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zeneca zd 6169 and Muscle Relaxation

zeneca zd 6169 has been researched along with Muscle Relaxation in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's6 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Antane, MM; Antane, SA; Argentieri, TM; Butera, JA; Freeden, C; Graceffa, RF; Hirth, BH; Jenkins, D; Lennox, JR; Matelan, E; Norton, NW; Quagliato, D; Sheldon, JH; Spinelli, W; Warga, D; Wojdan, A; Woods, M1
Antane, MM; Argentieri, TM; Butera, JA; Francisco, GD; Freeden, C; Gilbert, AM; Graceffa, RF; Gundersen, EG; Herbst, D; Hirth, BH; Lennox, JR; McFarlane, G; Norton, NW; Quagliato, D; Sheldon, JH; Warga, D; Wojdan, A; Woods, M1
Brune, ME; Buckner, SA; Carroll, WA; Coghlan, MJ; Fey, TA; Gopalakrishnan, M; Gregg, RJ; Kort, ME; Perez-Medrano, A; Scott, VE; Sullivan, JP; Whiteaker, KL1
Brioni, JD; Buckner, SA; Carroll, WA; Chapple, CR; Chess-Williams, R; Coghlan, MJ; Davis-Taber, R; Daza, AV; Gopalakrishnan, M; Liu, D; Liu, Y; Milicic, I; Molinari, EJ; Scott, VE; Sellers, D; Shieh, CC; Sullivan, JP; Whiteaker, KL; Williams, M1
Brioni, JD; Buckner, SA; Coghlan, MJ; Feng, J; Gopalakrishnan, M; Shieh, CC; Sullivan, JP1
Ikawa, S; Ito, Y; Naito, S; Seki, N; Takano, N; Tanaka, K; Teramoto, N; Yunoki, T1

Other Studies

6 other study(ies) available for zeneca zd 6169 and Muscle Relaxation

ArticleYear
Design and SAR of novel potassium channel openers targeted for urge urinary incontinence. 1. N-Cyanoguanidine bioisosteres possessing in vivo bladder selectivity.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Adenosine Triphosphate; Animals; Blood Pressure; Cyclobutanes; Drug Design; Drug Evaluation, Preclinical; Female; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitriles; Patch-Clamp Techniques; Potassium Channels; Potassium Chloride; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Urinary Bladder; Urinary Incontinence

2000
Design and SAR of novel potassium channel openers targeted for urge urinary incontinence. 2. Selective and potent benzylamino cyclobutenediones.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Adenosine Triphosphate; Animals; Benzylamines; Blood Pressure; Cyclobutanes; Drug Design; Drug Evaluation, Preclinical; Female; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Potassium Channels; Potassium Chloride; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Urinary Bladder; Urinary Incontinence

2000
Structure-activity studies of novel cyanoguanidine ATP-sensitive potassium channel openers for the treatment of overactive bladder.
    Journal of medicinal chemistry, 2007, Nov-29, Volume: 50, Issue:24

    Topics: Administration, Oral; Animals; Benzamides; Biological Availability; Crystallography, X-Ray; Dogs; Electric Stimulation; Female; Guanidines; Humans; In Vitro Techniques; Ion Channel Gating; KATP Channels; Muscle Relaxation; Muscle, Smooth; Potassium Channels, Inwardly Rectifying; Structure-Activity Relationship; Swine; Urinary Bladder; Urinary Bladder, Overactive; Urodynamics

2007
(-)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637): a novel ATP-sensitive potassium channel opener efficacious in suppressing urinary bladder contractions. I. In vitro characterization.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: Amides; Animals; Aorta, Thoracic; ATP-Binding Cassette Transporters; Benzophenones; Cyclic S-Oxides; Cyclobutanes; Guinea Pigs; Humans; In Vitro Techniques; Ion Channel Gating; KATP Channels; Kinetics; Male; Membrane Potentials; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Nitriles; Patch-Clamp Techniques; Portal Vein; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Quinolones; Rats; Rats, Sprague-Dawley; Urinary Bladder

2002
Functional implication of spare ATP-sensitive K(+) channels in bladder smooth muscle cells.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:3

    Topics: Acetylcholine; Amides; Animals; Benzophenones; Drug Interactions; Electrophysiology; Guanidines; Guinea Pigs; In Vitro Techniques; Membrane Potentials; Membrane Proteins; Muscle Relaxation; Muscle, Smooth; Pinacidil; Potassium Channels; Pyridines; Swine; Urinary Bladder; Vasodilator Agents

2001
The involvement of L-type Ca(2+) channels in the relaxant effects of the ATP-sensitive K(+) channel opener ZD6169 on pig urethral smooth muscle.
    British journal of pharmacology, 2001, Volume: 134, Issue:7

    Topics: Adenosine Triphosphate; Amides; Animals; Barium; Benzophenones; Calcium Channel Blockers; Calcium Channels, L-Type; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gene Expression; Glyburide; In Vitro Techniques; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channels; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Urethra

2001