Page last updated: 2024-08-08 00:24:42

Glycogen synthase kinase-3 beta

A glycogen synthase kinase-3 beta that is encoded in the genome of mouse. [OMA:Q9WV60, PRO:DNx]

Synonyms

GSK-3 beta;
EC 2.7.11.26;
Serine/threonine-protein kinase GSK3B;
2.7.11.1

Research

Bioassay Publications (3)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Compounds (3)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaMus musculus (house mouse)IC500.100011
tws 119Mus musculus (house mouse)IC500.030011
azd2858Mus musculus (house mouse)IC500.076011

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tws 119Mus musculus (house mouse)EC501.000033
tws 119Mus musculus (house mouse)Kd0.126011