Proteins > kallikrein-5 preproprotein
Page last updated: 2024-08-07 19:24:30

kallikrein-5 preproprotein

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (53)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
carbarylHomo sapiens (human)IC5050.000010
2,3-trimethylene-4-quinazoloneHomo sapiens (human)IC504.263410
1-(4-nitrophenyl)piperidineHomo sapiens (human)IC5050.000010
1-(10-methyl-2-phenothiazinyl)ethanoneHomo sapiens (human)IC5050.000010
3-phenyl-1H-quinoxalin-2-oneHomo sapiens (human)IC5050.000010
3-methyl-2-[[oxo-(4-pentoxyphenyl)methyl]amino]butanoic acidHomo sapiens (human)IC5050.000010
2-[5-[4-(dimethylamino)phenyl]-2-tetrazolyl]-N-[2-(4-morpholinyl)phenyl]acetamideHomo sapiens (human)IC5050.000010
N-[1-(2-methoxyphenyl)-5-benzimidazolyl]benzenesulfonamideHomo sapiens (human)IC5050.000010
benzoic acid [5-amino-1-(4-methoxyphenyl)sulfonyl-3-pyrazolyl] esterHomo sapiens (human)IC502.541810
2-[[6,6-dimethyl-2-(propan-2-ylthio)-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-4-yl]thio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)IC5050.000010
4-(benzylsulfanyl)thieno[2,3-d]pyrimidineHomo sapiens (human)IC5050.000010
1-(4-chlorophenyl)-3-(4-sulfamoylphenyl)ureaHomo sapiens (human)IC5050.000010
N-(4-methylphenyl)carbamic acid (cyclopentylideneamino) esterHomo sapiens (human)IC5050.000010
2-methyl-N-(2,4,6-trimethylphenyl)-3-furancarboxamideHomo sapiens (human)IC5050.000010
(4-Methoxyphenyl)-(2-methylsulfanyl-6,7-dihydro-[1,4]dioxino[2,3-f]benzimidazol-3-yl)methanoneHomo sapiens (human)IC501.359210
[5-phenyl-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-(1-piperidinyl)methanoneHomo sapiens (human)IC5050.000010
2-[[2-(3,4-dimethylanilino)-2-oxoethyl]thio]acetamideHomo sapiens (human)IC5050.000010
N-[[3-chloro-2-(4-morpholinyl)anilino]-sulfanylidenemethyl]-4-methoxy-3-nitrobenzamideHomo sapiens (human)IC5050.000010
N-(2-fluorophenyl)-2-[2-(4-thiazolyl)-1-benzimidazolyl]acetamideHomo sapiens (human)IC5050.000010
2,4-dichloro-5-(diethylsulfamoyl)-N-(1,3,4-thiadiazol-2-yl)benzamideHomo sapiens (human)IC5050.000010
N-(9,9-dimethyl-7-oxo-8,10-dihydronaphtho[1,2-b]benzofuran-5-yl)-4-methoxybenzenesulfonamideHomo sapiens (human)IC5050.000010
4-phenyl-N-[sulfanylidene-(2,4,6-trimethylanilino)methyl]benzamideHomo sapiens (human)IC5050.000010
2-[[1-oxo-2-(2-pyrimidinylthio)ethyl]amino]-6-(phenylmethyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)IC5050.000010
4,6-dimethyl-2-[3-(4-morpholinyl)propylamino]-3-pyridinecarbonitrileHomo sapiens (human)IC5050.000010
5-(thiophen-2-ylmethyl)-1,3-diazinane-2,4,6-trioneHomo sapiens (human)IC5050.000010
N-[5-(2,4-dimethoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-phenylacetamideHomo sapiens (human)IC5050.000010
[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]-[4-(1-piperidinylsulfonyl)phenyl]methanoneHomo sapiens (human)IC5050.000010
2-(2-methyl-1-benzimidazolyl)acetic acid [2-(2-methyl-1H-indol-3-yl)-2-oxoethyl] esterHomo sapiens (human)IC5050.000010
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneHomo sapiens (human)IC5050.000010
1-anilino-3-[4-(3-anilino-2-hydroxypropoxy)phenoxy]-2-propanolHomo sapiens (human)IC5050.000010
kl001Homo sapiens (human)IC5050.000010
5-bromo-3-hydroxy-3-(4-methyl-1-piperidinyl)-1H-indol-2-oneHomo sapiens (human)IC5050.000010
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methoxy-4-propan-2-yloxybenzamideHomo sapiens (human)IC5050.000010
4-[1-(4-fluorophenyl)ethyl]-3-thiophen-2-yl-1H-1,2,4-triazole-5-thioneHomo sapiens (human)IC5050.000010
N-(5-chloro-2-pyridinyl)-2-[(1-phenyl-5-tetrazolyl)thio]propanamideHomo sapiens (human)IC5050.000010
(2,5-dimethylphenyl)-(6-methyl-5-imidazo[2,1-b]thiazolyl)methanoneHomo sapiens (human)IC5050.000010
N-(4-fluorophenyl)-5-nitro-2-pyridinamineHomo sapiens (human)IC5050.000010
7-(5-chloro-2-methoxyanilino)-6-[(4-methoxyphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-oneHomo sapiens (human)IC507.230510
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidineHomo sapiens (human)IC5050.000010
4-(2-methylphenoxy)-6-phenylfuro[2,3-d]pyrimidineHomo sapiens (human)IC5050.000010
N-[4-[[(4-tert-butylphenyl)-oxomethyl]amino]phenyl]-2-furancarboxamideHomo sapiens (human)IC5050.000010
2-chloro-N-[3-[4-[3-[[(2-chloro-5-nitrophenyl)-oxomethyl]amino]propyl]-1-piperazinyl]propyl]-5-nitrobenzamideHomo sapiens (human)IC5050.000010
5-(4-fluorophenyl)-7-(3-methoxyphenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amineHomo sapiens (human)IC5050.000010
4-chloro-N-[2-(1H-indol-3-yl)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]benzamideHomo sapiens (human)IC5050.000010
4-(3-methoxyanilino)-2-methyl-5-oxo-1-phenyl-2-pyrrolecarboxylic acid ethyl esterHomo sapiens (human)IC5050.000010
3-ethyl-2-sulfanylidene-6,7,8,9-tetrahydro-1H-pyrimido[4,5-b]quinolin-4-oneHomo sapiens (human)IC5050.000010
cladrinHomo sapiens (human)IC5050.000010
5-Chloro-3-pyridinyl 2-furoateHomo sapiens (human)IC502.441410
2-[3-[(2-chloro-4-fluorophenyl)methyl]-2-oxo-1,3-diazinan-1-yl]-N-cyclooctylacetamideHomo sapiens (human)IC5050.000010
N-(2-methoxyethyl)-2-[[3-[(4-methoxyphenyl)methyl]-6-(4-morpholinyl)-4-oxo-2-quinazolinyl]thio]acetamideHomo sapiens (human)IC5050.000010
N-[4-methyl-5-[2-(4-methylanilino)-4-thiazolyl]-2-thiazolyl]-2-furancarboxamideHomo sapiens (human)IC5050.000010
3-[5-(5-methyl-2-thiophenyl)-1,3,4-oxadiazol-2-yl]-N-[2-(3-pyridinyloxy)propyl]propanamideHomo sapiens (human)IC5050.000010
N-[4-(6-chloro-5-nitro-1H-benzimidazol-2-yl)phenyl]acetamideHomo sapiens (human)IC5050.000010