Page last updated: 2024-08-07 16:22:11
Protein kinase C delta type
A protein kinase C delta type that is encoded in the genome of mouse. [OMA:P28867, PRO:DNx]
Synonyms
EC 2.7.11.13;
Tyrosine-protein kinase PRKCD;
2.7.10.2;
nPKC-delta
Research
Bioassay Publications (5)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (20.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 1 (20.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (4)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
phorbol 12,13-dibutyrate | Mus musculus (house mouse) | Ki | 0.0275 | 11 | 11 |
phorbol-12,13-diacetate | Mus musculus (house mouse) | Ki | 0.0346 | 8 | 8 |
indolactam v | Mus musculus (house mouse) | Ki | 1.1925 | 15 | 15 |
7-octylindolactam v | Mus musculus (house mouse) | Ki | 0.0001 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
phorbol 12,13-dibutyrate | Mus musculus (house mouse) | Kd | 0.1284 | 3 | 3 |