An endothelin-1 receptor that is encoded in the genome of pig. [OMA:Q29010, PRO:DNx]
Endothelin receptor type A;
ET-A;
ET-AR
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 5 (71.43) | 18.2507 |
| 2000's | 2 (28.57) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| rolipram | Sus scrofa (pig) | Ki | 0.0045 | 1 | 1 |
| enoximone | Sus scrofa (pig) | IC50 | 2.9000 | 1 | 1 |
| bosentan anhydrous | Sus scrofa (pig) | IC50 | 0.0075 | 1 | 1 |
| ro 46-2005 | Sus scrofa (pig) | IC50 | 0.1600 | 1 | 1 |
| rp 73401 | Sus scrofa (pig) | IC50 | 0.0010 | 1 | 1 |
| bq 123 | Sus scrofa (pig) | IC50 | 22.0000 | 1 | 1 |
| endothelins | Sus scrofa (pig) | IC50 | 0.0001 | 1 | 1 |