A monoglyceride lipase that is encoded in the genome of rat. [OMA:Q8R431, PRO:DNx]
MGL;
EC 3.1.1.23;
Monoacylglycerol lipase;
MAGL
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (37.50) | 29.6817 |
2010's | 3 (37.50) | 24.3611 |
2020's | 2 (25.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
ro 48-8071 | Rattus norvegicus (Norway rat) | IC50 | 0.0065 | 1 | 1 |
1,2-benzisothiazoline-3-one | Rattus norvegicus (Norway rat) | IC50 | 0.3065 | 1 | 1 |
2-n-octyl-4-isothiazolin-3-one | Rattus norvegicus (Norway rat) | IC50 | 0.0880 | 1 | 1 |
celastrol methyl ester | Rattus norvegicus (Norway rat) | IC50 | 0.0930 | 1 | 1 |
euphol | Rattus norvegicus (Norway rat) | IC50 | 0.3150 | 1 | 1 |
urb602 | Rattus norvegicus (Norway rat) | IC50 | 119.7500 | 4 | 4 |
jzl 184 | Rattus norvegicus (Norway rat) | IC50 | 0.0250 | 1 | 1 |