Page last updated: 2024-08-07 19:23:27

dual specificity tyrosine-phosphorylation-regulated kinase 1A isoform 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (43)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
2-(4-amino-5-iodo-7-pyrrolo[2,3-d]pyrimidinyl)-5-(hydroxymethyl)oxolane-3,4-diolHomo sapiens (human)Potency0.013010
erlotinibHomo sapiens (human)Potency18.419110
tg 003Homo sapiens (human)Potency0.367520
ml106Homo sapiens (human)Potency0.140530
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency0.116210
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency1.035810
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency26.017610
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency3.675110
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.463110
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency8.227510
6-(2-chlorophenyl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency13.039710
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency7.332810
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency9.231410
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency29.192210
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
6-(2-chlorophenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency9.231410
6-(3-methoxyphenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency8.227510
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency3.675110
6-(2-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency6.535310
6-(3-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency13.039710
6-(3-pyridinyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
6-(3-methylphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency18.419110
6-(1-methyl-5-indolyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency46.266610
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.367510
N-(1,3-benzodioxol-5-ylmethyl)-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-quinazolinamineHomo sapiens (human)Potency4.123510
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.162210
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.462710
6-(3-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency18.419110
6-(3-methylphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.412410
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-methoxyphenyl)-4-quinazolinamineHomo sapiens (human)Potency9.231410
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-furanyl)-4-quinazolinamineHomo sapiens (human)Potency18.419110
6-(2-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency11.621610
6-(3-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency14.630810
6-(3-methoxyphenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency5.824610
N-[(4-methyl-2-thiophenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency23.188210
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.462710
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency1.641610
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency3.675110
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.052220
[5-[4-[(5-methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanolHomo sapiens (human)Potency12.810230