Page last updated: 2024-08-07 20:52:34

UDP-glucuronosyltransferase 1A1

A UDP-glucuronosyltransferase 1-2 that is encoded in the genome of rat. [PRO:DNx]

Synonyms

UGT1A1;
EC 2.4.1.17;
B1;
UDP-glucuronosyltransferase 1-1;
UDPGT 1-1;
UGT1*1;
UGT1-01;
UGT1.1

Research

Bioassay Publications (2)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (4)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
atazanavirRattus norvegicus (Norway rat)IC504.200011
mercaptopurineRattus norvegicus (Norway rat)Ki100.000011
6-thioxanthineRattus norvegicus (Norway rat)Ki100.000011
6-thiouric acidRattus norvegicus (Norway rat)Ki100.000011