Page last updated: 2024-08-07 11:21:38
Neuromedin-U receptor 1
A neuromedin-U receptor 1 that is encoded in the genome of mouse. [OMA:O55040, PRO:DNx]
Synonyms
NMU-R1;
G-protein coupled receptor 66;
G-protein coupled receptor FM-3
Research
Bioassay Publications (3)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 3 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (1)
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| neuromedin u 8 | Mus musculus (house mouse) | EC50 | 0.0036 | 3 | 3 |
A potent neuromedin U receptor 2-selective alkylated peptide.Bioorganic & medicinal chemistry letters, , 10-15, Volume: 27, Issue:20, 2017
Potent Body Weight-Lowering Effect of a Neuromedin U Receptor 2-selective PEGylated Peptide.Journal of medicinal chemistry, , 07-27, Volume: 60, Issue:14, 2017
Discovery of selective hexapeptide agonists to human neuromedin U receptors types 1 and 2.Journal of medicinal chemistry, , Aug-14, Volume: 57, Issue:15, 2014