Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
2-(4-amino-5-iodo-7-pyrrolo[2,3-d]pyrimidinyl)-5-(hydroxymethyl)oxolane-3,4-diol | Homo sapiens (human) | Potency | 0.0130 | 1 | 0 |
erlotinib | Homo sapiens (human) | Potency | 18.4191 | 1 | 0 |
tg 003 | Homo sapiens (human) | Potency | 0.3675 | 2 | 0 |
ml106 | Homo sapiens (human) | Potency | 0.1405 | 3 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1162 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 1.0358 | 1 | 0 |
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 26.0176 | 1 | 0 |
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 3.6751 | 1 | 0 |
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 1.4631 | 1 | 0 |
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 8.2275 | 1 | 0 |
6-(2-chlorophenyl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamine | Homo sapiens (human) | Potency | 13.0397 | 1 | 0 |
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 7.3328 | 1 | 0 |
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 9.2314 | 1 | 0 |
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 29.1922 | 1 | 0 |
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
6-(2-chlorophenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 9.2314 | 1 | 0 |
6-(3-methoxyphenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 8.2275 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 3.6751 | 1 | 0 |
6-(2-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 6.5353 | 1 | 0 |
6-(3-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 13.0397 | 1 | 0 |
6-(3-pyridinyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
6-(3-methylphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 18.4191 | 1 | 0 |
6-(1-methyl-5-indolyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 46.2666 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.3675 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-quinazolinamine | Homo sapiens (human) | Potency | 4.1235 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 1.1622 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.4627 | 1 | 0 |
6-(3-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 18.4191 | 1 | 0 |
6-(3-methylphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.4124 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-methoxyphenyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 9.2314 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-furanyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 18.4191 | 1 | 0 |
6-(2-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 11.6216 | 1 | 0 |
6-(3-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 14.6308 | 1 | 0 |
6-(3-methoxyphenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 5.8246 | 1 | 0 |
N-[(4-methyl-2-thiophenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 23.1882 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.4627 | 1 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 1.6416 | 1 | 0 |
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 3.6751 | 1 | 0 |
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.0522 | 2 | 0 |
[5-[4-[(5-methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanol | Homo sapiens (human) | Potency | 12.8102 | 3 | 0 |