Proteins > orexin/Hypocretin receptor type 1 [Homo sapiens]
Page last updated: 2024-08-07 22:54:37

orexin/Hypocretin receptor type 1 [Homo sapiens]

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (10)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
8-[2-(4-methoxyphenyl)-5-phenyl-7-pyrazolo[1,5-a]pyrimidinyl]-1,4-dioxa-8-azaspiro[4.5]decaneHomo sapiens (human)IC5014.633020
6-(4-methoxyphenyl)-3-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)IC503.984020
2-(2,4,5-trimethoxyphenyl)-1,3-benzothiazoleHomo sapiens (human)IC509.047840
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2-quinolinecarboxamideHomo sapiens (human)IC504.763020
1-(1-benzotriazolyl)-3-(10-phenothiazinyl)-2-propanolHomo sapiens (human)IC5014.870020
9-chloro-6-methylindolo[3,2-b]quinoxalineHomo sapiens (human)IC502.686020
7-[(3-hydroxy-3,4-dihydro-2H-benzo[h]quinolin-1-yl)methyl]-5-thiazolo[3,2-a]pyrimidinoneHomo sapiens (human)IC5012.943840
N-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-2-quinolinecarboxamideHomo sapiens (human)IC504.417520
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidHomo sapiens (human)IC504.480020
1H-indole-4-carboxylic acid 4-[[5-(1-naphthalenyl)-1,3,4-oxadiazol-2-yl]thio]but-2-ynyl esterHomo sapiens (human)IC507.257520