Page last updated: 2024-08-07 11:24:57
Oxytocin receptor
An oxytocin receptor that is encoded in the genome of mouse. [OMA:P97926, PRO:DNx]
Synonyms
OT-R
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
way 267464 | Mus musculus (house mouse) | Ki | 0.0516 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
oxytocin | Mus musculus (house mouse) | EC50 | 0.0020 | 1 | 1 |
carbetocin | Mus musculus (house mouse) | EC50 | 0.0620 | 1 | 1 |
way 267464 | Mus musculus (house mouse) | EC50 | 0.0535 | 2 | 2 |
LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism.Journal of medicinal chemistry, , 10-11, Volume: 61, Issue:19, 2018
Targets for Drug Therapy for Autism Spectrum Disorder: Challenges and Future Directions.Journal of medicinal chemistry, , 11-22, Volume: 60, Issue:22, 2017