aq-ra 741 has been researched along with piperidines in 18 studies
Studies (aq-ra 741) | Trials (aq-ra 741) | Recent Studies (post-2010) (aq-ra 741) | Studies (piperidines) | Trials (piperidines) | Recent Studies (post-2010) (piperidines) |
---|---|---|---|---|---|
25 | 0 | 3 | 40,235 | 5,221 | 14,545 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 16 (88.89) | 18.2507 |
2000's | 1 (5.56) | 29.6817 |
2010's | 1 (5.56) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Hendriks, MG; Pfaffendorf, M; Van Zwieten, PA | 2 |
Bungardt, E; Feifel, R; Lambrecht, G; Moser, U; Mutschler, E; Surprenant, A; Tacke, R; Vockert, E | 1 |
Brann, MR; Gdula, D; Wess, J | 1 |
Doods, H; Entzeroth, M; Mayer, N | 1 |
Roffel, AF; ten Berge, RE; Zaagsma, J | 2 |
Classen, M; Schaffer, K; Schepp, W; Schusdziarra, V; Wegner, U; Weigert, N | 1 |
Hamstra, JJ; Roffel, AF; Santing, RE; ten Berge, RE; Zaagsma, J | 1 |
Birdsall, NJ; Lazareno, S | 1 |
Baumgold, J; Cohen, VI; De La Cruz, R; Jin, B; Reba, RC; Rzeszotarski, WJ | 1 |
Bechtel, WD; Doods, HN; Engel, W; Ensinger, HA; Entzeroth, M; Ladinsky, H; Mihm, G; Quirion, R; Rudolf, K; Schiavi, GB | 1 |
Dingermann, T; Voith, G | 1 |
Gillberg, PG; Nilvebrant, L; Sundquist, S | 1 |
Budriesi, R; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S; Tumiatti, V | 1 |
Eglen, RM; Watson, N | 1 |
Daniels, DV; Eglen, RM; Ford, AP; Hegde, SS; Meloy, TD | 1 |
Bayles, J; Dosdall, DJ; Fisher, SJ; Hirahara, AM; Huang, Y; Oxspring, M; Reno, CM | 1 |
2 review(s) available for aq-ra 741 and piperidines
Article | Year |
---|---|
Therapeutic potential of CNS-active M2 antagonists: novel structures and pharmacology.
Topics: Animals; Benzodiazepinones; Brain; CHO Cells; Cognition Disorders; Cricetinae; Dibenzazepines; Drug Design; Motor Activity; Parasympatholytics; Piperidines; Pirenzepine; Pyridines; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1993 |
Muscarinic receptor antagonists.
Topics: Airway Obstruction; Animals; Asthma; Benzodiazepinones; Bronchi; Gallamine Triethiodide; Humans; Muscarinic Antagonists; Muscle, Smooth; Piperidines; Trachea | 1999 |
16 other study(ies) available for aq-ra 741 and piperidines
Article | Year |
---|---|
Characterization of the muscarinic receptor subtype mediating vasodilation in the rat perfused mesenteric vascular bed preparation.
Topics: Animals; Atropine; Benzodiazepinones; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Methacholine Chloride; Parasympatholytics; Perfusion; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Muscarinic; Vasodilation | 1992 |
Characterization of muscarinic receptors mediating vasodilation in guinea-pig ileum submucosal arterioles by the use of computer-assisted videomicroscopy.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Arterioles; Benzodiazepinones; Carbachol; Guinea Pigs; Ileum; Methacholine Chloride; Muscarine; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Parasympathomimetics; Piperidines; Pirenzepine; Prostaglandin Endoperoxides, Synthetic; Receptors, Muscarinic; Vasodilation | 1992 |
Structural basis of the subtype selectivity of muscarinic antagonists: a study with chimeric m2/m5 muscarinic receptors.
Topics: Alkaloids; Amino Acid Sequence; Benzodiazepinones; Chimera; Dibenzazepines; Furans; Humans; Molecular Sequence Data; Muscarinic Antagonists; N-Methylscopolamine; Naphthalenes; Parasympatholytics; Piperazines; Piperidines; Receptors, Muscarinic; Scopolamine Derivatives; Sequence Homology, Nucleic Acid | 1992 |
Cardioselectivity of AQ-RA 741, a novel tricyclic antimuscarinic drug.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Cats; Female; Guinea Pigs; Heart; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1991 |
Conditional involvement of muscarinic M1 receptors in vagally mediated contraction of guinea-pig bronchi.
Topics: Adrenergic beta-Antagonists; Animals; Benzodiazepinones; Bronchoconstriction; Electric Stimulation; Female; Guinea Pigs; Hexamethonium; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nicotinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Timolol; Vagus Nerve | 1995 |
Functional characterization of a muscarinic receptor stimulating gastrin release from rabbit antral G-cells in primary culture.
Topics: Animals; Arecoline; Atropine; Benzodiazepinones; Carbachol; Cell Adhesion; Cell Separation; Cells, Cultured; Gastrins; Immunohistochemistry; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pyloric Antrum; Rabbits; Receptors, Muscarinic | 1994 |
Dysfunction of muscarinic M2 receptors after the early allergic reaction: possible contribution to bronchial hyperresponsiveness in allergic guinea-pigs.
Topics: Administration, Inhalation; Allergens; Animals; Asthma; Benzodiazepinones; Bronchial Hyperreactivity; Diamines; Disease Models, Animal; Electric Stimulation; Female; Gallamine Triethiodide; Guinea Pigs; Heart; Histamine; Hypersensitivity; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle, Smooth; Neuromuscular Junction; Parasympatholytics; Pilocarpine; Piperidines; Pirenzepine; Receptors, Muscarinic; Trachea | 1995 |
Characterization of the muscarinic receptors in the mesenteric vascular bed of spontaneously hypertensive rats.
Topics: Animals; Atropine; Benzodiazepinones; Endothelium, Vascular; Hypertension; Male; Mesenteric Artery, Superior; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Muscarinic; Vasodilation | 1993 |
Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng-Prusoff equations.
Topics: Acetylcholine; Animals; Benzodiazepinones; Binding, Competitive; CHO Cells; Cricetinae; Drug Antagonism; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indicators and Reagents; Membranes; Models, Biological; Parasympatholytics; Piperidines; Pirenzepine; Receptors, Muscarinic; Regression Analysis | 1993 |
Synthesis and structure-activity relationship of some 5-[[[(dialkylamino)alkyl]-1-piperidinyl]acetyl]-10,11-dihydro-5H- benzo[b,e][1,4]diazepin-11-ones as M2-selective antimuscarinics.
Topics: Animals; Benzodiazepinones; Brain; Mice; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1993 |
Muscarinic inhibitory autoreceptors in different generations of human airways.
Topics: Acetylcholine; Aged; Atropine; Autoreceptors; Benzodiazepinones; Bronchi; Cholinergic Fibers; Chromatography, High Pressure Liquid; Electric Stimulation; Female; Gallamine Triethiodide; Humans; In Vitro Techniques; Male; Middle Aged; Muscarinic Antagonists; Muscle Contraction; Nerve Endings; Piperidines; Receptors, Muscarinic; Trachea | 1996 |
Expression of the human muscarinic receptor gene m2 in Dictyostelium discoideum.
Topics: Amino Acid Sequence; Animals; Base Sequence; Benzodiazepinones; Cell Membrane; Dictyostelium; Discoidins; Fungal Proteins; Gene Expression; Humans; Lectins; Molecular Sequence Data; Muscarinic Antagonists; Parasympatholytics; Piperidines; Promoter Regions, Genetic; Protein Sorting Signals; Protozoan Proteins; Receptors, Muscarinic | 1995 |
Comparison of the in vitro and in vivo profiles of tolterodine with those of subtype-selective muscarinic receptor antagonists.
Topics: Animals; Benzhydryl Compounds; Benzodiazepinones; Benzofurans; Cats; Cerebral Cortex; CHO Cells; Cresols; Cricetinae; Dibenzazepines; Electric Stimulation; Female; Guinea Pigs; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Myocardium; Phenylpropanolamine; Piperidines; Pyrrolidines; Receptors, Muscarinic; Saliva; Salivary Glands; Tolterodine Tartrate; Urinary Bladder | 1998 |
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists.
Topics: Animals; Atrial Function; Benzodiazepines; Benzodiazepinones; Diamines; Drug Design; Guinea Pigs; Heart Atria; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Submandibular Gland; Trachea | 1995 |
Functional characterization of rat submaxillary gland muscarinic receptors using microphysiometry.
Topics: Alkaloids; Animals; Atropine; Benzhydryl Compounds; Benzodiazepinones; Binding, Competitive; Biosensing Techniques; Carbachol; Cholinergic Agonists; Cresols; Diamines; Dose-Response Relationship, Drug; Furans; Male; Mandelic Acids; Muscarinic Antagonists; Naphthalenes; Phenethylamines; Phenylpropanolamine; Piperidines; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Tolterodine Tartrate | 2001 |
Severe Hypoglycemia-Induced Fatal Cardiac Arrhythmias Are Mediated by the Parasympathetic Nervous System in Rats.
Topics: Animals; Arrhythmias, Cardiac; Benzodiazepinones; Disease Models, Animal; Hypoglycemia; Male; Mecamylamine; Muscarinic Antagonists; Nicotinic Antagonists; Parasympathetic Nervous System; Piperidines; Rats; Rats, Sprague-Dawley; Sympathectomy, Chemical; Vagotomy | 2019 |