Compounds > azides
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azides and prazosin

azides has been researched along with prazosin in 70 studies

Research

Studies (70)

TimeframeStudies, this research(%)All Research%
pre-199012 (17.14)18.7374
1990's28 (40.00)18.2507
2000's23 (32.86)29.6817
2010's7 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Holohan, PD; Rebbeor, J; Sokol, PP; White, KE1
Naito, M; Oh-hara, T; Sugawara, I; Tatsuta, T; Tsuruo, T1
Arceci, RJ; Bierer, BE; Stieglitz, K1
Cohen, HT; Katz, AI; Satoh, T; Takemoto, F1
Greenberger, LM; Horwitz, SB; Lisanti, CJ; Silva, JT1
Agresti, M; Mehta, ND; Safa, AR; Tamai, I; Vahabi, S1
Gindin, E; Greenberger, LM; Horwitz, SB; Yang, CP1
Cheung, DW; Fujioka, M1
Cornett, LE; Graham, RM; Sawutz, DG; Sena, LM1
Brown, RD; Insel, PA; Reece, JF; Terman, BI1
Cornett, LE; Norris, JS2
Insel, PA; Terman, BI1
Bergström, A; Wikberg, JE1
Duerden, BI; Jones, BM; Kinghorn, GR1
Graham, RM; Hess, HJ; Homcy, CJ; Seidman, CE1
Fedan, JS; Sneddon, P; Westfall, DP1
Graham, RM; Hess, HJ; Homcy, CJ1
Colby, J; Fedan, JS; Sneddon, P; Westfall, DP1
Beliveau, R; Jetté, L; Leclerc, JM; Murphy, GF1
Croop, JM; Kronauge, JF; Piwnica-Worms, D; Rao, VV1
Agresti, M; Grizzuti, K; Gros, P; Kajiji, S; Safa, AR; Talbot, F; Van Dyke-Phillips, V1
Collins, KI; Greenberger, LM; Zhang, X1
Greenberger, LM1
Chen, MF; Hwang, TL; Lau, YT; Liu, MS; Tang, C1
Canessa, LM; Felder, RA; Jose, PA; Piccio, MM; Porter, CC; Robillard, JE; Sidhu, A; Vachvanichsanong, P1
Beaulieu, E; Béliveau, R; Jetté, L; Leclerc, JM1
Chen, G; Dumontet, C; Durán, GE; Jaffrézou, JP; Lacayo, NJ; Sikic, BI; Steger, KA1
Beaulieu, E; Béliveau, R; Demeule, M; Ghitescu, L1
Ambudkar, SV; Dey, S; Gottesman, MM; Pastan, I; Ramachandra, M2
Ambudkar, SV; Cardarelli, CO; Dey, S; Gottesman, MM; Jeang, KT; Lee, CG; Pastan, I; Ramachandra, M1
Béliveau, R; Jetté, L; Murphy, GF1
Beaudet, L; Gros, P; Urbatsch, IL2
Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M1
Airan, LE; Ambudkar, SV; Germann, UA; Gottesman, MM; Hrycyna, CA; Pastan, I1
Dey, S; Gottesman, MM; Pastan, I; Shoshani, T; Zhang, S1
Dey, S; Gottesman, MM; Hafkemeyer, P; Pastan, I1
Cheng, PW; Germann, UA; Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M1
Ambudkar, SV; Dey, S; Gribar, JJ; Hrycyna, CA; Ramachandra, M1
Ambudkar, SV; Sauna, ZE1
Demmer, A; Isenberg, B; Thole, H; Tümmler, B1
Melera, PW; Song, J2
Ambudkar, SV; Anuchapreeda, S; Leechanachai, P; Limtrakul, PN; Smith, MM1
Andrus, MB; Mettath, SN; Song, C1
Minneman, KP; Pupo, AS; Uberti, MA1
Ambudkar, SV; Nandigama, K; Peng, XH; Sauna, ZE; Tekle, S1
Ambudkar, SV; Andrus, MB; Sauna, ZE; Turner, TM1
Ambudkar, SV; Anuchapreeda, S; Chearwae, W; Limtrakul, P; Nandigama, K1
Ambudkar, SV; Ferenz, M; Golin, J; Hanson, L; Keeven, J; May, L; Mehl, P; Tuma, P1
Dey, S; Ghosh, P; Maki, N; Moitra, K1
Dey, S; Maki, N1
Ambudkar, SV; Bates, SE; Robey, RW; Shukla, S1
Chattopadhyay, A; Dey, S; Fong, WF; Shen, XL; Wan, CK; Zhu, GY1
Ambudkar, SV; Chearwae, W; Limtrakul, P; Shukla, S1
Chmielewski, J; Hrycyna, CA; Pires, MM1
Abraham, I; Ambudkar, SV; Chen, ZS; El Sayed, K; Fu, LW; Jain, S; Kim, IW; Peng, XX; Shi, Z; Youssef, DT1
Ambudkar, SV; Barnett, D; Bates, SE; Finley, EM; Fojo, T; Oldham, RK; Robey, RW; Shukla, S1
Ambudkar, SV; Bauer, B; Hartz, A; Shukla, S; Ware, JA; Zaher, H1
Ambudkar, SV; Bahr, JC; Bates, SE; Di Pietro, A; Macalou, S; Obrzut, T; Polgar, O; Robey, RW; Shukla, S1
Ambudkar, SV; Gaur, M; Prasad, R; Puri, N; Sharma, M; Shukla, S1
Katayama, K; Kawahara, H; Mitsuhashi, J; Noguchi, K; Sugimoto, Y1
Ambudkar, SV; Kumar, A; Mandal, A; Prasad, R; Shukla, S1
Ambudkar, SV; Limtrakul, P; Ohnuma, S; Pintha, K; Pitchakarn, P; Pompimon, W1
Ambudkar, SV; Chanmahasathien, W; Limtrakul, P; Ohnuma, S1
Ambudkar, SV; Chen, X; Chen, ZS; Dai, CL; Fu, LW; Korlipara, VL; Kuang, YH; Liao, LQ; Patel, A; Patel, JP; Sodani, K; Tiwari, AK; Wu, CP1
Ambudkar, SV; Chufan, EE; Fukuda, M; Ishida, M; Iwabuchi, Y; Kanehara, K; Kudoh, K; Murakami, M; Naitoh, T; Ohnuma, S; Shibata, H; Sugisawa, N; Unno, M1
Abel, B; Ambudkar, SV; Durell, SR; Jacobson, KA; Murakami, M; Tosh, DK; Vahedi, S1

Trials

1 trial(s) available for azides and prazosin

ArticleYear
Inhibition of P-glycoprotein (ABCB1)- and multidrug resistance-associated protein 1 (ABCC1)-mediated transport by the orally administered inhibitor, CBT-1((R)).
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Adenosine Triphosphatases; Alkaloids; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Factors; Biological Transport; Cell Line; Cell Line, Tumor; Cyclosporins; Depsipeptides; Fluorescent Dyes; Fluorouracil; Humans; Insecta; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Prazosin; Quinolines; Rhodamine 123; Verapamil; Vinblastine

2008

Other Studies

69 other study(ies) available for azides and prazosin

ArticleYear
Photoaffinity labeling of the organic cation/H+ exchanger in renal brush border membrane vesicles.
    The Journal of biological chemistry, 1992, Jul-05, Volume: 267, Issue:19

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cations; Dihydropyridines; Dithiothreitol; Dogs; Electrophoresis, Polyacrylamide Gel; Ethylmaleimide; Hydrogen; Kidney Cortex; Membrane Glycoproteins; Microvilli; Photochemistry; Prazosin; Substrate Specificity

1992
Functional involvement of P-glycoprotein in blood-brain barrier.
    The Journal of biological chemistry, 1992, Oct-05, Volume: 267, Issue:28

    Topics: Alkaline Phosphatase; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blood-Brain Barrier; Brain; Capillaries; Cells, Cultured; Drug Interactions; Endothelium, Vascular; gamma-Glutamyltransferase; Humans; Membrane Glycoproteins; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Microscopy, Immunoelectron; Prazosin; Tumor Cells, Cultured; Verapamil; Vincristine

1992
Immunosuppressants FK506 and rapamycin function as reversal agents of the multidrug resistance phenotype.
    Blood, 1992, Sep-15, Volume: 80, Issue:6

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Daunorubicin; Drug Resistance; Drug Synergism; Humans; Iodine Radioisotopes; Membrane Glycoproteins; Phenotype; Polyenes; Prazosin; Sirolimus; Tacrolimus; Tumor Cells, Cultured

1992
Renal adrenergic receptors: localization of [125I]prazosin binding sites along the microdissected rat nephron.
    Canadian journal of physiology and pharmacology, 1992, Volume: 70, Issue:7

    Topics: Animals; Autoradiography; Azides; Binding Sites; Binding, Competitive; In Vitro Techniques; Kidney; Kidney Tubules, Proximal; Kinetics; Male; Nephrons; Norepinephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic

1992
Domain mapping of the photoaffinity drug-binding sites in P-glycoprotein encoded by mouse mdr1b.
    The Journal of biological chemistry, 1991, Nov-05, Volume: 266, Issue:31

    Topics: Affinity Labels; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Blotting, Western; Cross Reactions; Drug Resistance; Humans; Membrane Glycoproteins; Mice; Molecular Sequence Data; Peptide Mapping; Peptides; Photochemistry; Prazosin; Species Specificity

1991
The alpha 1-adrenergic photoaffinity probe [125I]arylazidoprazosin binds to a specific peptide of P-glycoprotein in multidrug-resistant cells.
    Biochemical and biophysical research communications, 1990, Jan-15, Volume: 166, Issue:1

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Neoplasm Proteins; Peptide Mapping; Prazosin; Quinazolines; Vinca Alkaloids; Vincristine

1990
Photoaffinity probes for the alpha 1-adrenergic receptor and the calcium channel bind to a common domain in P-glycoprotein.
    The Journal of biological chemistry, 1990, Mar-15, Volume: 265, Issue:8

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Binding, Competitive; Calcium Channels; Cell Line; Cell Membrane; Chymotrypsin; Dihydropyridines; Drug Resistance; Macrophages; Membrane Glycoproteins; Mice; Peptide Mapping; Prazosin; Receptors, Adrenergic, alpha; Sequence Homology, Nucleic Acid; Verapamil

1990
Autoregulation of neuromuscular transmission in the guinea-pig saphenous artery.
    European journal of pharmacology, 1987, Jul-09, Volume: 139, Issue:2

    Topics: Adenosine Triphosphate; Affinity Labels; Animals; Arteries; Azides; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Muscle, Smooth, Vascular; Neuromuscular Junction; Prazosin; Propranolol; Receptors, Adrenergic; Synaptic Transmission; Yohimbine

1987
Alpha 1-adrenergic receptor photoaffinity labeling in intact cells.
    Biochemical pharmacology, 1987, Nov-15, Volume: 36, Issue:22

    Topics: Affinity Labels; Alprenolol; Animals; Azides; Cells, Cultured; Electrophoresis, Polyacrylamide Gel; Molecular Weight; Muscle, Smooth; Photochemistry; Prazosin; Quinazolines; Receptors, Adrenergic, alpha

1987
The oligosaccharide component of alpha 1-adrenergic receptors from BC3H1 and DDT1 muscle cells. Studies with glycosidases and photoaffinity labelling of intact cells.
    The Biochemical journal, 1988, Jul-15, Volume: 253, Issue:2

    Topics: Acetylglucosaminidase; Affinity Labels; alpha-Mannosidase; Animals; Azides; Cell Line; Chromatography, Affinity; Cricetinae; Electrophoresis, Polyacrylamide Gel; Glycoside Hydrolases; Iodine Radioisotopes; Mannosidases; Mannosyl-Glycoprotein Endo-beta-N-Acetylglucosaminidase; Mice; Muscles; Oligosaccharides; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Tumor Cells, Cultured

1988
Photoaffinity labeling of the DDT1 MF-2 cell alpha 1-adrenergic receptor.
    Molecular and cellular biochemistry, 1985, Volume: 67, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Affinity Labels; Animals; Azides; Cell Line; Muscle, Smooth; Photochemistry; Prazosin; Quinazolines; Receptors, Adrenergic, alpha; Yohimbine

1985
Photoaffinity labeling of alpha 1-adrenergic receptors of rat heart.
    The Journal of biological chemistry, 1986, Apr-25, Volume: 261, Issue:12

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Dithiothreitol; Epinephrine; Heart Ventricles; Iodine Radioisotopes; Macromolecular Substances; Microbial Collagenase; Myocardium; Norepinephrine; Phentolamine; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Yohimbine

1986
Structural and pharmacological differences between codfish and rat brain alpha 1-adrenergic receptors revealed by photoaffinity labeling with 125I-APDQ.
    Acta pharmacologica et toxicologica, 1986, Volume: 58, Issue:2

    Topics: Affinity Labels; Animals; Azides; Electrophoresis, Polyacrylamide Gel; Fishes; Isoproterenol; Molecular Weight; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, alpha; Species Specificity; Stereoisomerism

1986
Affinity labeling of the DDT1 MF-2 cell alpha 1-adrenergic receptor with [3H]phenoxybenzamine.
    Biochemical pharmacology, 1986, May-15, Volume: 35, Issue:10

    Topics: Affinity Labels; Animals; Azides; Cells, Cultured; Cricetinae; Epinephrine; Male; Mesocricetus; Molecular Weight; Phenoxybenzamine; Prazosin; Receptors, Adrenergic, alpha; Stereoisomerism; Tritium; Vas Deferens

1986
In vitro activity of azithromycin and erythromycin against organisms associated with bacterial vaginosis and chancroid.
    European journal of clinical microbiology & infectious diseases : official publication of the European Society of Clinical Microbiology, 1988, Volume: 7, Issue:4

    Topics: Azides; Bacteroides; Chancroid; Erythromycin; Female; Gardnerella vaginalis; Gram-Negative Bacteria; Haemophilus ducreyi; Humans; Prazosin; Quinazolines; Vaginitis

1988
Photoaffinity labeling of the alpha 1-adrenergic receptor using an 125I-labeled aryl azide analogue of prazosin.
    Biochemistry, 1984, Jul-31, Volume: 23, Issue:16

    Topics: Affinity Labels; Animals; Azides; Binding, Competitive; Cell Membrane; Female; Indicators and Reagents; Kinetics; Liver; Molecular Weight; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1984
Cotransmitters in the motor nerves of the guinea pig vas deferens: electrophysiological evidence.
    Science (New York, N.Y.), 1982, Nov-12, Volume: 218, Issue:4573

    Topics: Adenosine Triphosphate; Animals; Azides; Guinea Pigs; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha; Receptors, Cell Surface; Vas Deferens

1982
Photoaffinity label for the alpha 1-adrenergic receptor: synthesis and effects on membrane and affinity-purified receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1983, Volume: 80, Issue:8

    Topics: Affinity Labels; Animals; Azides; Cell Membrane; Liver; Photochemistry; Prazosin; Quinazolines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha

1983
A pharmacological investigation of the biphasic nature of the contractile response of rabbit and rat vas deferens to field stimulation.
    Life sciences, 1984, Nov-05, Volume: 35, Issue:19

    Topics: Adenosine Triphosphate; Animals; Azides; Electric Stimulation; Guinea Pigs; Male; Muscle Contraction; Norepinephrine; Prazosin; Rabbits; Rats; Species Specificity; Vas Deferens

1984
Interaction of drugs with P-glycoprotein in brain capillaries.
    Biochemical pharmacology, 1995, Nov-09, Volume: 50, Issue:10

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blood-Brain Barrier; Brain; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Glycerol; In Vitro Techniques; Iodine Radioisotopes; Male; Prazosin; Rats; Rats, Sprague-Dawley; Time Factors; Tritium

1995
Characterization of multidrug resistance P-glycoprotein transport function with an organotechnetium cation.
    Biochemistry, 1995, Sep-26, Volume: 34, Issue:38

    Topics: Adenosine Triphosphate; Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cations; Cell Survival; Cells, Cultured; Colchicine; Cricetinae; Dose-Response Relationship, Drug; Doxorubicin; Humans; Kinetics; Lipid Bilayers; Pharmaceutical Preparations; Phloretin; Prazosin; Quinidine; Technetium Tc 99m Sestamibi; Tetraphenylborate

1995
Functional analysis of P-glycoprotein mutants identifies predicted transmembrane domain 11 as a putative drug binding site.
    Biochemistry, 1993, Apr-27, Volume: 32, Issue:16

    Topics: Affinity Labels; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Cell Membrane; CHO Cells; Cloning, Molecular; Colchicine; Cricetinae; Dactinomycin; Doxorubicin; Drug Resistance; Gramicidin; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Mice; Mutagenesis, Site-Directed; Phenylalanine; Prazosin; Serine; Transfection; Vinblastine

1993
Functional evidence that transmembrane 12 and the loop between transmembrane 11 and 12 form part of the drug-binding domain in P-glycoprotein encoded by MDR1.
    The Journal of biological chemistry, 1995, Mar-10, Volume: 270, Issue:10

    Topics: Affinity Labels; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line; Cisplatin; Colchicine; Dactinomycin; Doxorubicin; Drug Resistance, Multiple; Humans; Iodine Radioisotopes; Melanoma; Molecular Sequence Data; Phenotype; Prazosin; Protein Structure, Secondary; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Transfection; Tumor Cells, Cultured; Vincristine

1995
Major photoaffinity drug labeling sites for iodoaryl azidoprazosin in P-glycoprotein are within, or immediately C-terminal to, transmembrane domains 6 and 12.
    The Journal of biological chemistry, 1993, May-25, Volume: 268, Issue:15

    Topics: Affinity Labels; Amino Acid Sequence; Animals; Antibody Specificity; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Carrier Proteins; Cell Line; Cell Membrane; Chymotrypsin; Drug Resistance; Immunoblotting; Iodine Radioisotopes; Macrophages; Membrane Glycoproteins; Mice; Models, Structural; Molecular Weight; Peptide Fragments; Prazosin; Protein Structure, Secondary; Trypsin

1993
Biphasic intracellular redistribution of alpha 1-adrenergic receptors in rat liver during sepsis.
    The American journal of physiology, 1993, Volume: 265, Issue:2 Pt 2

    Topics: Animals; Autoradiography; Azides; Cell Membrane; Electrophoresis, Polyacrylamide Gel; Endoplasmic Reticulum; Infections; Intracellular Membranes; Liver; Male; Photolysis; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Tissue Distribution

1993
Alpha 1B-adrenergic receptors in rat renal microvessels.
    Kidney international, 1995, Volume: 48, Issue:5

    Topics: Affinity Labels; Alkylating Agents; Animals; Azides; Binding Sites; Blood Vessels; Clonidine; Male; Microcirculation; Prazosin; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Renal Circulation; RNA, Messenger

1995
Cyclosporin A treatment induces overexpression of P-glycoprotein in the kidney and other tissues.
    The American journal of physiology, 1996, Volume: 270, Issue:5 Pt 2

    Topics: Administration, Oral; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cyclosporine; Cyclosporins; Immunosuppressive Agents; Injections, Subcutaneous; Kidney; Male; Microvilli; Prazosin; Rats; Rats, Sprague-Dawley; Time Factors

1996
Multidrug-resistant human sarcoma cells with a mutant P-glycoprotein, altered phenotype, and resistance to cyclosporins.
    The Journal of biological chemistry, 1997, Feb-28, Volume: 272, Issue:9

    Topics: Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Survival; Cyclosporins; Dihydropyridines; DNA Topoisomerases, Type II; Doxorubicin; Drug Resistance, Multiple; Humans; Neoplasm Proteins; Phenotype; Polymerase Chain Reaction; Prazosin; Rhodamine 123; Rhodamines; Sarcoma; Vault Ribonucleoprotein Particles; Verapamil

1997
P-glycoprotein is strongly expressed in the luminal membranes of the endothelium of blood vessels in the brain.
    The Biochemical journal, 1997, Sep-01, Volume: 326 ( Pt 2)

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Brain; Capillaries; Cell Membrane; Cerebral Cortex; Endothelium, Vascular; Glycosylation; Iodine Radioisotopes; Male; Prazosin; Rats; Rats, Sprague-Dawley

1997
Evidence for two nonidentical drug-interaction sites in the human P-glycoprotein.
    Proceedings of the National Academy of Sciences of the United States of America, 1997, Sep-30, Volume: 94, Issue:20

    Topics: 3T3 Cells; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Cell Line; Cyclosporine; Flupenthixol; Humans; Insecta; Iodine Radioisotopes; Mice; Models, Biological; Prazosin; Radioligand Assay; Vanadates; Vinblastine

1997
HIV-1 protease inhibitors are substrates for the MDR1 multidrug transporter.
    Biochemistry, 1998, Mar-17, Volume: 37, Issue:11

    Topics: 3T3 Cells; Adenosine Triphosphatases; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Biological Transport; Carcinoma, Squamous Cell; Drug Resistance, Multiple; Enzyme Activation; Genes, MDR; HIV Protease Inhibitors; HIV-1; Humans; Iodine Radioisotopes; Mice; Prazosin; Spodoptera; Substrate Specificity; Tumor Cells, Cultured; Vinblastine

1998
Drug binding to P-glycoprotein is inhibited in normal tissues following SDZ-PSC 833 treatment.
    International journal of cancer, 1998, May-29, Volume: 76, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Brain; Calcium Channel Blockers; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Fluorescent Dyes; Injections, Subcutaneous; Iodine Radioisotopes; Kidney; Liver; Male; Microvilli; Photoaffinity Labels; Prazosin; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Verapamil; Vinblastine

1998
Mutations in the nucleotide-binding sites of P-glycoprotein that affect substrate specificity modulate substrate-induced adenosine triphosphatase activity.
    Biochemistry, 1998, Jun-23, Volume: 37, Issue:25

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Binding Sites; Iodine Radioisotopes; Mice; Molecular Sequence Data; Mutagenesis, Insertional; Photoaffinity Labels; Pichia; Prazosin; Recombinant Proteins; Substrate Specificity

1998
Photoaffinity labeling of human P-glycoprotein: effect of modulator interaction and ATP hydrolysis on substrate binding.
    Methods in enzymology, 1998, Volume: 292

    Topics: Adenosine Triphosphate; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Baculoviridae; Cell Culture Techniques; Cell Line; Cell Membrane; Chromatography, Affinity; Drug Resistance, Multiple; Electrophoresis, Polyacrylamide Gel; Humans; Indicators and Reagents; Iodine Radioisotopes; Kinetics; Prazosin; Recombinant Proteins; Spodoptera; Transfection; Vanadates

1998
High-level expression of mouse Mdr3 P-glycoprotein in yeast Pichia pastoris and characterization of ATPase activity.
    Methods in enzymology, 1998, Volume: 292

    Topics: Adenosine Triphosphatases; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Binding, Competitive; Cell Fractionation; Cell Membrane; Cloning, Molecular; Colchicine; Doxorubicin; Drug Resistance, Multiple; Iodine Radioisotopes; Kinetics; Mice; Pichia; Plasmids; Prazosin; Recombinant Proteins; Time Factors; Transformation, Genetic; Valinomycin; Vinblastine

1998
Functional expression of human P-glycoprotein from plasmids using vaccinia virus-bacteriophage T7 RNA polymerase system.
    Methods in enzymology, 1998, Volume: 292

    Topics: Adenosine Triphosphatases; Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Membrane; Cloning, Molecular; Colchicine; Daunorubicin; Dihydropyridines; DNA-Directed RNA Polymerases; Drug Resistance, Multiple; Electrophoresis, Polyacrylamide Gel; Escherichia coli; HeLa Cells; Humans; Indicators and Reagents; Iodine Radioisotopes; Osteosarcoma; Plasmids; Polymerase Chain Reaction; Prazosin; Recombinant Proteins; Restriction Mapping; Transfection; Tritium; Tumor Cells, Cultured; Vaccinia virus; Vinblastine; Viral Proteins

1998
Structural flexibility of the linker region of human P-glycoprotein permits ATP hydrolysis and drug transport.
    Biochemistry, 1998, Sep-29, Volume: 37, Issue:39

    Topics: 3T3 Cells; Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Sequence; Animals; Antibodies, Monoclonal; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Base Sequence; Biological Transport; Cell Membrane; Drug Resistance, Multiple; Genetic Vectors; HeLa Cells; Humans; Hydrolysis; Iodine Radioisotopes; Mice; Molecular Sequence Data; Mutagenesis, Insertional; Osteosarcoma; Peptide Fragments; Prazosin; Protein Binding; Protein Conformation; Recombinant Proteins; Sequence Deletion; Tumor Cells, Cultured; Verapamil

1998
Analysis of random recombination between human MDR1 and mouse mdr1a cDNA in a pHaMDR-dihydrofolate reductase bicistronic expression system.
    Molecular pharmacology, 1998, Volume: 54, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; DNA, Complementary; Genetic Vectors; Humans; Iodine Radioisotopes; KB Cells; Mice; Photoaffinity Labels; Prazosin; Protein Structure, Tertiary; Recombinant Fusion Proteins; Recombinant Proteins; Recombination, Genetic; Sensitivity and Specificity; Tetrahydrofolate Dehydrogenase; Transfection

1998
A single amino acid residue contributes to distinct mechanisms of inhibition of the human multidrug transporter by stereoisomers of the dopamine receptor antagonist flupentixol.
    Biochemistry, 1999, May-18, Volume: 38, Issue:20

    Topics: Adenosine Triphosphate; Alanine; Amino Acid Substitution; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Dopamine Antagonists; Flupenthixol; HeLa Cells; Humans; Hydrolysis; Iodine Radioisotopes; Mutagenesis, Site-Directed; Phenylalanine; Photoaffinity Labels; Prazosin; Receptors, Dopamine; Stereoisomerism; Substrate Specificity; Tumor Cells, Cultured; Verapamil

1999
Both ATP sites of human P-glycoprotein are essential but not symmetric.
    Biochemistry, 1999, Oct-19, Volume: 38, Issue:42

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Motifs; Amino Acid Substitution; Antibodies, Monoclonal; Asparagine; Aspartic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Body Temperature; Cell Membrane; Consensus Sequence; Enzyme Activation; Freezing; HeLa Cells; Humans; Peptide Fragments; Phosphorus Radioisotopes; Photoaffinity Labels; Point Mutation; Prazosin; Protein Conformation; Recombinant Fusion Proteins; Vanadates; Verapamil

1999
Functional characterization of glycosylation-deficient human P-glycoprotein using a vaccinia virus expression system.
    The Journal of membrane biology, 2000, Feb-01, Volume: 173, Issue:3

    Topics: Acetylcysteine; Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cysteine Endopeptidases; Cysteine Proteinase Inhibitors; Flow Cytometry; Glycosylation; HeLa Cells; Humans; Membrane Glycoproteins; Multienzyme Complexes; Mutation; Photoaffinity Labels; Prazosin; Proteasome Endopeptidase Complex; Transfection; Trypsin; Vaccinia virus

2000
Characterization of the catalytic cycle of ATP hydrolysis by human P-glycoprotein. The two ATP hydrolysis events in a single catalytic cycle are kinetically similar but affect different functional outcomes.
    The Journal of biological chemistry, 2001, Apr-13, Volume: 276, Issue:15

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Catalysis; Humans; Hydrolysis; Iodine Radioisotopes; Kinetics; Prazosin; Protein Conformation

2001
Identification and localization of three photobinding sites of iodoarylazidoprazosin in hamster P-glycoprotein.
    European journal of biochemistry, 2001, Volume: 268, Issue:9

    Topics: Amino Acid Sequence; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; CHO Cells; Cricetinae; Drug Resistance, Multiple; Humans; In Vitro Techniques; Iodine Radioisotopes; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Photoaffinity Labels; Photochemistry; Prazosin

2001
Transmembrane domain (TM) 9 represents a novel site in P-glycoprotein that affects drug resistance and cooperates with TM6 to mediate [125I]iodoarylazidoprazosin labeling.
    Molecular pharmacology, 2001, Volume: 60, Issue:2

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Cells, Cultured; Cricetinae; Cyclosporine; Drug Interactions; Drug Resistance; Drug Resistance, Multiple; Iodine Radioisotopes; Membrane Proteins; Mutagenesis, Site-Directed; Prazosin; Protein Structure, Tertiary; Transfection; Verapamil

2001
Further characterization of the sixth transmembrane domain of Pgp1 by site-directed mutagenesis.
    Cancer chemotherapy and pharmacology, 2001, Volume: 48, Issue:5

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line; Cricetinae; Hydrophobic and Hydrophilic Interactions; Membrane Proteins; Mutagenesis, Site-Directed; Photoaffinity Labels; Prazosin; Structure-Activity Relationship; Transfection; Verapamil

2001
Modulation of P-glycoprotein expression and function by curcumin in multidrug-resistant human KB cells.
    Biochemical pharmacology, 2002, Aug-15, Volume: 64, Issue:4

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cell Survival; Curcumin; Down-Regulation; Drug Resistance, Multiple; Fluorescent Dyes; Gene Expression; Humans; KB Cells; Photoaffinity Labels; Prazosin; Rhodamine 123; Tumor Cells, Cultured; Vinblastine

2002
A modified synthesis of iodoazidoaryl prazosin.
    The Journal of organic chemistry, 2002, Nov-15, Volume: 67, Issue:23

    Topics: Antihypertensive Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Drug Resistance, Multiple; Piperazine; Piperazines; Prazosin

2002
N-terminal truncation of human alpha1D-adrenoceptors increases expression of binding sites but not protein.
    European journal of pharmacology, 2003, Feb-21, Volume: 462, Issue:1-3

    Topics: Amino Acid Sequence; Azides; Binding Sites; Binding, Competitive; Calcium; Cell Line; Glycosylation; Humans; Iodine Radioisotopes; Kinetics; Molecular Sequence Data; Norepinephrine; Oligopeptides; Peptides; Phenethylamines; Photoaffinity Labels; Prazosin; Precipitin Tests; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sequence Deletion; Tetralones; Transfection; Uridine Triphosphate

2003
The molecular basis of the action of disulfiram as a modulator of the multidrug resistance-linked ATP binding cassette transporters MDR1 (ABCB1) and MRP1 (ABCC1).
    Molecular pharmacology, 2004, Volume: 65, Issue:3

    Topics: 3T3 Cells; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cells, Cultured; Dihydropyridines; Disulfiram; Drug Interactions; Drug Resistance, Multiple; Enzyme Inhibitors; Humans; Hydrolysis; Mice; Multidrug Resistance-Associated Proteins; Phosphorus Radioisotopes; Prazosin

2004
Biochemical basis of polyvalency as a strategy for enhancing the efficacy of P-glycoprotein (ABCB1) modulators: stipiamide homodimers separated with defined-length spacers reverse drug efflux with greater efficacy.
    Biochemistry, 2004, Mar-02, Volume: 43, Issue:8

    Topics: Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Binding, Competitive; Biological Transport; Boron Compounds; Dimerization; Drug Carriers; Fluoresceins; Humans; Hydrolysis; Iodine Radioisotopes; Mice; NIH 3T3 Cells; Photoaffinity Labels; Polyenes; Prazosin

2004
Biochemical mechanism of modulation of human P-glycoprotein (ABCB1) by curcumin I, II, and III purified from Turmeric powder.
    Biochemical pharmacology, 2004, Nov-15, Volume: 68, Issue:10

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Cell Survival; Curcuma; Curcumin; Diarylheptanoids; Drug Combinations; Drug Interactions; Fluoresceins; Humans; Iodine Radioisotopes; KB Cells; Multidrug Resistance-Associated Proteins; Photoaffinity Labels; Plant Extracts; Prazosin; Rhodamine 123; Vinblastine

2004
The role of hydrogen bond acceptor groups in the interaction of substrates with Pdr5p, a major yeast drug transporter.
    Biochemistry, 2005, Jul-19, Volume: 44, Issue:28

    Topics: Antifungal Agents; Antineoplastic Agents; ATP-Binding Cassette Transporters; Azides; Binding Sites; Biological Transport; Carbazoles; Clotrimazole; Cross-Linking Reagents; Ellipticines; Hydrogen Bonding; Multidrug Resistance-Associated Proteins; Prazosin; Rhodamines; Saccharomyces cerevisiae Proteins; Substrate Specificity; Tritium; Trityl Compounds; Xenobiotics

2005
Allosteric modulation bypasses the requirement for ATP hydrolysis in regenerating low affinity transition state conformation of human P-glycoprotein.
    The Journal of biological chemistry, 2006, Apr-21, Volume: 281, Issue:16

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Allosteric Site; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Catalytic Domain; Cell Line; Cell Membrane; Flupenthixol; Humans; Hydrolysis; Insecta; Ligands; Molecular Conformation; Prazosin; Protein Binding; Protein Conformation; Protein Structure, Tertiary; Thioxanthenes; Time Factors; Trypsin; Vanadates

2006
Biochemical and pharmacological properties of an allosteric modulator site of the human P-glycoprotein (ABCB1).
    Biochemical pharmacology, 2006, Jul-14, Volume: 72, Issue:2

    Topics: Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Chromatography, Affinity; Electrophoresis, Polyacrylamide Gel; Flupenthixol; Humans; Phenothiazines; Prazosin; Xanthines

2006
The calcium channel blockers, 1,4-dihydropyridines, are substrates of the multidrug resistance-linked ABC drug transporter, ABCG2.
    Biochemistry, 2006, Jul-25, Volume: 45, Issue:29

    Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Calcium Channel Blockers; Cell Line; Chlorophyll; Dihydropyridines; Drug Interactions; Humans; Mitoxantrone; Neoplasm Proteins; Nicardipine; Nifedipine; Photoaffinity Labels; Prazosin

2006
Gomisin A alters substrate interaction and reverses P-glycoprotein-mediated multidrug resistance in HepG2-DR cells.
    Biochemical pharmacology, 2006, Sep-28, Volume: 72, Issue:7

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Anticarcinogenic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Line, Tumor; Cell Survival; Cyclooctanes; Dioxoles; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Hydrolysis; Lignans; Prazosin; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Vanadates; Verapamil; Vinblastine

2006
Modulation of the function of the multidrug resistance-linked ATP-binding cassette transporter ABCG2 by the cancer chemopreventive agent curcumin.
    Molecular cancer therapeutics, 2006, Volume: 5, Issue:8

    Topics: Adenosine Triphosphate; Anticarcinogenic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Biological Transport; Chlorophyll; Curcumin; Dihydropyridines; Drug Resistance, Neoplasm; Humans; Hydrolysis; Mitoxantrone; Mutation; Neoplasm Proteins; Prazosin; Toxicity Tests; Tumor Cells, Cultured

2006
Bivalent probes of the human multidrug transporter P-glycoprotein.
    Biochemistry, 2006, Sep-26, Volume: 45, Issue:38

    Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cross-Linking Reagents; Dimerization; Doxorubicin; Emetine; Flow Cytometry; Humans; Hydrolysis; Inhibitory Concentration 50; Models, Biological; Molecular Probes; Photoaffinity Labels; Prazosin; Rhodamine 123; Substrate Specificity; Tumor Cells, Cultured

2006
Sipholenol A, a marine-derived sipholane triterpene, potently reverses P-glycoprotein (ABCB1)-mediated multidrug resistance in cancer cells.
    Cancer science, 2007, Volume: 98, Issue:9

    Topics: Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Callyspongia; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Iodine Radioisotopes; KB Cells; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Photoaffinity Labels; Prazosin; Triterpenes

2007
Curcumin inhibits the activity of ABCG2/BCRP1, a multidrug resistance-linked ABC drug transporter in mice.
    Pharmaceutical research, 2009, Volume: 26, Issue:2

    Topics: Administration, Oral; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Biological Availability; Blood-Brain Barrier; Boron Compounds; Cell Line, Tumor; Curcumin; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Neoplasm; Humans; Mice; Mice, Knockout; Neoplasm Proteins; Prazosin; Rats; Rats, Sprague-Dawley; Sulfasalazine

2009
Becatecarin (rebeccamycin analog, NSC 655649) is a transport substrate and induces expression of the ATP-binding cassette transporter, ABCG2, in lung carcinoma cells.
    Cancer chemotherapy and pharmacology, 2009, Volume: 64, Issue:3

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Biological Transport; Carbazoles; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescence; Gene Expression Regulation, Neoplastic; Glucosides; Humans; Immunoblotting; Iodine Radioisotopes; Lung Neoplasms; Neoplasm Proteins; Prazosin

2009
The amino acid residues of transmembrane helix 5 of multidrug resistance protein CaCdr1p of Candida albicans are involved in substrate specificity and drug transport.
    Biochimica et biophysica acta, 2009, Volume: 1788, Issue:9

    Topics: Adenosine Triphosphatases; Amino Acid Sequence; Azides; Fluconazole; Fungal Proteins; Itraconazole; Ketoconazole; Membrane Transport Proteins; Miconazole; Mutagenesis, Site-Directed; Prazosin; Protein Transport; Rhodamines; Saccharomyces cerevisiae; Substrate Specificity

2009
Pharmacological interaction with sunitinib is abolished by a germ-line mutation (1291T>C) of BCRP/ABCG2 gene.
    Cancer science, 2010, Volume: 101, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Drug Resistance, Neoplasm; Estrone; Germ-Line Mutation; Humans; Indoles; K562 Cells; Mice; Neoplasm Proteins; Prazosin; Protein Kinase Inhibitors; Pyrroles; Sunitinib; Vincristine

2010
Divergent signature motifs of nucleotide binding domains of ABC multidrug transporter, CaCdr1p of pathogenic Candida albicans, are functionally asymmetric and noninterchangeable.
    Biochimica et biophysica acta, 2010, Volume: 1798, Issue:9

    Topics: Adenosine Triphosphate; Amino Acid Motifs; Azides; Binding Sites; Fungal Proteins; Membrane Transport Proteins; Mutagenesis, Site-Directed; Prazosin; Structure-Activity Relationship

2010
Kuguacin J isolated from Momordica charantia leaves inhibits P-glycoprotein (ABCB1)-mediated multidrug resistance.
    The Journal of nutritional biochemistry, 2012, Volume: 23, Issue:1

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Fluoresceins; Humans; Molecular Structure; Momordica charantia; Paclitaxel; Plant Leaves; Prazosin; Rhodamine 123; Triterpenes; Uterine Cervical Neoplasms; Vinblastine

2012
Biochemical mechanism of modulation of human P-glycoprotein by stemofoline.
    Planta medica, 2011, Volume: 77, Issue:18

    Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Heterocyclic Compounds, 4 or More Rings; Humans; Insecta; Membranes; Photoaffinity Labels; Plant Roots; Prazosin; Protein Binding; Rhodamine 123; Stemonaceae; Vinblastine

2011
OSI-930 analogues as novel reversal agents for ABCG2-mediated multidrug resistance.
    Biochemical pharmacology, 2012, Sep-15, Volume: 84, Issue:6

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Azides; Benzene Derivatives; Biological Transport; Cells, Cultured; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Mitoxantrone; Neoplasm Proteins; Nitro Compounds; Photoaffinity Labels; Prazosin; Pyridines; Quinolines; Structure-Activity Relationship; Thiophenes; Transfection

2012
Synthetic Analogs of Curcumin Modulate the Function of Multidrug Resistance-Linked ATP-Binding Cassette Transporter ABCG2.
    Drug metabolism and disposition: the biological fate of chemicals, 2017, Volume: 45, Issue:11

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; Azides; Benzene Derivatives; Biological Availability; Biological Transport; Camptothecin; Cell Line, Tumor; Curcumin; Drug Resistance, Neoplasm; Drug Synergism; Flow Cytometry; Humans; Irinotecan; Ketones; Mitoxantrone; Neoplasm Proteins; Prazosin

2017
Evidence for the Interaction of A
    Molecular pharmacology, 2019, Volume: 96, Issue:2

    Topics: Adenosine A3 Receptor Agonists; ATP Binding Cassette Transporter, Subfamily B; Azides; Binding Sites; HeLa Cells; Humans; Models, Molecular; Molecular Docking Simulation; Paclitaxel; Prazosin; Structure-Activity Relationship; Verapamil

2019