Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
2-hydroxyjuglone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
homophthalic acid | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-cyclopentyl-2-[[4-methyl-5-[4-(4-morpholinylsulfonyl)phenyl]-1,2,4-triazol-3-yl]thio]acetamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2,6-dimethyl-4-(1-phenyl-4-pyrazolyl)furo[2,3-d]pyrimidine | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
(4-Methyl-2-oxochromen-7-yl) furan-2-carboxylate | Homo sapiens (human) | IC50 | 0.9487 | 1 | 0 |
[5-(4-nitrophenyl)-2-furanyl]-(1-piperidinyl)methanone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2-furancarboxylic acid (2-acetyl-1-benzothiophen-3-yl) ester | Homo sapiens (human) | IC50 | 2.1679 | 1 | 0 |
1-[3-(4-chlorophenyl)-5-(methylthio)-1,2,4-triazol-1-yl]-1-butanone | Homo sapiens (human) | IC50 | 3.5704 | 1 | 0 |
[3-(4-chlorophenyl)-5-(methylthio)-1,2,4-triazol-1-yl]-(2-furanyl)methanone | Homo sapiens (human) | IC50 | 2.3124 | 1 | 0 |
N-(4-methyl-2-pyridinyl)-5-nitro-2-furancarboxamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
1,3-benzothiazol-2-yl-[4-(2-pyridinyl)-1-piperazinyl]methanone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
6-(chloromethyl)-N2-(3-methylphenyl)-1,3,5-triazine-2,4-diamine | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
(4-Methoxyphenyl)-(2-methylsulfanyl-6,7-dihydro-[1,4]dioxino[2,3-f]benzimidazol-3-yl)methanone | Homo sapiens (human) | IC50 | 0.9553 | 1 | 0 |
N-(4-acetylphenyl)-2-[[1-(3,5-dimethoxyphenyl)-5-tetrazolyl]thio]acetamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
4-(4-methylphenyl)-2-[[3-(4-morpholinyl)-1-oxopropyl]amino]-3-thiophenecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2-(3-chlorophenoxy)acetic acid [4-[(4-methylanilino)-oxomethyl]phenyl] ester | Homo sapiens (human) | IC50 | 0.5956 | 1 | 0 |
1-[5-(2-furanylmethylamino)-3-phenyl-1,2,4-triazol-1-yl]-2-(4-methoxyphenyl)ethanone | Homo sapiens (human) | IC50 | 8.7544 | 1 | 0 |
3-[[(4-tert-butylphenyl)-oxomethyl]amino]-1H-1,2,4-triazole-5-carboxylic acid methyl ester | Homo sapiens (human) | IC50 | 2.3916 | 1 | 0 |
1-[1-(3-fluorophenyl)-2,5-dimethyl-3-pyrrolyl]-2-[(1-methyl-5-tetrazolyl)thio]ethanone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
[3-(2-furanyl)-5-(thiophen-2-ylmethylamino)-1,2,4-triazol-1-yl]-(3-pyridinyl)methanone | Homo sapiens (human) | IC50 | 0.0010 | 1 | 0 |
1-(4-bromophenyl)-N-(3,4-dichlorophenyl)-5-oxo-3-pyrrolidinecarboxamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamide | Homo sapiens (human) | IC50 | 14.6895 | 1 | 0 |
1-[5-(2-furanylmethylamino)-3-phenyl-1,2,4-triazol-1-yl]-2-phenylethanone | Homo sapiens (human) | IC50 | 0.1000 | 1 | 0 |
2-(2,3-dimethoxyphenyl)-3-(4-methoxyphenyl)-4-thiazolidinone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |