Page last updated: 2024-08-07 16:00:07
Dopamine beta-hydroxylase
A dopamine beta-hydroxylase that is encoded in the genome of cow. [OMA:P15101, PRO:DNx]
Synonyms
EC 1.14.17.1;
Dopamine beta-monooxygenase
Research
Bioassay Publications (8)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 4 (50.00) | 18.7374 |
1990's | 3 (37.50) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (12.50) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
fusaric acid | Bos taurus (cattle) | IC50 | 0.0500 | 1 | 1 |
fusaric acid | Bos taurus (cattle) | Ki | 0.1490 | 2 | 2 |
4-vinylphenol | Bos taurus (cattle) | Ki | 700.0000 | 1 | 1 |
methimazole | Bos taurus (cattle) | IC50 | 754.0000 | 1 | 1 |
methimazole | Bos taurus (cattle) | Ki | 380.5000 | 2 | 2 |
1-(4-hydroxybenzyl)imidazole-2-thiol | Bos taurus (cattle) | IC50 | 2.6000 | 3 | 3 |
1-(4-hydroxybenzyl)imidazole-2-thiol | Bos taurus (cattle) | Ki | 0.1513 | 3 | 3 |
sk&f 102698 | Bos taurus (cattle) | IC50 | 0.8700 | 3 | 3 |
sk&f 102698 | Bos taurus (cattle) | Ki | 0.0410 | 1 | 1 |
Drugs with Other Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
tyramine | Bos taurus (cattle) | Km | 2,000.0000 | 1 | 1 |
3-phenylpropylamine | Bos taurus (cattle) | Km | 20,400.0000 | 1 | 1 |
1-(4-hydroxybenzyl)imidazole-2-thiol | Bos taurus (cattle) | Kis | 0.1623 | 3 | 3 |
sk&f 102698 | Bos taurus (cattle) | Kis | 0.0410 | 1 | 1 |