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Cytochrome P450 2D1

A protein that is a translation product of the Cyp2d1 gene in rat. [PRO:DNx, UniProtKB:P10633]

Synonyms

EC 1.14.14.1;
CYPIID1;
Cytochrome P450-CMF1A;
Cytochrome P450-DB1;
Cytochrome P450-UT-7;
Debrisoquine 4-hydroxylase

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (7)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
debrisoquinRattus norvegicus (Norway rat)IC50529.000011
nortriptylineRattus norvegicus (Norway rat)IC50204.000011
dexpropranololRattus norvegicus (Norway rat)IC50182.000011
quinidineRattus norvegicus (Norway rat)IC5019.900011
quinineRattus norvegicus (Norway rat)IC5046.500011
codeineRattus norvegicus (Norway rat)IC501,320.000011
dextromethorphanRattus norvegicus (Norway rat)IC50264.000011