Page last updated: 2024-08-07 21:16:17
Bile acid receptor
A bile acid receptor that is encoded in the genome of mouse. [OMA:Q60641, PRO:DNx]
Synonyms
Farnesoid X-activated receptor;
Farnesol receptor HRR-1;
Nuclear receptor subfamily 1 group H member 4;
Retinoid X receptor-interacting protein 14;
RXR-interacting protein 14
Research
Bioassay Publications (5)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (20.00) | 29.6817 |
2010's | 4 (80.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pregna-4,17-diene-3,16-dione | Mus musculus (house mouse) | IC50 | 66.5000 | 2 | 6 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
chenodeoxycholic acid | Mus musculus (house mouse) | EC50 | 16.8000 | 2 | 2 |
ganoderiol f | Mus musculus (house mouse) | EC50 | 5.0000 | 1 | 1 |
Ganodermanontriol | Mus musculus (house mouse) | EC50 | 2.5000 | 1 | 1 |
ergosterol-5,8-peroxide | Mus musculus (house mouse) | EC50 | 0.8500 | 1 | 1 |
pregna-4,17-diene-3,16-dione | Mus musculus (house mouse) | EC50 | 34.6000 | 2 | 3 |
gw 4064 | Mus musculus (house mouse) | EC50 | 2.0000 | 1 | 1 |
way-362450 | Mus musculus (house mouse) | EC50 | 0.1520 | 1 | 1 |