Page last updated: 2024-08-07 12:40:43
potassium voltage-gated channel subfamily KQT member 2
[no definition available]
Synonyms
Research
Bioassay Publications (0)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0) | 18.7374 |
1990's | 0 (0) | 18.2507 |
2000's | 0 (0) | 29.6817 |
2010's | 0 (0) | 24.3611 |
2020's | 0 (0) | 2.80 |
Compounds (10)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
3-[1-azepanyl-[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl]-6,7-dimethoxy-1H-quinolin-2-one | Rattus norvegicus (Norway rat) | IC50 | 4.9554 | 1 | 0 |
N-[2-[[2-(4-chlorophenyl)-2-oxoethyl]thio]-4-oxo-3-quinazolinyl]benzamide | Rattus norvegicus (Norway rat) | IC50 | 1.5340 | 1 | 0 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
(4-chlorophenyl)-(5-hydroxy-2-methyl-4,6-dinitro-3-benzofuranyl)methanone | Rattus norvegicus (Norway rat) | EC50 | 554.6400 | 1 | 0 |
4-butyl-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thione | Rattus norvegicus (Norway rat) | EC50 | 308.3500 | 1 | 0 |
N-(4-propan-2-ylphenyl)-3-bicyclo[2.2.1]heptanecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 0.7200 | 1 | 0 |
N-(2,4,6-trimethylphenyl)-3-bicyclo[2.2.1]heptanecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 4.5716 | 6 | 0 |
n-(6-chloropyridin-3-yl)-4-fluorobenzamide | Rattus norvegicus (Norway rat) | EC50 | 3.6800 | 2 | 0 |
ica 27243 | Rattus norvegicus (Norway rat) | EC50 | 14.4000 | 1 | 0 |
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 17.3000 | 1 | 0 |
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamide | Rattus norvegicus (Norway rat) | EC50 | 38.9000 | 1 | 0 |