Page last updated: 2024-08-07 20:25:55

Short transient receptor potential channel 4

A short transient receptor potential cation channel TRPC4 that is encoded in the genome of mouse. [OMA:Q9QUQ5, PRO:DNx]

Synonyms

TrpC4;
Capacitative calcium entry channel Trp4;
Receptor-activated cation channel TRP4

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (4)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
clemizoleMus musculus (house mouse)IC506.400011
ml 204Mus musculus (house mouse)IC501.780022
N-butyl-1H-benzimidazol-2-amineMus musculus (house mouse)IC507.000022

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
4-[3-(4-fluorophenyl)-2-methyl-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid ethyl esterMus musculus (house mouse)EC504.700011