Page last updated: 2024-08-07 13:30:53
Dihydroorotate dehydrogenase (quinone), mitochondrial
[no definition available]
Synonyms
DHOdehase;
EC 1.3.5.2;
Dihydroorotate oxidase
Research
Bioassay Publications (3)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (66.67) | 29.6817 |
2010's | 1 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (5)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pd 156252 | Plasmodium falciparum 3D7 | IC50 | 34.7833 | 1 | 3 |
n-(3,5-dichlorophenyl)-2-methyl-3-nitrobenzamide | Plasmodium falciparum 3D7 | Ki | 32.2150 | 1 | 2 |
dsm 74 | Plasmodium falciparum 3D7 | IC50 | 26.2080 | 2 | 5 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
5,6-dihydroorotate | Plasmodium falciparum 3D7 | Km | 33,666,666.6667 | 3 | 3 |
2,3-dimethoxy-5-methyl-6-decyl-1,4-benzoquinone | Plasmodium falciparum 3D7 | Km | 16,333,333.3333 | 3 | 3 |