Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
dimethylphenobarbital | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
n-benzyloxycarbonylphenylalanyl-valine | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-(3-dibenzofuranyl)-4-morpholinecarboxamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-[1-[4-(4-methylphenyl)-2-thiazolyl]-4-piperidinyl]-2,3-dihydro-1,4-benzodioxin-6-sulfonamide | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
(4-Methyl-2-oxochromen-7-yl) furan-2-carboxylate | Homo sapiens (human) | IC50 | 0.0497 | 1 | 0 |
2-furancarboxylic acid (2-acetyl-1-benzothiophen-3-yl) ester | Homo sapiens (human) | IC50 | 1.5028 | 1 | 0 |
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamide | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
(4-Methoxyphenyl)-(2-methylsulfanyl-6,7-dihydro-[1,4]dioxino[2,3-f]benzimidazol-3-yl)methanone | Homo sapiens (human) | IC50 | 3.5062 | 1 | 0 |
N-(4-fluorophenyl)-3-([1,2,4]triazolo[4,3-a]quinolin-1-ylthio)propanamide | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
2-[[cyclohexyl(oxo)methyl]amino]acetic acid [2-(4-cyanoanilino)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 50.0000 | 2 | 0 |
3-chloro-1-(4-methoxyphenyl)-4-(3-methyl-1-piperidinyl)pyrrole-2,5-dione | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
2-bromo-6-[1,4-dioxa-8-azaspiro[4.5]decan-8-yl(oxo)methyl]-11-pyrido[2,1-b]quinazolinone | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
N-(4-ethylphenyl)-3-(1-pyrrolyl)propanamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |
5-Chloro-3-pyridinyl 2-furoate | Homo sapiens (human) | IC50 | 0.7412 | 1 | 0 |
N-[4-(6-chloro-5-nitro-1H-benzimidazol-2-yl)phenyl]acetamide | Homo sapiens (human) | IC50 | 50.0000 | 1 | 0 |