adenine and hki 272

adenine has been researched along with hki 272 in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Chiba, M; Shibata, Y1
Alexander, WM; Browne, CM; Buhrlage, SJ; Card, JD; Dhe-Paganon, S; Eck, MJ; Ficarro, SB; Gray, NS; Lamberto, I; Marto, JA; McNally, R; Park, E; Seo, HS; Zhang, T1
Cui, Y; Feng, D; Liu, X; Zheng, M; Zhong, D1

Other Studies

3 other study(ies) available for adenine and hki 272

ArticleYear
The role of extrahepatic metabolism in the pharmacokinetics of the targeted covalent inhibitors afatinib, ibrutinib, and neratinib.
    Drug metabolism and disposition: the biological fate of chemicals, 2015, Volume: 43, Issue:3

    Topics: Adenine; Afatinib; Animals; Area Under Curve; Cytosol; Dogs; Glutathione; Hepatocytes; Humans; Kidney; Liver; Macaca fascicularis; Male; Piperidines; Pyrazoles; Pyrimidines; Quinazolines; Quinolines; Rats

2015
Leveraging Gas-Phase Fragmentation Pathways for Improved Identification and Selective Detection of Targets Modified by Covalent Probes.
    Analytical chemistry, 2016, 12-20, Volume: 88, Issue:24

    Topics: Adenine; Amino Acid Sequence; Cell Line, Tumor; Drug Discovery; Humans; Molecular Targeted Therapy; Peptides; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Pyrazoles; Pyrimidines; Quinolines; Tandem Mass Spectrometry

2016
Characterization of covalent binding of tyrosine kinase inhibitors to plasma proteins.
    Drug metabolism and pharmacokinetics, 2020, Volume: 35, Issue:5

    Topics: Acrylamides; Adenine; Aminoquinolines; Aniline Compounds; Animals; Binding Sites; Dogs; Haplorhini; Humans; Indoles; Lysine; Mice; Molecular Docking Simulation; Molecular Structure; Piperidines; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Quinolines; Rabbits; Rats; Serum Albumin, Human

2020
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