Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
3H-benzo[e]indole-2-carboxylic acid | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
7-(4-methoxyphenyl)-5-phenyl-1,7-dihydrotetrazolo[1,5-a]pyrimidine | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-(3-bicyclo[2.2.1]heptanyl)-2-[5-(4-chlorophenyl)-2-tetrazolyl]acetamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
5,8-dimethoxy-4-(4-methyl-1-piperazinyl)-2-(trifluoromethyl)quinoline | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
arachin | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
2-[[(1-propan-2-yl-2-benzimidazolyl)amino]methyl]-6-prop-2-enylphenol | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid cyclohexyl ester | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
6-(2,5-dimethoxyphenyl)-3-(3-propan-2-yloxyphenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
1-[(4-fluorophenyl)methyl]-3-(2-furanylmethyl)-4-imino-6,6-dimethyl-5,8-dihydropyrano[2,3]thieno[2,4-b]pyrimidin-2-one | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
2-(2-phenylethyl)-1,3-benzoxazol-5-amine | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-(4-methoxyphenyl)-N-thiophen-2-ylsulfonyl-2-furancarboxamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
3,4-dimethoxybenzoic acid [2-(3,4-dimethoxyphenyl)-2-oxoethyl] ester | Saccharomyces cerevisiae S288C | IC50 | 17.3500 | 1 | 0 |
2-furanyl-[4-(2-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl)-1-piperazinyl]methanone | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
7-(4-ethyl-1-piperazinyl)-2-(3-fluorophenyl)-5-phenylpyrazolo[1,5-a]pyrimidine | Saccharomyces cerevisiae S288C | IC50 | 13.7600 | 1 | 0 |
2-[3-(2-furanylmethyl)-2,4-dioxo-6,7,8,9-tetrahydro-5H-cyclohepta[2,3]thieno[2,4-b]pyrimidin-1-yl]acetamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
3,4-dihydro-2H-quinolin-1-yl-(4-propoxyphenyl)methanone | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
acetic acid [4-[(1-oxo-2-phenylethyl)amino]phenyl] ester | Saccharomyces cerevisiae S288C | IC50 | 13.6800 | 1 | 0 |
7-methyl-N-[4-(4-morpholinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide | Saccharomyces cerevisiae S288C | IC50 | 18.0600 | 1 | 0 |
5-(4-methoxyanilino)-2-[(3-methylphenoxy)methyl]-4-oxazolecarbonitrile | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-3-isoxazolecarboxamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-(4-acetylphenyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamide | Saccharomyces cerevisiae S288C | IC50 | 100.0000 | 1 | 0 |
N-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamide | Saccharomyces cerevisiae S288C | IC50 | 84.9100 | 1 | 0 |
5-tert-butyl-7-(4-ethyl-1-piperazinyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidine | Saccharomyces cerevisiae S288C | IC50 | 19.1700 | 1 | 0 |