Proteins > Inositol 1,4,5-trisphosphate receptor type 1
Page last updated: 2024-08-07 16:24:00
Inositol 1,4,5-trisphosphate receptor type 1
An inositol 1,4,5-trisphosphate receptor type 1 that is encoded in the genome of rat. [OMA:P29994, PRO:DNx]
Synonyms
IP3 receptor isoform 1;
IP-3-R;
IP3R 1;
InsP3R1;
Type 1 inositol 1,4,5-trisphosphate receptor;
Type 1 InsP3 receptor
Research
Bioassay Publications (7)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 3 (42.86) | 29.6817 |
| 2010's | 2 (28.57) | 24.3611 |
| 2020's | 2 (28.57) | 2.80 |
Compounds (3)
Drugs with Activation Measurements
Both d- and l-Glucose Polyphosphates Mimic d-Journal of medicinal chemistry, , 05-28, Volume: 63, Issue:10, 2020
[no title available]Journal of medicinal chemistry, , 03-26, Volume: 63, Issue:6, 2020
Contribution of phosphates and adenine to the potency of adenophostins at the IP₃ receptor: synthesis of all possible bisphosphates of adenophostin A.Journal of medicinal chemistry, , Feb-23, Volume: 55, Issue:4, 2012
Synthetic partial agonists reveal key steps in IP3 receptor activation.Nature chemical biology, , Volume: 5, Issue:9, 2009
Synthesis of adenophostin A analogues conjugating an aromatic group at the 5'-position as potent IP3 receptor ligands.Journal of medicinal chemistry, , Sep-21, Volume: 49, Issue:19, 2006
A systematic study of C-glucoside trisphosphates as myo-inositol trisphosphate receptor ligands. Synthesis of beta-C-glucoside trisphosphates based on the conformational restriction strategy.Journal of medicinal chemistry, , Mar-23, Volume: 49, Issue:6, 2006
Both d- and l-Glucose Polyphosphates Mimic d-Journal of medicinal chemistry, , 05-28, Volume: 63, Issue:10, 2020
[no title available]Journal of medicinal chemistry, , 03-26, Volume: 63, Issue:6, 2020
A synthetic diphosphoinositol phosphate analogue of inositol trisphosphate.MedChemComm, , Jul-01, Volume: 9, Issue:7, 2018
Contribution of phosphates and adenine to the potency of adenophostins at the IP₃ receptor: synthesis of all possible bisphosphates of adenophostin A.Journal of medicinal chemistry, , Feb-23, Volume: 55, Issue:4, 2012
Synthetic partial agonists reveal key steps in IP3 receptor activation.Nature chemical biology, , Volume: 5, Issue:9, 2009
Synthesis of adenophostin A analogues conjugating an aromatic group at the 5'-position as potent IP3 receptor ligands.Journal of medicinal chemistry, , Sep-21, Volume: 49, Issue:19, 2006
A systematic study of C-glucoside trisphosphates as myo-inositol trisphosphate receptor ligands. Synthesis of beta-C-glucoside trisphosphates based on the conformational restriction strategy.Journal of medicinal chemistry, , Mar-23, Volume: 49, Issue:6, 2006