clonidine and eedq

clonidine has been researched along with eedq in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19902 (9.52)18.7374
1990's18 (85.71)18.2507
2000's1 (4.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Nowak, G; Pilc, A; Zak, J1
Barturen, F; Garcia-Sevilla, JA1
Engberg, G; Eriksson, E1
Agneter, E; Drobny, H; Singer, EA1
Takano, Y; Yaksh, TL1
Agnati, L; Fredholm, B; Fuxe, K; Härfstrand, A1
Enna, SJ; Nomura, S; Pilc, A; Vetulani, J1
García-Sevilla, JA; Pineda, J; Ruiz-Ortega, JA; Ugedo, L2
Goiny, M; Herrera-Marschitz, M; Meana, JJ1
Gabilondo, AM; García-Sevilla, JA1
Badia, A; Giraldo, J; Sallés, J1
Oriowo, MA1
Fröhlich, R; Illes, P; Szabo, B1
Badia, A; Giraldo, J; Sallés, J; Vila, E1
Ruiz-Ortega, JA; Ugedo, L1
Pineda, J; Ruiz-Ortega, JA; Ugedo, L1
Agneter, E; Feuerstein, TJ; Sauermann, W; Singer, EA1
García-Sevilla, JA; Pineda, J; Ugedo, L1
Esteban, S; García-Sevilla, JA; Sastre-Coll, A1
Busquets, X; García-Sevilla, JA; Miralles, A; Ribas, C1

Other Studies

21 other study(ies) available for clonidine and eedq

ArticleYear
N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline, an irreversible receptor inactivator, as a tool for measurement of alpha 2-adrenoceptor occupancy in vivo.
    European journal of pharmacology, 1992, Feb-25, Volume: 212, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Clonidine; Male; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1992
Long term treatment with desipramine increases the turnover of alpha 2-adrenoceptors in the rat brain.
    Molecular pharmacology, 1992, Volume: 42, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Clonidine; Desipramine; Male; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha

1992
Effects of alpha 2-adrenoceptor agonists on locus coeruleus firing rate and brain noradrenaline turnover in N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ)-treated rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:5

    Topics: Animals; Brain; Clonidine; Dose-Response Relationship, Drug; Electrodes; Guanfacine; In Vitro Techniques; Locus Coeruleus; Male; Norepinephrine; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1991
Estimation of agonist dissociation constants at central presynaptic alpha-2 autoreceptors in the absence of autoinhibition.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Brain; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Male; Norepinephrine; Quinolines; Quinoxalines; Rats; Receptors, Adrenergic, alpha

1991
Relative efficacy of spinal alpha-2 agonists, dexmedetomidine, clonidine and ST-91, determined in vivo by using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline, an irreversible antagonist.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Injections, Spinal; Male; Medetomidine; Morphine; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Spinal Cord

1991
Reciprocal interactions between alpha 2-adrenoceptor agonist and neuropeptide Y binding sites in the nucleus tractus solitarius of the rat. A biochemic and autoradiographic analysis.
    Journal of neural transmission, 1989, Volume: 75, Issue:2

    Topics: Animals; Binding, Competitive; Clonidine; Dioxanes; Idazoxan; Kinetics; Male; Medulla Oblongata; Neuropeptide Y; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Neuropeptide Y; Receptors, Neurotransmitter; Subcellular Fractions

1989
An in vivo procedure for the selective inactivation of rat brain cerebral cortical alpha-adrenoceptors using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
    Brain research, 1989, Jul-24, Volume: 493, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Cell Membrane; Cerebral Cortex; Clonidine; Cyclic AMP; Dihydroalprenolol; Inositol Phosphates; Isoproterenol; Male; Norepinephrine; Prazosin; Quinolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1989
The stimulatory effect of clonidine through imidazoline receptors on locus coeruleus noradrenergic neurones is mediated by excitatory amino acids and modulated by serotonin.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: Adrenergic alpha-Antagonists; alpha-Methyltyrosine; Animals; Catecholamines; Clonidine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Amino Acids; Extracellular Space; Imidazoline Receptors; Kynurenic Acid; Locus Coeruleus; Male; Methyltyrosines; Neurons; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Serotonin; Sympathetic Nervous System; Sympatholytics; Tyrosine 3-Monooxygenase

1995
In vivo modulation of norepinephrine and glutamate release through imidazoline receptors in the rat central nervous system.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Central Nervous System; Clonidine; Dioxanes; Glutamic Acid; Idazoxan; Imidazoline Receptors; Norepinephrine; Quinolines; Rats; Receptors, Drug

1995
The stimulatory effect of clonidine on locus coeruleus noradrenergic neurons through imidazoline receptors is modulated by excitatory amino acids.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-Antagonists; alpha-Methyltyrosine; Animals; Clonidine; Excitatory Amino Acids; Fenclonine; Imidazoline Receptors; Locus Coeruleus; Male; Methyltyrosines; Neurons; Norepinephrine; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reserpine

1995
Spontaneous withdrawal from long-term treatment with morphine accelerates the turnover of alpha 2-adrenoceptors in the rat brain: up-regulation of receptors associated with increased receptor appearance.
    Journal of neurochemistry, 1995, Volume: 64, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Clonidine; Male; Morphine; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Substance Withdrawal Syndrome; Time Factors; Up-Regulation

1995
Analysis of agonism at functional prejunctional alpha 2-adrenoceptors of rat vas deferens using operational and null approaches.
    European journal of pharmacology, 1994, Jun-13, Volume: 258, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Algorithms; Alkylation; Animals; Clonidine; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Neuromuscular Junction; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Vas Deferens

1994
The prejunctional inhibitory effect of alpha-methylnoradrenaline in the rat vas deferens is not mediated via alpha 2-adrenoceptors.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Benzazepines; Clonidine; Dioxanes; Electric Stimulation; Idazoxan; Imidazoles; Isometric Contraction; Male; Neuromuscular Junction; Nordefrin; Phenoxybenzamine; Phentolamine; Quinolines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Adrenergic, alpha-2; Vas Deferens; Vasoconstrictor Agents; Yohimbine

1995
No evidence for functional imidazoline receptors on locus coeruleus neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Locus Coeruleus; Male; Microelectrodes; Neurons; Oxazoles; Quinolines; Rats; Rats, Wistar; Receptors, Drug; Rilmenidine

1996
Modelling the changes induced by chronic desipramine treatment on the factors governing the agonism at prejunctional alpha 2-adrenoceptors.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: Adrenergic Uptake Inhibitors; Animals; Clonidine; Desipramine; Dose-Response Relationship, Drug; Logistic Models; Male; Models, Biological; Muscle, Smooth; Quinolines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Vas Deferens; Xylazine

1996
The stimulatory effect of clonidine on locus coeruleus neurons of rats with inactivated alpha 2-adrenoceptors: involvement of imidazoline receptors located in the nucleus paragigantocellularis.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Clonidine; Electrophysiology; Imidazoline Receptors; Locus Coeruleus; Male; Medulla Oblongata; Microinjections; Neurons; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Drug

1997
Receptor reserve and turnover of alpha-2 adrenoceptors that mediate the clonidine-induced inhibition of rat locus coeruleus neurons in vivo.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Locus Coeruleus; Male; Neurons; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1997
The slope parameter of concentration-response curves used as a touchstone for the existence of spare receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Brimonidine Tartrate; Cerebral Cortex; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Models, Theoretical; Norepinephrine; Quinolines; Quinoxalines; Rats

1997
Enhanced alpha2A-autoreceptor reserve for clonidine induced by reserpine and cholinomimetic agents in the rat vas deferens.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Male; Muscle Contraction; Muscle, Smooth; Neostigmine; Parasympathomimetics; Pilocarpine; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reserpine; Vas Deferens

1997
Effects of imidazoline drugs on tyrosine and tryptophan hydroxylase activity in rat brain in vivo.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Brain; Clonidine; Dihydroxyphenylalanine; Imidazoles; Male; Quinolines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Tryptophan Hydroxylase; Tyrosine 3-Monooxygenase

1999
Brain alpha(2)-adrenoceptors in monoamine-depleted rats: increased receptor density, G coupling proteins, receptor turnover and receptor mRNA.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Brain; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Gene Expression Regulation; GTP-Binding Proteins; Idazoxan; Male; Membranes; Norepinephrine; Quinolines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reserpine; RNA, Messenger; Tritium

2001