Page last updated: 2024-09-04

cyc 202 and thiazoles

cyc 202 has been researched along with thiazoles in 10 studies

Compound Research Comparison

Studies
(cyc 202)
Trials
(cyc 202)
Recent Studies (post-2010)
(cyc 202)
Studies
(thiazoles)
Trials
(thiazoles)
Recent Studies (post-2010) (thiazoles)
979739333,1792,10012,330

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (50.00)29.6817
2010's4 (40.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Agbottah, E; Barnett, A; de La Fuente, C; Gianella-Borradori, A; Kashanchi, F; Nekhai, S; Pumfery, A1
Cress, WD; Freeman, SN; Ma, Y1
Blagden, S; de Bono, J1
Kellogg, DR; McCusker, D; Royou, A; Sullivan, W1
Chen, R; Chubb, S; Fox, JA; Gandhi, V; Hawtin, RE; Keating, MJ; Plunkett, W; Wierda, WG1
Hu, LY; Li, X; Wu, ZH; Xu, DQ1
Karess, RE; Menant, A1
Crews, LA; Gonzales, T; Kouznetsova, VL; Masliah, E; Overk, CR; Patrick, C; Paulino, A; Price, D; Rockenstein, E; Stocking, E; Tsigelny, IF; Wrasidlo, W1
Giordano, A; Morales, F1
Boucher, J; Harms, M; Maurer, S1

Reviews

3 review(s) available for cyc 202 and thiazoles

ArticleYear
Drugging cell cycle kinases in cancer therapy.
    Current drug targets, 2005, Volume: 6, Issue:3

    Topics: Adenosine Triphosphate; Animals; Antineoplastic Agents; Binding Sites; Cyclin-Dependent Kinases; Flavonoids; Humans; Neoplasms; Oxazoles; Piperidines; Protein Kinase Inhibitors; Purines; Roscovitine; Staurosporine; Sulfonamides; Thiazoles

2005
Overview of CDK9 as a target in cancer research.
    Cell cycle (Georgetown, Tex.), 2016, Volume: 15, Issue:4

    Topics: Bridged Bicyclo Compounds, Heterocyclic; Cell Cycle; Cyclic N-Oxides; Cyclin-Dependent Kinase 9; Flavonoids; Humans; Indolizines; Molecular Targeted Therapy; Neoplasms; Oxazoles; Piperidines; Protein Kinase Inhibitors; Purines; Pyrazoles; Pyridinium Compounds; Roscovitine; Thiazoles; Urea

2016
The colorful versatility of adipocytes: white-to-brown transdifferentiation and its therapeutic potential in humans.
    The FEBS journal, 2021, Volume: 288, Issue:12

    Topics: Acetanilides; Adipocytes, Beige; Adipocytes, Brown; Adipocytes, White; Adipose Tissue, Brown; Adipose Tissue, White; Animals; Cell Lineage; Cell Transdifferentiation; Diabetes Mellitus; Drugs, Investigational; Energy Metabolism; Humans; Imatinib Mesylate; Obesity; Roscovitine; Thermogenesis; Thiazoles

2021

Other Studies

7 other study(ies) available for cyc 202 and thiazoles

ArticleYear
Antiviral activity of CYC202 in HIV-1-infected cells.
    The Journal of biological chemistry, 2005, Jan-28, Volume: 280, Issue:4

    Topics: Antiretroviral Therapy, Highly Active; Antiviral Agents; Apoptosis; CDC2-CDC28 Kinases; Cell Cycle; Chromatin Immunoprecipitation; Cyclin E; Cyclin-Dependent Kinase 2; DNA Fragmentation; DNA, Viral; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Escherichia coli; Flow Cytometry; Genome, Viral; HIV-1; Humans; Immunoblotting; Inhibitory Concentration 50; Leukocytes, Mononuclear; Monocytes; Mutation; Phosphorylation; Purines; RNA Interference; RNA, Small Interfering; Roscovitine; Tetrazolium Salts; Thiazoles; Time Factors; Transcription, Genetic

2005
E2F4 deficiency promotes drug-induced apoptosis.
    Cancer biology & therapy, 2004, Volume: 3, Issue:12

    Topics: Animals; Antineoplastic Agents; Apoptosis; Breast Neoplasms; Carcinoma, Non-Small-Cell Lung; Cell Cycle Proteins; DNA-Binding Proteins; E2F Transcription Factors; E2F1 Transcription Factor; E2F4 Transcription Factor; Fibroblasts; Flavonoids; Humans; Lung Neoplasms; Mice; Mice, Knockout; Oxazoles; Piperidines; Protein Kinase Inhibitors; Purines; RNA, Small Interfering; Roscovitine; Thiazoles; Transcription Factors; Tumor Cells, Cultured

2004
Grapes(Chk1) prevents nuclear CDK1 activation by delaying cyclin B nuclear accumulation.
    The Journal of cell biology, 2008, Oct-06, Volume: 183, Issue:1

    Topics: Active Transport, Cell Nucleus; Animals; Aphidicolin; CDC2 Protein Kinase; Cell Cycle; Cell Cycle Proteins; Cell Nucleus; Cell Nucleus Division; Checkpoint Kinase 1; Cyclin B; Cycloheximide; Cytokinesis; Cytoplasm; Drosophila melanogaster; Drosophila Proteins; Embryo, Nonmammalian; Kinetochores; Mitosis; Mutation; Nuclear Envelope; Nuclear Proteins; Protein Kinase Inhibitors; Protein Kinases; Protein-Tyrosine Kinases; Purines; Quinolines; Recombinant Proteins; Roscovitine; Spindle Apparatus; Thiazoles

2008
Mechanism of action of SNS-032, a novel cyclin-dependent kinase inhibitor, in chronic lymphocytic leukemia.
    Blood, 2009, May-07, Volume: 113, Issue:19

    Topics: Adult; Aged; Aged, 80 and over; Apoptosis; Caspases; Cyclin-Dependent Kinases; Female; Flavonoids; Humans; Immunoblotting; Leukemia, Lymphocytic, Chronic, B-Cell; Lymphocytes; Male; Membrane Potential, Mitochondrial; Middle Aged; Myeloid Cell Leukemia Sequence 1 Protein; Oxazoles; Phosphorylation; Piperidines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-bcl-2; Purines; RNA Polymerase II; RNA, Neoplasm; Roscovitine; Thiazoles; Transcription, Genetic; X-Linked Inhibitor of Apoptosis Protein

2009
A cell-based assay for screening spindle checkpoint inhibitors.
    Assay and drug development technologies, 2012, Volume: 10, Issue:4

    Topics: Antineoplastic Agents; Aurora Kinases; Blotting, Western; Cell Cycle; Cell Cycle Checkpoints; Cell Line; Coloring Agents; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Fluorescent Antibody Technique; HeLa Cells; High-Throughput Screening Assays; Humans; Mitotic Index; Nocodazole; Protein Serine-Threonine Kinases; Purines; Roscovitine; Spindle Apparatus; Tetrazolium Salts; Thiazoles

2012
Inducing "cytokinesis" without mitosis in unfertilized Drosophila eggs.
    Cell cycle (Georgetown, Tex.), 2012, Aug-01, Volume: 11, Issue:15

    Topics: Actins; Animals; CDC2 Protein Kinase; Cell Division; Cells, Cultured; Contractile Proteins; Cyclin B; Cytokinesis; Drosophila; Drosophila Proteins; Embryo, Nonmammalian; GTPase-Activating Proteins; Microtubule-Associated Proteins; Mitosis; Myosins; Ovum; Protein Kinase Inhibitors; Purines; Quinolines; rhoA GTP-Binding Protein; Roscovitine; Spindle Apparatus; Thiazoles

2012
Neuroprotective effects of the anti-cancer drug sunitinib in models of HIV neurotoxicity suggests potential for the treatment of neurodegenerative disorders.
    British journal of pharmacology, 2014, Volume: 171, Issue:24

    Topics: AIDS Dementia Complex; Animals; Antineoplastic Agents; Cyclin-Dependent Kinase 5; Dasatinib; Erlotinib Hydrochloride; Flavonoids; HIV Envelope Protein gp120; In Vitro Techniques; Indoles; Lapatinib; Mice; Mice, Transgenic; Neurodegenerative Diseases; Neurons; Neuroprotective Agents; Protein Kinase Inhibitors; Purines; Pyrimidines; Pyrroles; Quinazolines; Rats; Roscovitine; Sunitinib; Thiazoles

2014