Page last updated: 2024-08-07 12:38:17

translation initiation factor eIF2B catalytic subunit epsilon

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (24)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
3H-benzo[e]indole-2-carboxylic acidSaccharomyces cerevisiae S288CIC50100.000010
7-(4-methoxyphenyl)-5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidineSaccharomyces cerevisiae S288CIC50100.000010
N-(3-bicyclo[2.2.1]heptanyl)-2-[5-(4-chlorophenyl)-2-tetrazolyl]acetamideSaccharomyces cerevisiae S288CIC50100.000010
5,8-dimethoxy-4-(4-methyl-1-piperazinyl)-2-(trifluoromethyl)quinolineSaccharomyces cerevisiae S288CIC50100.000010
arachinSaccharomyces cerevisiae S288CIC50100.000010
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenolSaccharomyces cerevisiae S288CIC50100.000010
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl esterSaccharomyces cerevisiae S288CIC50100.000010
6-(2,5-dimethoxyphenyl)-3-(3-propan-2-yloxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazineSaccharomyces cerevisiae S288CIC50100.000010
1-[(4-fluorophenyl)methyl]-3-(2-furanylmethyl)-4-imino-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-2-oneSaccharomyces cerevisiae S288CIC50100.000010
2-(2-phenylethyl)-1,3-benzoxazol-5-amineSaccharomyces cerevisiae S288CIC50100.000010
N-(4-methoxyphenyl)-N-thiophen-2-ylsulfonyl-2-furancarboxamideSaccharomyces cerevisiae S288CIC50100.000010
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamideSaccharomyces cerevisiae S288CIC50100.000010
3,4-dimethoxybenzoic acid [2-(3,4-dimethoxyphenyl)-2-oxoethyl] esterSaccharomyces cerevisiae S288CIC5017.350010
2-furanyl-[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]methanoneSaccharomyces cerevisiae S288CIC50100.000010
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidineSaccharomyces cerevisiae S288CIC5013.760010
2-[3-(2-furanylmethyl)-2,4-dioxo-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b]pyrimidin-1-yl]acetamideSaccharomyces cerevisiae S288CIC50100.000010
3,4-dihydro-2H-quinolin-1-yl-(4-propoxyphenyl)methanoneSaccharomyces cerevisiae S288CIC50100.000010
acetic acid [4-[(1-oxo-2-phenylethyl)amino]phenyl] esterSaccharomyces cerevisiae S288CIC5013.680010
7-methyl-N-[4-(4-morpholinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamideSaccharomyces cerevisiae S288CIC5018.060010
5-(4-methoxyanilino)-2-[(3-methylphenoxy)methyl]-4-oxazolecarbonitrileSaccharomyces cerevisiae S288CIC50100.000010
N-(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-3-isoxazolecarboxamideSaccharomyces cerevisiae S288CIC50100.000010
N-(4-acetylphenyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideSaccharomyces cerevisiae S288CIC50100.000010
N-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamideSaccharomyces cerevisiae S288CIC5084.910010
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidineSaccharomyces cerevisiae S288CIC5019.170010