cimetidine and n-methylnicotinamide

cimetidine has been researched along with n-methylnicotinamide in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19901 (4.55)18.7374
1990's13 (59.09)18.2507
2000's7 (31.82)29.6817
2010's1 (4.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dresser, MJ; Giacomini, KM; Gray, AT; Terashita, S; Yost, SC; Zhang, L1
Babbitt, PC; Chun, JK; Dresser, MJ; Giacomini, KM; Zhang, L1
Fei, YJ; Ganapathy, V; Kekuda, R; Leibach, FH; Prasad, PD; Wang, H; Wu, X1
Giacomini, KM; Schaner, ME; Zhang, L1
Inui, KI; Masuda, S; Okuda, M; Saito, H; Urakami, Y1
Inui, K; Okuda, M; Saito, H; Urakami, Y1
Nezu, J; Oku, A; Sai, Y; Sakamoto, K; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Nezu, JI; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Conway, SJ; Ganapathy, ME; Ganapathy, V; Huang, W; Kekuda, R; Leibach, FH; Wang, H; Wu, X1
Akazawa, M; Inui, K; Okuda, M; Saito, H; Urakami, Y1
Kakehi, M; Koyabu, N; Kuwano, M; Nakamura, T; Ohtani, H; Sawada, Y; Uchiumi, T1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Dutt, A; Kuo, MT; Nelson, JA; Priebe, TS; Teeter, LD1
Daley-Yates, PT; Maiza, A1
Brändle, E; Greven, J1
Acara, M; Feld, L; Fildes, R; Hasan, M; Rennick, B; Springate, J1
Chan, BS; Duggin, GG; Lazzaro, VA; Seale, JP1
Bendayan, R1
Aavula, BR; Bednarczyk, D; Mash, EA; Wright, SH1
O'Donnell, MJ; Plaumann, JS; Rheault, MR1

Other Studies

22 other study(ies) available for cimetidine and n-methylnicotinamide

ArticleYear
Cloning and functional expression of a human liver organic cation transporter.
    Molecular pharmacology, 1997, Volume: 51, Issue:6

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Humans; Liver; Membrane Proteins; Molecular Sequence Data; Oocytes; Organic Cation Transporter 1; Polymerase Chain Reaction; Rats; RNA, Messenger; Sequence Homology, Amino Acid; Species Specificity; Tissue Distribution; Xenopus laevis

1997
Cloning and functional characterization of a rat renal organic cation transporter isoform (rOCT1A).
    The Journal of biological chemistry, 1997, Jun-27, Volume: 272, Issue:26

    Topics: Amino Acid Sequence; Animals; Base Sequence; Carrier Proteins; Cloning, Molecular; Kidney; Membrane Proteins; Molecular Sequence Data; Organic Cation Transporter 1; Protein Biosynthesis; Rats; RNA, Messenger; Tetraethylammonium Compounds; Xenopus laevis

1997
Cloning and functional characterization of a potential-sensitive, polyspecific organic cation transporter (OCT3) most abundantly expressed in placenta.
    The Journal of biological chemistry, 1998, Jun-26, Volume: 273, Issue:26

    Topics: Amino Acid Sequence; Animals; Cloning, Molecular; DNA-Binding Proteins; HeLa Cells; Humans; Hydrogen-Ion Concentration; Molecular Sequence Data; Octamer Transcription Factor-3; Oocytes; Placenta; Protein Conformation; Rats; Transcription Factors; Xenopus laevis

1998
Functional characterization of an organic cation transporter (hOCT1) in a transiently transfected human cell line (HeLa).
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Carrier Proteins; Corticosterone; HeLa Cells; Humans; Membrane Proteins; Midazolam; Organic Cation Transporter 1; Permeability; Recombinant Proteins; Structure-Activity Relationship; Tetraethylammonium Compounds; Transfection

1998
Functional characteristics and membrane localization of rat multispecific organic cation transporters, OCT1 and OCT2, mediating tubular secretion of cationic drugs.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:2

    Topics: Animals; Base Sequence; Carrier Proteins; Cations; Cell Line; Cell Membrane; DNA Primers; Dogs; Kidney Tubules; Membrane Proteins; Organic Cation Transport Proteins; Organic Cation Transporter 1; Organic Cation Transporter 2; Rats; Tetraethylammonium

1998
Molecular mechanisms of organic cation transport in OCT2-expressing Xenopus oocytes.
    Biochimica et biophysica acta, 1999, Mar-04, Volume: 1417, Issue:2

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Buffers; Carrier Proteins; Cells, Cultured; Hydrogen-Ion Concentration; Levofloxacin; Membrane Proteins; Ofloxacin; Oocytes; Organic Cation Transport Proteins; Organic Cation Transporter 1; Organic Cation Transporter 2; Potassium; Rats; Tetraethylammonium; Transfection; Xenopus laevis

1999
Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2

    Topics: Animals; Biological Transport, Active; Carrier Proteins; Cell Line; Gene Expression; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Oocytes; Organic Cation Transport Proteins; Quinidine; RNA, Messenger; Symporters; Tetraethylammonium Compounds; Xenopus laevis

1999
Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Biological Transport, Active; Carnitine; Carrier Proteins; Cations; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Humans; Hydrogen-Ion Concentration; Kidney; Membrane Proteins; Organic Cation Transport Proteins; Sodium; Solute Carrier Family 22 Member 5; Stereoisomerism

1999
Structure, function, and regional distribution of the organic cation transporter OCT3 in the kidney.
    American journal of physiology. Renal physiology, 2000, Volume: 279, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; 1-Methyl-4-phenylpyridinium; Amiloride; Animals; Binding, Competitive; Carbon Radioisotopes; Cations; Cloning, Molecular; DNA-Binding Proteins; DNA, Complementary; Dopamine Agents; Exons; Gene Expression Regulation; HeLa Cells; Herbicides; Humans; In Situ Hybridization; Introns; Kidney; Mice; Niacinamide; Octamer Transcription Factor-3; Oocytes; Pigment Epithelium of Eye; RNA, Messenger; Tetraethylammonium; Transcription Factors; Tritium; Xenopus laevis

2000
cDNA cloning, functional characterization, and tissue distribution of an alternatively spliced variant of organic cation transporter hOCT2 predominantly expressed in the human kidney.
    Journal of the American Society of Nephrology : JASN, 2002, Volume: 13, Issue:7

    Topics: Alternative Splicing; Amino Acid Sequence; Base Sequence; Cations; Cell Line; Cloning, Molecular; DNA, Complementary; Genetic Variation; Humans; Kidney; Molecular Sequence Data; Organic Cation Transport Proteins; Organic Cation Transporter 2; Tetraethylammonium; Tissue Distribution; Transfection

2002
Functional characterization of mouse cation transporter mOCT2 compared with mOCT1.
    Biochemical and biophysical research communications, 2002, Aug-23, Volume: 296, Issue:3

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Base Sequence; Biological Transport; Cations; Cells, Cultured; Cloning, Molecular; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Kinetics; Membrane Potentials; Mice; Organic Cation Transport Proteins; Organic Cation Transporter 1; Organic Cation Transporter 2; Tetraethylammonium; Xenopus

2002
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Postnatal development of organic cation transport and mdr gene expression in mouse kidney.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Animals; Animals, Newborn; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cimetidine; Culture Techniques; Gene Expression; Kidney; Liver; Membrane Glycoproteins; Mice; Niacinamide; Tetraethylammonium; Tetraethylammonium Compounds

1992
Prediction of the renal clearance of cimetidine using endogenous N-1-methylnicotinamide.
    Journal of pharmacokinetics and biopharmaceutics, 1991, Volume: 19, Issue:2

    Topics: Acute Kidney Injury; Animals; Cimetidine; Glomerular Filtration Rate; Kidney; Kidney Tubules, Proximal; Male; Niacinamide; Predictive Value of Tests; Rats; Rats, Inbred Strains

1991
Transport of cimetidine across the basolateral membrane of rabbit kidney proximal tubules: characterization of transport mechanisms.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:3

    Topics: Animals; Basement Membrane; Biological Transport; Chlorides; Cimetidine; Female; Hydrogen-Ion Concentration; Intracellular Fluid; Kidney Tubules, Proximal; Male; Membrane Potentials; Niacinamide; Osmolar Concentration; Potassium; Quinine; Rabbits; Tetraethylammonium; Tetraethylammonium Compounds

1991
Relation between transport maxima and inhibition of organic cation excretion in the chicken kidney.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:2

    Topics: Animals; Binding, Competitive; Biological Transport; Cations; Chickens; Choline; Cimetidine; Kidney Tubules, Proximal; Niacinamide; Quinine; Tetraethylammonium Compounds

1987
Transport of paraquat in a renal epithelial cell line LLC-PK1.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Biological Transport; Cimetidine; Epithelium; Herbicides; Hydrogen-Ion Concentration; Kidney; LLC-PK1 Cells; Niacinamide; Paraquat; Putrescine; Swine; Temperature

1996
Interaction of dipyridamole, a nucleoside transport inhibitor, with the renal transport of organic cations by LLCPK1 cells.
    Canadian journal of physiology and pharmacology, 1997, Volume: 75, Issue:1

    Topics: Animals; Biological Transport; Cell Line; Cimetidine; Dipyridamole; Epithelium; Ions; Kidney; Kinetics; Niacinamide; Swine; Tetraethylammonium; Tetraethylammonium Compounds

1997
NBD-TMA: a novel fluorescent substrate of the peritubular organic cation transporter of renal proximal tubules.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 440, Issue:1

    Topics: Animals; Biological Transport; Carrier Proteins; Cell Survival; Cimetidine; Diffusion Chambers, Culture; Fluorescence; Fluorescent Dyes; Histamine H2 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Kidney Tubules, Proximal; Models, Biological; Niacinamide; Quaternary Ammonium Compounds; Rabbits; Reproducibility of Results; Tetraethylammonium

2000
Tetraethylammonium and nicotine transport by the Malpighian tubules of insects.
    Journal of insect physiology, 2006, Volume: 52, Issue:5

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Chromatography, Thin Layer; Cimetidine; Female; In Vitro Techniques; Insecta; Male; Malpighian Tubules; Niacinamide; Nicotine; Quinidine; Rhodnius; Tetraethylammonium; Time Factors

2006
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