A phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform that is encoded in the genome of rat. [OMA:Q9Z1L0, PRO:DNx]
PI3-kinase subunit beta;
PI3K-beta;
PI3Kbeta;
PtdIns-3-kinase subunit beta;
EC 2.7.1.153;
Phosphatidylinositol 4,5-bisphosphate 3-kinase 110 kDa catalytic subunit beta;
PtdIns-3-kinase subunit p110-beta;
p110beta
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 1 (50.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
dactolisib | Rattus norvegicus (Norway rat) | IC50 | 0.0100 | 1 | 1 |
buparlisib | Rattus norvegicus (Norway rat) | IC50 | 0.5230 | 1 | 1 |
gdc 0941 | Rattus norvegicus (Norway rat) | IC50 | 0.1460 | 1 | 1 |
byl719 | Rattus norvegicus (Norway rat) | IC50 | 2.2000 | 1 | 1 |