Page last updated: 2024-08-07 17:14:14

[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial

A [pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial that is encoded in the genome of rat. [OMA:Q63065, PRO:DNx]

Synonyms

EC 2.7.11.2;
PDK p48;
Pyruvate dehydrogenase kinase isoform 1;
PDH kinase 1

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (1)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
sodium dichloroacetateRattus norvegicus (Norway rat)IC501,000.000011