Page last updated: 2024-09-04

als 8123 and esmolol

als 8123 has been researched along with esmolol in 3 studies

Compound Research Comparison

Studies
(als 8123)
Trials
(als 8123)
Recent Studies (post-2010)
(als 8123)
Studies
(esmolol)
Trials
(esmolol)
Recent Studies (post-2010) (esmolol)
5011,023309266

Protein Interaction Comparison

ProteinTaxonomyals 8123 (IC50)esmolol (IC50)
Beta-1 adrenergic receptorHomo sapiens (human)0.197

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19902 (66.67)18.7374
1990's1 (33.33)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anderson, WG; Erhardt, PW; Gorczynski, RJ; Woo, CM1
Flaherty, JF; Gambertoglio, JG; Hulse, JD; La Follette, G; Warnock, DG; Wong, B1
Allen, SJ; Bischoff, I; Davis, KL; Geissler, HJ; Mehlhorn, U; Mutschler, E; Warters, RD1

Other Studies

3 other study(ies) available for als 8123 and esmolol

ArticleYear
Ultra-short-acting beta-adrenergic receptor blocking agents. 2. (Aryloxy)propanolamines containing esters on the aryl function.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Chemical Phenomena; Chemistry; Dogs; Guinea Pigs; In Vitro Techniques; Muscle, Smooth; Muscle, Smooth, Vascular; Propanolamines; Structure-Activity Relationship; Time Factors

1982
Pharmacokinetics of esmolol and ASL-8123 in renal failure.
    Clinical pharmacology and therapeutics, 1989, Volume: 45, Issue:3

    Topics: Adrenergic beta-Antagonists; Adult; Aged; Humans; Kidney Failure, Chronic; Male; Middle Aged; Peritoneal Dialysis, Continuous Ambulatory; Propanolamines; Renal Dialysis

1989
Beta-blockade as an alternative to cardioplegic arrest during cardiopulmonary bypass.
    The Annals of thoracic surgery, 1998, Volume: 65, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Body Water; Cardioplegic Solutions; Cardiopulmonary Bypass; Coronary Vessels; Crystalloid Solutions; Dogs; Edema, Cardiac; Female; Heart; Heart Arrest, Induced; Heart Rate; Infusions, Intravenous; Injections, Intravenous; Isotonic Solutions; Lactates; Male; Myocardial Contraction; Myocardial Ischemia; Myocardium; Plasma Substitutes; Propanolamines; Stroke Volume; Ventricular Function, Left

1998