Proteins > Fibroblast growth factor receptor 1
Page last updated: 2024-08-07 13:02:23
Fibroblast growth factor receptor 1
A fibroblast growth factor receptor 1 that is encoded in the genome of mouse. [OMA:P16092, PRO:DAN]
Synonyms
FGFR-1;
bFGF-R-1;
EC 2.7.10.1;
Basic fibroblast growth factor receptor 1;
MFR;
Proto-oncogene c-Fgr
Research
Bioassay Publications (3)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (66.67) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 1 (33.33) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| su 5402 | Mus musculus (house mouse) | IC50 | 10.0000 | 2 | 2 |
| pd 166285 | Mus musculus (house mouse) | IC50 | 0.0430 | 1 | 1 |
| su 4984 | Mus musculus (house mouse) | IC50 | 20.0000 | 2 | 2 |
An overview of the binding models of FGFR tyrosine kinases in complex with small molecule inhibitors.European journal of medicinal chemistry, , Jan-27, Volume: 126, 2017
Structures of the tyrosine kinase domain of fibroblast growth factor receptor in complex with inhibitors.Science (New York, N.Y.), , May-09, Volume: 276, Issue:5314, 1997
An overview of the binding models of FGFR tyrosine kinases in complex with small molecule inhibitors.European journal of medicinal chemistry, , Jan-27, Volume: 126, 2017
Structures of the tyrosine kinase domain of fibroblast growth factor receptor in complex with inhibitors.Science (New York, N.Y.), , May-09, Volume: 276, Issue:5314, 1997