Page last updated: 2024-08-07 20:09:44
Bombesin receptor subtype-3
A bombesin receptor subtype-3 that is encoded in the genome of rat. [OMA:Q8K418, PRO:DNx]
Synonyms
BRS-3
Research
Bioassay Publications (1)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (1)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
mk 5046 | Rattus norvegicus (Norway rat) | IC50 | 0.0012 | 1 | 1 |
mk 5046 | Rattus norvegicus (Norway rat) | Ki | 0.0006 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
mk 5046 | Rattus norvegicus (Norway rat) | EC50 | 0.0022 | 1 | 1 |