A protein kinase C alpha type that is encoded in the genome of cow. [OMA:P04409, PRO:DNx]
PKC-A;
PKC-alpha;
EC 2.7.11.13
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
pd 153035 | Bos taurus (cattle) | IC50 | 40.2872 | 1 | 5 |
phorbol 12,13-dibutyrate | Bos taurus (cattle) | Ki | 0.0002 | 1 | 1 |
1,2-dioctanoylglycerol | Bos taurus (cattle) | Ki | 0.0330 | 1 | 1 |
12-deoxyphorbol 13-acetate | Bos taurus (cattle) | Ki | 0.0048 | 1 | 1 |