Proteins > Diacylglycerol O-acyltransferase 1
Page last updated: 2024-08-08 00:28:08
Diacylglycerol O-acyltransferase 1
A diacylglycerol O-acyltransferase 1 that is encoded in the genome of mouse. [OMA:Q9Z2A7, PRO:DNx]
Synonyms
EC 2.3.1.20;
Acyl-CoA retinol O-fatty-acyltransferase;
ARAT;
Retinol O-fatty-acyltransferase;
2.3.1.76;
Diglyceride acyltransferase
Research
Bioassay Publications (4)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (25.00) | 29.6817 |
2010's | 3 (75.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
azd3988 | Mus musculus (house mouse) | IC50 | 0.0011 | 1 | 1 |
a-922500 | Mus musculus (house mouse) | IC50 | 0.0183 | 2 | 3 |
azd7687 | Mus musculus (house mouse) | IC50 | 30.0000 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
pradigastat | Mus musculus (house mouse) | EC50 | 0.0710 | 1 | 1 |