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adenosine and diazepam

adenosine has been researched along with diazepam in 72 studies

Research

Studies (72)

TimeframeStudies, this research(%)All Research%
pre-199047 (65.28)18.7374
1990's15 (20.83)18.2507
2000's8 (11.11)29.6817
2010's2 (2.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Schultz, J4
Phillis, JW2
Jones, DJ; Medina, MA; Palmer, GC; Stavinoha, WB1
Advenier, C; Candenas, ML; Devillier, P; Naline, E1
Haraguchi, H; Kuribara, H1
Poltavchenko, GM1
Advenier, C; Blanc, M; Devillier, P; Gnassounou, JP1
Connick, JH; Mally, J; Stone, TW1
Czuczwar, SJ; Janusz, W; Kleinrok, Z; Szczepanik, B; Wamil, A1
Bridson, PK; Daly, JW; Hide, I1
Dragunow, M1
Altman, HJ; Barraco, RA; Brown, BD; Commissaris, RL; Damian, GM; McCloskey, TC1
Holtzman, SG1
De Mendonça, A; Ribeiro, JA1
Davies, LP; Dodd, PR; Dyer, JA; Johnston, GA; Nielsen, B; Watson, WE; Wong, LS1
O'Regan, MH; Phillis, JW1
Bender, AS; Hertz, L1
Hernández, J; Ribeiro, JA; Ruiz, F1
Akahane, K; Chiba, S; Furukawa, Y; Haniuda, M; Ogiwara, Y; Takeda, M1
Arvidsson, S; Ekström-Jodal, B; Martinell, S; Niemand, D; Svedmyr, N2
Sanderson, G; Scholfield, CN1
Clanachan, AS; Hammond, JR1
Fukuda, H; Ishida, Y; Kotani, M; Moritoki, H; Takei, M; Ueyama, T1
Furukawa, T; Katsuragi, T; Ushijima, I1
Bender, AS; Phillis, JW; Wu, PH3
Barker, PH; Clanachan, AS1
Paul, SM; Skolnick, P1
Phillis, JW; Wu, PH1
Galloway, MP; Roth, RH1
Annau, Z; Katims, JJ; Snyder, SH1
Annau, Z; Bruns, RF; Daly, JW; Katims, JJ; Snyder, SH1
Irmscher, K; Jones, R; Lock, KL; Marangos, PJ; Paul, SM; Skolnick, P1
Davies, LP; York, MJ1
Boulenger, JP; Marangos, PJ; Patel, J1
Boulenger, JP; Marangos, PJ; Parma, AM; Patel, J; Post, RM1
Davies, LP; Hambley, JW1
Snyder, SH1
Lloyd, HG; Morgan, PF; Stone, TW2
Kulkarni, SK; Mehta, AK1
Barraco, RA; Delong, RE; Phillis, JW1
Waszczak, BL1
Katsuragi, T; Su, C1
Crawley, JN; Marangos, PJ; Patel, J1
Clanachan, AS; Marshall, RJ2
Cook, AF; Davies, LP; Poonian, M; Taylor, KM1
Lock, KL; Marangos, P; Paugh, B; Paul, S; Skolnick, P; Windsor, R1
Phillis JW Siemens, RK; Siemens, RK; Wu, PH1
Biggio, G; Concas, A; Dazzi, L; Maciocco, E; Mascia, MP; Ongini, E; Santoro, G1
Chang, CC; Chiou, LC; Ling, JY1
Fisher, CE; Hughes, RN1
Busch, L; Tessler, J; Werner, S1
Brown, JK; O'Regan, ME1
Cseppentö, A; Kovács, P; Nagy, E; Szabó, JZ; Szentmiklósi, AJ; Ujfalusi, A1
Ben-Ari, Y; Dzhala, V; Khalilov, I; Khazipov, R1
Büyükokuroğlu, ME; Demirezer, LO; Güvenalp, Z1
Drooglever-Fortuyn, H; Rongen, GA; Smits, P; van Ginneken, EE1
Tuovinen, K1
Fidecka, S; Listos, J; Malec, D1
Fidecka, S; Listos, J; Talarek, S1

Reviews

6 review(s) available for adenosine and diazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
The role of adenosine in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1988, Volume: 12, Issue:4

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Arousal; Benzodiazepinones; Brain; Carbolines; Diazepam; Flumazenil; gamma-Aminobutyric Acid; Neural Inhibition; Neurons; Purkinje Cells; Rats; Receptors, GABA-A

1988
The mechanism(s) of action of the benzodiazepines.
    Medicinal research reviews, 1981,Spring, Volume: 1, Issue:1

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Caffeine; Carbolines; Cats; Cattle; Diazepam; gamma-Aminobutyric Acid; Humans; Molecular Weight; Muscle Relaxation; Neurotransmitter Agents; Niacinamide; Purines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Sleep Wake Disorders

1981
Adenosine's role in the central actions of the benzodiazepines.
    Progress in neuro-psychopharmacology & biological psychiatry, 1984, Volume: 8, Issue:4-6

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepinones; Brain; Cats; Cell Line; Cerebral Cortex; Diazepam; Flumazenil; Rats; Synaptosomes; Thioinosine

1984
Adenosine receptor interactions and anxiolytics.
    Neuropharmacology, 1983, Volume: 22, Issue:12B

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Animals; Anti-Anxiety Agents; Benzodiazepines; Caffeine; Diazepam; Humans; Motor Activity; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Purinergic

1983
Neurotransmitter receptor binding and drug discovery.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:12

    Topics: 2-Chloroadenosine; Adenosine; Animals; Barbiturates; Binding, Competitive; Diazepam; gamma-Aminobutyric Acid; Phenylisopropyladenosine; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Receptors, Purinergic; Xanthines

1983

Trials

4 trial(s) available for adenosine and diazepam

ArticleYear
Adenosine in the inhibition of diazepam sedation by aminophylline.
    Acta anaesthesiologica Scandinavica, 1986, Volume: 30, Issue:7

    Topics: Adenosine; Aged; Aged, 80 and over; Aminophylline; Anesthesia, Spinal; Clinical Trials as Topic; Diazepam; Drug Interactions; Humans; Male; Middle Aged; Prostatectomy; Receptors, Purinergic; Xanthines

1986
Aminophylline inhibition of diazepam sedation: is adenosine blockade of GABA-receptors the mechanism?
    Lancet (London, England), 1984, Feb-25, Volume: 1, Issue:8374

    Topics: Adenosine; Aminophylline; Diazepam; Humans; Receptors, Cell Surface; Receptors, GABA-A

1984
Is ACTH a key to understanding anticonvulsant action?
    Developmental medicine and child neurology, 1998, Volume: 40, Issue:2

    Topics: Adenosine; Adrenocorticotropic Hormone; Anticonvulsants; Benzodiazepines; Binding Sites; Child; Child, Preschool; Cohort Studies; Diazepam; Electroencephalography; Epilepsy; Female; Follow-Up Studies; gamma-Aminobutyric Acid; Humans; Infant; Male; Receptors, GABA-A; Severity of Illness Index

1998
The influence of diazepam and midazolam on adenosine-induced forearm vasodilation in humans.
    Journal of cardiovascular pharmacology, 2004, Volume: 43, Issue:2

    Topics: Adenosine; Adult; Anticonvulsants; Diazepam; Drug Interactions; Female; Forearm; Humans; Male; Midazolam; Plethysmography; Regional Blood Flow; Vasodilation

2004

Other Studies

62 other study(ies) available for adenosine and diazepam

ArticleYear
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Cyclic adenosine 3',5'-monophosphate in guinea-pig cerebral cortical slices: studies on the role of adenosine.
    Journal of neurochemistry, 1975, Volume: 24, Issue:6

    Topics: Adenosine; Animals; Calcium; Cerebral Cortex; Cyclic AMP; Diazepam; Guinea Pigs; Histamine; In Vitro Techniques; Norepinephrine; Time Factors

1975
Diazepam potentiation of purinergic depression of central neurons.
    Canadian journal of physiology and pharmacology, 1979, Volume: 57, Issue:4

    Topics: Adenosine; Animals; Blood Pressure; Brain; Cyclic AMP; Diazepam; Drug Synergism; Male; Neurons; Purine Nucleosides; Purines; Rats; Time Factors

1979
Anticonvulsant drug actions on in vitro and in vivo levels of cyclic AMP in the mouse brain.
    Epilepsia, 1979, Volume: 20, Issue:2

    Topics: Adenosine; Animals; Anticonvulsants; Brain; Carbamazepine; Cerebellum; Cerebral Cortex; Clonazepam; Culture Techniques; Cyclic AMP; Diazepam; Male; Mice; Norepinephrine; Ouabain; Pentylenetetrazole; Phenobarbital; Phenytoin; Potassium; Premedication; Seizures

1979
Influence of diazepam, alpidem, zolpidem and zopiclone, on the response to adenosine of the guinea pig isolated trachea.
    Fundamental & clinical pharmacology, 1991, Volume: 5, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Animals; Anti-Anxiety Agents; Diazepam; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Histamine; Hypnotics and Sedatives; Imidazoles; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, GABA-A; Trachea; Zolpidem

1991
Behavioral effects of adenosine agonists: evaluation by punishment, discrete shuttle avoidance and activity tests in mice.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:3

    Topics: Adenosine; Animals; Avoidance Learning; Caffeine; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Mice, Inbred Strains; Motor Activity; Phenylisopropyladenosine; Punishment; Reinforcement Schedule; Xanthines

1991
[Effects of diazepam and N(6)-cyclohexyladenosine on the level of diazepam-binding inhibitor in structures of the hippocampus during immobilization stress].
    Biulleten' eksperimental'noi biologii i meditsiny, 1990, Volume: 110, Issue:8

    Topics: Adenosine; Animals; Diazepam; Diazepam Binding Inhibitor; Hippocampus; Immobilization; Male; Models, Biological; Neuropeptides; Rats; Receptors, GABA-A; Receptors, Purinergic; Stress, Physiological

1990
Peripheral type benzodiazepine receptors and response to adenosine on the guinea-pig isolated trachea.
    Pulmonary pharmacology, 1990, Volume: 3, Issue:3

    Topics: Adenosine; Animals; Benzodiazepines; Clonazepam; Diazepam; Dipyridamole; Drug Synergism; GABA-A Receptor Antagonists; Guinea Pigs; Histamine; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Receptors, GABA-A; Theophylline; Trachea

1990
Chronic benzodiazepine treatment and cortical responses to adenosine and GABA.
    Brain research, 1990, Oct-22, Volume: 530, Issue:2

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Cerebral Cortex; Clonazepam; Diazepam; Electrodes; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; N-Methylaspartate; Serotonin; Theophylline

1990
Differential effects of agents enhancing purinergic transmission upon the antielectroshock efficacy of carbamazepine, diphenylhydantoin, diazepam, phenobarbital, and valproate in mice.
    Journal of neural transmission. General section, 1990, Volume: 81, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anticonvulsants; Body Temperature Regulation; Diazepam; Electroshock; Female; Mice; Phenylisopropyladenosine; Receptors, Purinergic; Seizures; Valproic Acid

1990
Imidazodiazepinediones: a new class of adenosine receptor antagonists.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:10

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Azepines; Binding, Competitive; Cell Membrane; Cerebral Cortex; Diazepam; Imidazoles; In Vitro Techniques; Molecular Conformation; Phenylisopropyladenosine; Rats; Receptors, Purinergic; Structure-Activity Relationship

1990
Adenosine receptor antagonism accounts for the seizure-prolonging effects of aminophylline.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 36, Issue:4

    Topics: Adenosine; Aminophylline; Amygdala; Animals; Brain; Carbolines; Diazepam; Flumazenil; Kindling, Neurologic; Male; Picrotoxin; Pyrazoles; Pyrrolidinones; Rats; Rats, Inbred Strains; Receptors, Purinergic; Rolipram; Seizures; Theophylline; Xanthines

1990
Antagonism of the anti-conflict effects of phenobarbital, but not diazepam, by the A-1 adenosine agonist l-PIA.
    Psychopharmacology, 1990, Volume: 102, Issue:3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Conditioning, Operant; Conflict, Psychological; Diazepam; Drinking; Female; Male; Phenobarbital; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Purinergic

1990
Discriminative stimulus properties of caffeine in the rat: noradrenergic mediation.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Adrenergic alpha-Antagonists; Animals; Apomorphine; Avoidance Learning; Caffeine; Clonidine; Diazepam; Discrimination Learning; Male; Norepinephrine; Pentobarbital; Picrotoxin; Rats; Rats, Inbred Strains; Theobromine; Theophylline

1986
Diazepam enhances the inhibitory action of adenosine on transmission at the frog neuromuscular junction.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Diazepam; Dipyridamole; Drug Synergism; In Vitro Techniques; Membrane Potentials; Motor Endplate; Muscle Contraction; Neuromuscular Junction; Rana ridibunda; Synaptic Transmission; Theophylline

1989
Neurochemical studies on quinolone antibiotics: effects on glutamate, GABA and adenosine systems in mammalian CNS.
    Pharmacology & toxicology, 1989, Volume: 64, Issue:5

    Topics: 4-Quinolones; Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Infective Agents; Aspartic Acid; Brain Chemistry; Calcium; Chlorides; Diazepam; gamma-Aminobutyric Acid; Glutamates; Ibotenic Acid; Kainic Acid; Male; Rats; Rats, Inbred Strains

1989
Dissimilarities between benzodiazepine-binding sites and adenosine uptake sites in astrocytes and neurons in primary cultures.
    Journal of neuroscience research, 1987, Volume: 17, Issue:2

    Topics: Adenosine; Animals; Astrocytes; Benzodiazepines; Binding Sites; Cells, Cultured; Diazepam; Flumazenil; Isoquinolines; Neurons; Pyrazoles; Receptors, GABA-A

1987
Theophylline antagonizes the effect of diazepam on ventricular automaticity.
    European journal of pharmacology, 1988, Oct-18, Volume: 155, Issue:3

    Topics: Adenosine; Animals; Diazepam; Female; Flumazenil; Heart Rate; Heart Ventricles; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Theophylline; Ventricular Function

1988
Pharmacological analysis of chrono- and inotropic responses to diazepam in the isolated, blood-perfused canine atrium.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 290, Issue:2

    Topics: Acetylcholine; Adenosine; Animals; Atropine; Diazepam; Dogs; Drug Interactions; Heart Rate; Imipramine; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Perfusion; Propranolol; Tyramine

1987
Effects of adenosine uptake blockers and adenosine on evoked potentials of guinea-pig olfactory cortex.
    Pflugers Archiv : European journal of physiology, 1986, Volume: 406, Issue:1

    Topics: Adenosine; Adenosine Deaminase; Animals; Diazepam; Dilazep; Dipyridamole; Evoked Potentials; Flurazepam; Guanosine; Guinea Pigs; Hexobendine; In Vitro Techniques; Limbic System; Olfactory Pathways; Thioinosine; Thionucleosides

1986
Species differences in the binding of [3H]nitrobenzylthioinosine to the nucleoside transport system in mammalian central nervous system membranes: evidence for interconvertible conformations of the binding site/transporter complex.
    Journal of neurochemistry, 1985, Volume: 45, Issue:2

    Topics: Adenosine; Animals; Binding Sites; Biological Transport, Active; Brain; Cell Membrane; Diazepam; Dipyridamole; Dogs; Erythrocytes; Female; Guinea Pigs; Humans; Inosine; Male; Mice; Nucleosides; Rabbits; Rats; Rats, Inbred Strains; Species Specificity; Thioinosine

1985
Possible mechanism of action of diazepam as an adenosine potentiator.
    European journal of pharmacology, 1985, Jul-11, Volume: 113, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Triphosphate; Animals; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Guinea Pigs; In Vitro Techniques; Intestines; Male; Muscle Contraction; Myocardial Contraction; Myocardium; Rats

1985
Adenosine 3',5'-monophosphate in guinea pig cerebral cortical slices: effect of benzodiazepines.
    Journal of neurochemistry, 1974, Volume: 22, Issue:5

    Topics: Adenosine; Animals; Cerebral Cortex; Chlordiazepoxide; Cyclic AMP; Diazepam; Histamine; Kinetics; Male; Norepinephrine; Oxazepam; Time Factors; Tranquilizing Agents

1974
Proceedings: Adenosine 3',5'-monophosphate in cerebral cortical slices from guinea pig and rat: effect of benzodiazepines.
    Naunyn-Schmiedeberg's archives of pharmacology, 1974, Volume: 282, Issue:Suppl

    Topics: Adenosine; Animals; Benzodiazepinones; Cerebral Cortex; Chlordiazepoxide; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Guinea Pigs; Histamine; In Vitro Techniques; Norepinephrine; Oxazepam; Rats

1974
Inhibition of phosphodiesterase activity in brain cortical slices from guinea pig and rat.
    Pharmacological research communications, 1974, Volume: 6, Issue:4

    Topics: Adenosine; Animals; Benzyl Compounds; Cerebral Cortex; Chlordiazepoxide; Cyclic AMP; Diazepam; Ethers; Guinea Pigs; Histamine; Hydrazines; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Oxazepam; Phosphodiesterase Inhibitors; Pyrazoles; Pyridines; Rats; Species Specificity; Theophylline

1974
Involvement of adenosine receptor activities in aggressive responses produced by clonidine in mice.
    Psychopharmacology, 1984, Volume: 83, Issue:4

    Topics: Adenosine; Aggression; Animals; Apomorphine; Bicuculline; Clonidine; Diazepam; Dipyridamole; Humans; Male; Mice; Receptors, Cell Surface; Receptors, Purinergic; Theophylline

1984
Diazepam and flurazepam inhibit adenosine uptake by rat brain synaptosomes.
    The Journal of pharmacy and pharmacology, 1980, Volume: 32, Issue:4

    Topics: Adenosine; Animals; Brain; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Flurazepam; In Vitro Techniques; Male; Rats; Synaptosomes

1980
Do benzodiazepines bind at adenosine uptake sites in CNS?
    Life sciences, 1981, Mar-02, Volume: 28, Issue:9

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Benzodiazepines; Binding Sites; Cerebral Cortex; Diazepam; Male; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Synaptosomes

1981
Inhibition of adenosine accumulation into guinea pig ventricle by benzodiazepines.
    European journal of pharmacology, 1982, Feb-26, Volume: 78, Issue:2

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Biological Transport; Diazepam; Dipyridamole; Female; Guinea Pigs; Heart Ventricles; In Vitro Techniques; Myocardium

1982
Adenosine mediates sedative action of various centrally active drugs.
    Medical hypotheses, 1982, Volume: 9, Issue:4

    Topics: Adenosine; Animals; Antipsychotic Agents; Arousal; Brain; Caffeine; Diazepam; Hypnotics and Sedatives; Phenothiazines; Rats; Receptors, Cell Surface; Receptors, Purinergic; Synapses; Synaptic Transmission; Synaptosomes; Theophylline

1982
Neuropharmacology of 3-isobutylmethylxanthine: effects on central noradrenergic systems in vivo.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 2-Chloroadenosine; Adenosine; Animals; Axons; Brain; Clonidine; Diazepam; Dihydroxyphenylalanine; Hydroxylation; Male; Methoxyhydroxyphenylglycol; Neurons; Norepinephrine; Rats; Rats, Inbred Strains; Stimulation, Chemical; Theophylline; Tyrosine 3-Monooxygenase; Yohimbine

1983
Interactions in the behavioral effects of methylxanthines and adenosine derivatives.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: Adenosine; Animals; Blood Pressure; Brain; Caffeine; Cardiac Complexes, Premature; Diazepam; Drug Interactions; Heart Rate; Male; Mice; Mice, Inbred ICR; Motor Activity; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Purinergic; Stimulation, Chemical; Xanthines

1983
Increased benzodiazepine receptor number elicited in vitro by a novel purine, EMD 28422.
    European journal of pharmacology, 1980, Oct-17, Volume: 67, Issue:2-3

    Topics: Adenosine; Animals; Binding Sites; Brain; Diazepam; In Vitro Techniques; Male; Muscimol; Purines; Radioligand Assay; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Tritium

1980
The effect of diazepam on adenosine uptake and adenosine-stimulated adenylate cyclase in guinea-pig brain.
    Canadian journal of physiology and pharmacology, 1982, Volume: 60, Issue:3

    Topics: Adenosine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Brain; Cyclic AMP; Diazepam; Guinea Pigs; In Vitro Techniques

1982
Effects of caffeine and theophylline on adenosine and benzodiazepine receptors in human brain.
    Neuroscience letters, 1982, May-28, Volume: 30, Issue:2

    Topics: Adenosine; Binding, Competitive; Brain; Caffeine; Diazepam; Humans; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A; Receptors, Purinergic; Theophylline; Xanthines

1982
Chronic caffeine consumption increases the number of brain adenosine receptors.
    Life sciences, 1983, Mar-07, Volume: 32, Issue:10

    Topics: Adenosine; Animals; Brain; Caffeine; Diazepam; Diet; Mice; Receptors, Cell Surface; Receptors, Purinergic; Xanthines

1983
Diazepam inhibition of adenosine uptake in the CNS: lack of effect on adenosine kinase.
    General pharmacology, 1983, Volume: 14, Issue:2

    Topics: Adenosine; Adenosine Kinase; Animals; Brain; Diazepam; Dipyridamole; Guinea Pigs; In Vitro Techniques; Phosphotransferases; Rats

1983
Benzodiazepine inhibition of adenosine uptake is not prevented by benzodiazepine antagonists.
    European journal of pharmacology, 1983, Jan-28, Volume: 87, Issue:1

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Brain; Diazepam; Flumazenil; Flurazepam; Hexobendine; In Vitro Techniques; Pyrazoles; Rats; Rats, Inbred Strains; Synaptosomes; Temperature

1983
Inhibition of adenosine accumulation by a CNS benzodiazepine antagonist (Ro 15-1788) and a peripheral benzodiazepine receptor ligand (Ro 05-4864).
    Neuroscience letters, 1983, Oct-31, Volume: 41, Issue:1-2

    Topics: Adenosine; Animals; Benzodiazepines; Benzodiazepinones; Central Nervous System; Diazepam; Flumazenil; Flurazepam; Hexobendine; Male; Rats; Synaptosomes; Time Factors

1983
Mechanism of potentiation by diazepam of adenosine response.
    Life sciences, 1984, Jan-02, Volume: 34, Issue:1

    Topics: 2-Chloroadenosine; Adenosine; Animals; Benzodiazepinones; Cecum; Diazepam; Dipyridamole; Dose-Response Relationship, Drug; Drug Synergism; Female; Flumazenil; Hypoxanthine; Hypoxanthines; Inosine; Male; Rats; Rats, Inbred Strains

1984
Behavioral interaction of adenosine and diazepam in mice.
    Brain research, 1984, Dec-03, Volume: 323, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Brain; Depression, Chemical; Diazepam; Drug Synergism; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Motor Activity

1984
Diazepam potentiates GABA-, but not adenosine-mediated, inhibition of neurons of the nigral pars reticulata.
    Neuropharmacology, 1983, Volume: 22, Issue:8

    Topics: Adenosine; Adenosine Monophosphate; Animals; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Evoked Potentials; gamma-Aminobutyric Acid; Glycine; Male; Muscimol; Neural Inhibition; Neural Pathways; Neurons; Rats; Rats, Inbred Strains; Substantia Nigra

1983
Possible selective inhibition of [3H]adenosine uptake by papaverine in vascular adrenergic nerves.
    European journal of pharmacology, 1982, Apr-08, Volume: 79, Issue:1-2

    Topics: Adenosine; Animals; Blood Vessels; Diazepam; Dipyridamole; Epinephrine; Male; Papaverine; Potassium Chloride; Pulmonary Artery; Rabbits; Sympathetic Nervous System

1982
Behavioral characterization of two long-lasting adenosine analogs: sedative properties and interaction with diazepam.
    Life sciences, 1981, Dec-21, Volume: 29, Issue:25

    Topics: 2-Chloroadenosine; Adenosine; Analgesia; Animals; Behavior, Animal; Diazepam; Dose-Response Relationship, Drug; Exploratory Behavior; Hot Temperature; Hypnotics and Sedatives; Male; Mice; Motor Activity

1981
Therapeutic concentrations of diazepam potentiate the effects of adenosine on isolated cardiac and smooth muscle [proceedings].
    British journal of pharmacology, 1980, Volume: 68, Issue:1

    Topics: Adenosine; Animals; Diazepam; Drug Synergism; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Rats

1980
Displacement of [3H] diazepam binding in rat brain by dipyridamole and by 1-methylisoguanosine, a marine natural product with muscle relaxant activity.
    Life sciences, 1980, Mar-31, Volume: 26, Issue:13

    Topics: Adenosine; Animals; Binding, Competitive; Brain; Diazepam; Dipyridamole; In Vitro Techniques; Kinetics; Membranes; Muscle Relaxants, Central; Protein Binding; Purines; Rats

1980
Pharmacologic and behavioral effects of EMD 28422: a novel purine which enhances (3H) diazepam binding to brain benzodiazepine receptors.
    Pharmacology, biochemistry, and behavior, 1980, Volume: 12, Issue:5

    Topics: Adenosine; Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Brain; Conflict, Psychological; Diazepam; Male; Mice; Mice, Inbred C3H; Motor Activity; Rats; Receptors, Drug

1980
Inhibition of [3H] diazepam binding to rat brain cortical synaptosomal membranes by adenosine uptake blockers.
    European journal of pharmacology, 1980, Aug-08, Volume: 65, Issue:4

    Topics: Adenosine; Animals; Binding, Competitive; Brain; Diazepam; In Vitro Techniques; Membranes; Rats; Synaptosomes

1980
Effects of diazepam on adenosine and acetylcholine release from rat cerebral cortex: further evidence for a purinergic mechanism in action of diazepam.
    British journal of pharmacology, 1980, Volume: 70, Issue:2

    Topics: Acetylcholine; Adenosine; Animals; Brain; Diazepam; Male; Pentobarbital; Purines; Rats; Theophylline

1980
Potentiation of the effects of adenosine on isolated cardiac and smooth muscle by diazepam.
    British journal of pharmacology, 1980, Volume: 71, Issue:2

    Topics: Adenosine; Animals; Diazepam; Drug Synergism; Guinea Pigs; Heart; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rats; Vas Deferens

1980
Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1 receptor agonist, reduce GABAergic transmission in different areas of the mouse brain.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:2

    Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Convulsants; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Isoniazid; Male; Mice; Mice, Inbred Strains; Purinergic P1 Receptor Antagonists; Receptors, GABA; Receptors, Purinergic P1; Seizures; Sulfur Radioisotopes; Synaptic Transmission; Tritium; Xanthines

1993
Enhancement by benzodiazepines of the inhibitory effect of adenosine on skeletal neuromuscular transmission.
    British journal of pharmacology, 1995, Volume: 116, Issue:2

    Topics: Adenosine; Animals; Benzodiazepines; Diaphragm; Diazepam; Dose-Response Relationship, Drug; Female; Male; Mice; Muscle, Skeletal; Synaptic Transmission; Tubocurarine

1995
Effects of diazepam and cyclohexyladenosine on open-field behavior in rats perinatally exposed to caffeine.
    Life sciences, 1996, Volume: 58, Issue:8

    Topics: Adenosine; Animals; Caffeine; Diazepam; Eliminative Behavior, Animal; Emotions; Female; Grooming; Locomotion; Motor Activity; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Sex Characteristics

1996
Inhibitory effects of diazepam in rat vas deferens: role of calcium.
    Acta physiologica, pharmacologica et therapeutica latinoamericana : organo de la Asociacion Latinoamericana de Ciencias Fisiologicas y [de] la Asociacion Latinoamericana de Farmacologia, 1996, Volume: 46, Issue:4

    Topics: Adenosine; Adrenergic alpha-Agonists; Animals; Benzodiazepinones; Calcium; Calcium Channels; Diazepam; GABA Agents; Male; Potassium Chloride; Rats; Rats, Wistar; Vas Deferens

1996
Sensitization by chronic diazepam treatment of A2A adenosine receptor-mediated relaxation in rat pulmonary artery.
    Life sciences, 1999, Volume: 64, Issue:2

    Topics: Adenosine; Animals; Carrier Proteins; Diazepam; Dinucleoside Phosphates; Dipyridamole; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Muscle Relaxation; Phenethylamines; Pulmonary Artery; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Thioinosine; Triazines; Triazoles; Verapamil

1999
Neuronal mechanisms of the anoxia-induced network oscillations in the rat hippocampus in vitro.
    The Journal of physiology, 2001, Oct-15, Volume: 536, Issue:Pt 2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenosine; Anesthetics, Local; Animals; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; Hypoxia, Brain; In Vitro Techniques; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periodicity; Potassium; Rats; Rats, Wistar; Tetrodotoxin; Xanthines

2001
Sedative, anticonvulsant and behaviour modifying effects of Centranthus longiflorus ssp. longiflorus: a study of comparison to diazepam.
    Die Pharmazie, 2002, Volume: 57, Issue:8

    Topics: Adenosine; Animals; Anticonvulsants; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Depression; Diazepam; Female; gamma-Aminobutyric Acid; Hypnotics and Sedatives; Male; Mice; Plant Extracts; Plants, Medicinal; Rats; Rats, Sprague-Dawley; Seizures; Sleep; Swimming; Thiopental; Turkey; Valerianaceae

2002
Organophosphate-induced convulsions and prevention of neuropathological damages.
    Toxicology, 2004, Mar-01, Volume: 196, Issue:1-2

    Topics: Acetylcholinesterase; Adenosine; Animals; Antidotes; Atropine; Brain; Cholinesterase Inhibitors; Diazepam; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Modulators; Isoflurophate; Lung; Male; Nerve Tissue Proteins; Organophosphorus Compounds; Pralidoxime Compounds; Rats; Rats, Wistar; Seizures

2004
Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
    European journal of pharmacology, 2005, Oct-31, Volume: 523, Issue:1-3

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Flumazenil; Male; Mice; Pentylenetetrazole; Phenethylamines; Purinergic Agonists; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Seizures; Substance Withdrawal Syndrome; Temazepam

2005
Adenosine receptor agonists attenuate the development of diazepam withdrawal-induced sensitization in mice.
    European journal of pharmacology, 2008, Jun-24, Volume: 588, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Convulsants; Diazepam; Hypnotics and Sedatives; Male; Mice; Pentylenetetrazole; Phenethylamines; Purinergic P1 Receptor Agonists; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

2008
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