Page last updated: 2024-08-07 19:41:44
G protein-activated inward rectifier potassium channel 1
[no definition available]
Synonyms
Research
Bioassay Publications (0)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0) | 18.7374 |
1990's | 0 (0) | 18.2507 |
2000's | 0 (0) | 29.6817 |
2010's | 0 (0) | 24.3611 |
2020's | 0 (0) | 2.80 |
Compounds (5)
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
brimonidine | Rattus norvegicus (Norway rat) | EC50 | 0.0820 | 1 | 0 |
ellipticine | Rattus norvegicus (Norway rat) | EC50 | 3.0790 | 1 | 0 |
acetylcholine bromide | Rattus norvegicus (Norway rat) | EC50 | 0.1338 | 1 | 0 |
methamilane methiodide | Rattus norvegicus (Norway rat) | EC50 | 0.3933 | 1 | 0 |
1-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]urea | Rattus norvegicus (Norway rat) | EC50 | 3.2400 | 1 | 0 |