Page last updated: 2024-08-08 00:16:37
Protein-serine O-palmitoleoyltransferase porcupine
A protein-serine O-palmitoleoyltransferase porcupine that is encoded in the genome of mouse. [OMA:Q9JJJ7, PRO:DNx]
Synonyms
mPORC;
EC 2.3.1.250
Research
Bioassay Publications (5)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 5 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
lgk974 | Mus musculus (house mouse) | IC50 | 0.0007 | 3 | 3 |
g007-lk | Mus musculus (house mouse) | IC50 | 0.0250 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
N-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)thio]acetamide | Mus musculus (house mouse) | EC50 | 0.0300 | 1 | 1 |