Page last updated: 2024-09-05

ag 112 and cgp 57380

ag 112 has been researched along with cgp 57380 in 1 studies

Compound Research Comparison

Studies
(ag 112)
Trials
(ag 112)
Recent Studies (post-2010)
(ag 112)
Studies
(cgp 57380)
Trials
(cgp 57380)
Recent Studies (post-2010) (cgp 57380)
1901064044

Protein Interaction Comparison

ProteinTaxonomyag 112 (IC50)cgp 57380 (IC50)
Serine/threonine-protein kinase Sgk1Homo sapiens (human)2.7
Dual specificity tyrosine-phosphorylation-regulated kinase 3Homo sapiens (human)3.2
Cytochrome P450 1A2Homo sapiens (human)1.6
Proto-oncogene tyrosine-protein kinase LCK Mus musculus (house mouse)2.5
Eukaryotic translation initiation factor 4EHomo sapiens (human)3
Cytochrome P450 2D6Homo sapiens (human)1.6
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)5
Casein kinase I isoform deltaHomo sapiens (human)0.51
Serine/threonine-protein kinase BRSK2Homo sapiens (human)1.1
Aurora kinase BHomo sapiens (human)2.5
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)1.2182
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)2.06

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1

Other Studies

1 other study(ies) available for ag 112 and cgp 57380

ArticleYear
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013