zstk474 has been researched along with Primary-Myelofibrosis* in 1 studies
1 other study(ies) available for zstk474 and Primary-Myelofibrosis
Article | Year |
---|---|
Structural effects of morpholine replacement in ZSTK474 on Class I PI3K isoform inhibition: Development of novel MEK/PI3K bifunctional inhibitors.
Topics: Animals; Binding Sites; Cell Line, Tumor; Cell Proliferation; Disease Models, Animal; Humans; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase Kinases; Molecular Docking Simulation; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Primary Myelofibrosis; Protein Isoforms; Structure-Activity Relationship; Triazines | 2022 |