| Assay ID | Title | Year | Journal | Article |
|---|
| AID217938 | Growth inhibitory activity against human lymphoblastoid W1L2 cell line in presence of 10 uM thymidine/50 uM hypoxanthine | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID212491 | Growth inhibitory activity against mouse lymphoblastoid L1210TS cell line was determined as inhibition of thymidylate synthase | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID604932 | Cytotoxicity against human W1L2 cells | 2010 | Journal of medicinal chemistry, Dec-23, Volume: 53, Issue:24
| Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as potent inhibitors of nicotinamide phosphoribosyltransferase (Nampt). |
| AID767958 | Cytotoxicity against human W1L2 cells | 2013 | Journal of medicinal chemistry, Aug-22, Volume: 56, Issue:16
| Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors. |
| AID1057523 | Cytotoxicity against human W1L2 cells assessed as growth inhibition after 72 hrs by trypan blue assay | 2013 | Journal of medicinal chemistry, Nov-27, Volume: 56, Issue:22
| Nicotinamide phosphoribosyltransferase inhibitors, design, preparation, and structure-activity relationship. |
| AID604931 | Inhibition of thymidylate synthase | 2010 | Journal of medicinal chemistry, Dec-23, Volume: 53, Issue:24
| Analogues of 4-[(7-Bromo-2-methyl-4-oxo-3H-quinazolin-6-yl)methylprop-2-ynylamino]-N-(3-pyridylmethyl)benzamide (CB-30865) as potent inhibitors of nicotinamide phosphoribosyltransferase (Nampt). |
| AID217942 | Growth inhibitory activity against human lymphoblastoid W1L2:R865 cell line | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID28824 | Solubility at pH 6.0 | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID217937 | Growth inhibitory activity against human lymphoblastoid W1L2 cell line | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID28825 | Solubility at pH 7.4 | 2002 | Journal of medicinal chemistry, Aug-15, Volume: 45, Issue:17
| The design and synthesis of water-soluble analogues of CB30865, a quinazolin-4-one-based antitumor agent. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1347157 | Confirmatory screen GU Rhodamine qHTS for Zika virus inhibitors qHTS | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347161 | Confirmatory screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347169 | Tertiary RLuc qRT-PCR qHTS assay for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |