Page last updated: 2024-08-07 19:25:46
M1 family aminopeptidase
[no definition available]
Synonyms
EC 3.4.11.-;
Pfa-M1
Research
Bioassay Publications (2)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (50.00) | 29.6817 |
| 2010's | 1 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (1)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| ubenimex | Plasmodium falciparum FcB1/Columbia | IC50 | 0.2840 | 1 | 1 |
| ubenimex | Plasmodium falciparum FcB1/Columbia | Ki | 0.1900 | 1 | 1 |
Synthesis of new (-)-bestatin-based inhibitor libraries reveals a novel binding mode in the S1 pocket of the essential malaria M1 metalloaminopeptidase.Journal of medicinal chemistry, , Mar-24, Volume: 54, Issue:6, 2011
Design, synthesis and antimalarial activity of novel, quinoline-based, zinc metallo-aminopeptidase inhibitors.Bioorganic & medicinal chemistry letters, , Aug-18, Volume: 13, Issue:16, 2003