Page last updated: 2024-08-07 12:40:43

potassium voltage-gated channel subfamily KQT member 2

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (10)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
3-[1-azepanyl-[1-[(4-fluorophenyl)methyl]-5-tetrazolyl]methyl]-6,7-dimethoxy-1H-quinolin-2-oneRattus norvegicus (Norway rat)IC504.955410
N-[2-[[2-(4-chlorophenyl)-2-oxoethyl]thio]-4-oxo-3-quinazolinyl]benzamideRattus norvegicus (Norway rat)IC501.534010

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
(4-chlorophenyl)-(5-hydroxy-2-methyl-4,6-dinitro-3-benzofuranyl)methanoneRattus norvegicus (Norway rat)EC50554.640010
4-butyl-3-(5-propan-2-yl-3-thiophenyl)-1H-1,2,4-triazole-5-thioneRattus norvegicus (Norway rat)EC50308.350010
N-(4-propan-2-ylphenyl)-3-bicyclo[2.2.1]heptanecarboxamideRattus norvegicus (Norway rat)EC500.720010
N-(2,4,6-trimethylphenyl)-3-bicyclo[2.2.1]heptanecarboxamideRattus norvegicus (Norway rat)EC504.571660
n-(6-chloropyridin-3-yl)-4-fluorobenzamideRattus norvegicus (Norway rat)EC503.680020
ica 27243Rattus norvegicus (Norway rat)EC5014.400010
5-chloro-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(phenylmethyl)sulfonyl-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)EC5017.300010
5-chloro-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-[(4-fluorophenyl)methylsulfonyl]-4-pyrimidinecarboxamideRattus norvegicus (Norway rat)EC5038.900010