymowska, AK; Goss, GG; Schultz, AG1

Reviews

2 review(s) available for dapi and diminazene

ArticleYear
Some non-conventional biomolecular targets for diamidines. A short survey.
    Bioorganic & medicinal chemistry, 2014, Apr-01, Volume: 22, Issue:7

    Topics: Amidines; Animals; Diabetes Mellitus, Type 2; DNA; Enzymes; Humans; Hypertension; Ion Channels; Myotonic Dystrophy; Neoplasms; Neurodegenerative Diseases; Proteins; RNA; Thrombosis

2014
DNA minor-groove recognition by small molecules.
    Natural product reports, 2001, Volume: 18, Issue:3

    Topics: Base Sequence; Benzimidazoles; Bisbenzimidazole; Crystallography, X-Ray; Diminazene; Distamycins; DNA; DNA Probes; DNA-Binding Proteins; Indoles; Ligands; Molecular Conformation; Molecular Structure; Netropsin; Nylons; Oligodeoxyribonucleotides; Sequence Analysis, DNA

2001

Other Studies

16 other study(ies) available for dapi and diminazene

ArticleYear
Diaryl amidine derivatives as oncornaviral DNA polymerase inhibitors.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:7

    Topics: Amidines; Animals; Antineoplastic Agents; Kinetics; Leukemia, Experimental; Mice; Moloney murine leukemia virus; Retroviridae; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Tilorone

1980
Enhancement and alteration of bleomycin-catalyzed site-specific DNA cleavage by distamycin A and some minor groove binders.
    Biochemical and biophysical research communications, 1992, Feb-28, Volume: 183, Issue:1

    Topics: Base Sequence; Bisbenzimidazole; Bleomycin; Diminazene; Distamycins; DNA; DNA Damage; Indoles; Molecular Sequence Data; Nucleic Acid Conformation

1992
Trypanosoma congolense: the use of 4,6-diamidino-2-phenylindole (DAPI) in the akinetoplastic induction sensitivity test.
    The Journal of veterinary medical science, 1992, Volume: 54, Issue:4

    Topics: Animals; Diminazene; Drug Resistance; Fluorescent Dyes; Indoles; Mice; Phenanthridines; Staining and Labeling; Trypanocidal Agents; Trypanosoma congolense

1992
Flow cytofluorimetric analysis of drug accumulation by multidrug-resistant Trypanosoma brucei brucei and T. b. rhodesiense.
    Molecular and biochemical parasitology, 1987, Volume: 26, Issue:1-2

    Topics: Acriflavine; Animals; Benzimidazoles; Diminazene; Drug Resistance; Ethidium; Flow Cytometry; Fluorescent Dyes; Humans; Indoles; Melarsoprol; Mice; Pentamidine; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei

1987
Ligand-induced formation of nucleic acid triple helices.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Sep-27, Volume: 91, Issue:20

    Topics: Circular Dichroism; Diminazene; DNA; Ethidium; Fluorescent Dyes; Indoles; Netropsin; Nucleic Acid Conformation; Poly A; Poly T; RNA; Spectrophotometry; Thermodynamics

1994
DNA minor groove-binding ligands: a different class of mammalian DNA topoisomerase I inhibitors.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Sep-01, Volume: 90, Issue:17

    Topics: Animals; Base Sequence; Benzimidazoles; Bisbenzimidazole; Cattle; Diminazene; Distamycins; DNA; DNA Topoisomerases, Type I; DNA Topoisomerases, Type II; Indoles; Intercalating Agents; Kinetics; Ligands; Molecular Sequence Data; Oligodeoxyribonucleotides; Structure-Activity Relationship; Thymus Gland; Topoisomerase I Inhibitors

1993
Putrescine uptake inhibition by aromatic diamidines in Leishmania infantum promastigotes.
    Biochemical pharmacology, 1994, May-18, Volume: 47, Issue:10

    Topics: Amidines; Animals; Diminazene; Indoles; Kinetics; Leishmania infantum; Pentamidine; Putrescine; Stilbamidines

1994
Use of electric linear dichroism and competition experiments with intercalating drugs to investigate the mode of binding of Hoechst 33258, berenil and DAPI to GC sequences.
    Journal of biomolecular structure & dynamics, 1995, Volume: 13, Issue:2

    Topics: Base Sequence; Binding, Competitive; Bisbenzimidazole; Diminazene; Indoles; Intercalating Agents; Molecular Sequence Data; Molecular Structure; Poly dA-dT; Polydeoxyribonucleotides; Spectrum Analysis

1995
The binding mode of drugs to the TAR RNA of HIV-1 studied by electric linear dichroism.
    Nucleic acids research, 1996, Apr-15, Volume: 24, Issue:8

    Topics: Antiviral Agents; Bisbenzimidazole; Diminazene; Ethidium; HIV Long Terminal Repeat; HIV-1; Humans; Indoles; Intercalating Agents; Molecular Sequence Data; Netropsin; Nucleic Acid Conformation; Proflavine; RNA, Viral; Spectrum Analysis

1996
Linked lexitropsins and the in vitro inhibition of HIV-1 reverse transcriptase RNA-directed DNA polymerization: a novel induced-fit of 3,5 m-pyridyl bisdistamycin to enzyme-associated template-primer.
    Biochemistry, 1996, Dec-03, Volume: 35, Issue:48

    Topics: Antiviral Agents; Bisbenzimidazole; Diminazene; Distamycins; DNA Polymerase I; DNA Primers; Electrophoresis, Polyacrylamide Gel; HIV Reverse Transcriptase; Indoles; Kinetics; Models, Molecular; Netropsin; RNA-Directed DNA Polymerase; Templates, Genetic; Thymine Nucleotides

1996
Phosphatase-triggered guest release from a cyclodextrin complex.
    Organic letters, 2000, Jun-15, Volume: 2, Issue:12

    Topics: Alkaline Phosphatase; Antineoplastic Agents; Binding Sites; Cyclodextrins; Diminazene; Half-Life; Hydrolysis; Indoles; Intercalating Agents; Ligands; Magnetic Resonance Spectroscopy; Models, Chemical; Models, Molecular; Molecular Mimicry; Phosphorus Compounds; Phosphorylation; Titrimetry

2000
Determination of affinity, stoichiometry and sequence selectivity of minor groove binder complexes with double-stranded oligodeoxynucleotides by electrospray ionization mass spectrometry.
    Nucleic acids research, 2002, Aug-15, Volume: 30, Issue:16

    Topics: Base Sequence; Benzimidazoles; Bisbenzimidazole; Circular Dichroism; Diminazene; DNA; Indoles; Nucleic Acid Conformation; Oligodeoxyribonucleotides; Spectrometry, Fluorescence; Spectrometry, Mass, Electrospray Ionization; Substrate Specificity; Thermodynamics; Titrimetry

2002
Electron paramagnetic resonance dynamic signatures of TAR RNA-small molecule complexes provide insight into RNA structure and recognition.
    Biochemistry, 2002, Dec-17, Volume: 41, Issue:50

    Topics: Acridines; Anti-HIV Agents; Binding, Competitive; Bisbenzimidazole; Diminazene; Electron Spin Resonance Spectroscopy; Fluorescent Dyes; Framycetin; Guanidines; HIV Long Terminal Repeat; Indoles; Macromolecular Substances; RNA, Viral; Spin Labels; Structure-Activity Relationship; Thermodynamics

2002
The effects of hairpin loops on ligand-DNA interactions.
    The journal of physical chemistry. B, 2009, Oct-29, Volume: 113, Issue:43

    Topics: Base Sequence; Diminazene; DNA; Indoles; Ligands; Netropsin; Surface Plasmon Resonance

2009
Diarylamidines: high potency inhibitors of acid-sensing ion channels.
    Neuropharmacology, 2010, Volume: 58, Issue:7

    Topics: Acid Sensing Ion Channels; Amidines; Animals; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Diminazene; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Hippocampus; Indoles; Mice; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Oocytes; Pentamidine; Sodium Channels; Stilbamidines; Xenopus laevis

2010
Acid-sensing ion channels are involved in epithelial Na+ uptake in the rainbow trout Oncorhynchus mykiss.
    American journal of physiology. Cell physiology, 2014, Aug-01, Volume: 307, Issue:3

    Topics: Acid Sensing Ion Channel Blockers; Acid Sensing Ion Channels; Amiloride; Amino Acid Sequence; Animals; Antibodies; Biological Transport, Active; Cloning, Molecular; Diminazene; Gills; Indoles; Oncorhynchus mykiss; Sequence Alignment; Sodium; Sodium-Potassium-Exchanging ATPase; Trypanocidal Agents

2014