Page last updated: 2024-09-02

zacopride and Emesis

zacopride has been researched along with Emesis in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19903 (25.00)18.7374
1990's8 (66.67)18.2507
2000's1 (8.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Airey, JE; Campbell, HF; Darkes, P; Fitzpatrick, LR; Klein, S; Neuenschwander, K; Pendley, CE; Powers, M; Schnapper, M; Youssefyeh, RD1
Airey, JE; Campbell, HF; Golec, S; Klein, S; Powers, M; Rodriguez, W; Schnapper, M; Studt, W; Woodward, R; Youssefyeh, RD1
Imazumi, K; Matsui, S; Matsuo, M; Mutoh, S; Nakayama, H; Yamakuni, H1
Chen, Y; Matsuki, N; Saito, H1
Fink-Jensen, A; Hansen, JB; Honoré, T; Jacobsen, P; Judge, ME; Olney, J; Turski, L1
Andrews, PL; Bhandari, P1
Gandara, DR; Hesketh, PJ1
King, GL1
King, GL; Landauer, MR1
Bloomquist, W; Cohen, ML; Gidda, JS; Lacefield, W1
Alphin, RS; Jackson, CB; Sancilio, LF; Smith, WL1
Lucot, JB1

Other Studies

12 other study(ies) available for zacopride and Emesis

ArticleYear
Development of high-affinity 5-HT3 receptor antagonists. 1. Initial structure-activity relationship of novel benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Animals; Antiemetics; Benzamides; Benzofurans; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Male; Metoclopramide; Molecular Structure; Ondansetron; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting

1992
Development of high-affinity 5-HT3 receptor antagonists. 2. Two novel tricyclic benzamides.
    Journal of medicinal chemistry, 1992, Mar-06, Volume: 35, Issue:5

    Topics: Amides; Animals; Antiemetics; Benzamides; Benzofurans; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Cisplatin; Dogs; Ferrets; Guinea Pigs; Ileum; Molecular Structure; Muscle Contraction; Rats; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Vomiting; X-Ray Diffraction

1992
Inhibitory effect of zacopride on Cisplatin-induced delayed emesis in ferrets.
    Journal of pharmacological sciences, 2006, Volume: 101, Issue:1

    Topics: Animals; Antiemetics; Antineoplastic Agents; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Drug Therapy, Combination; Ferrets; Granisetron; Male; Serotonin Antagonists; Time Factors; Vomiting

2006
Ethanol-induced emesis in the house musk shrew, Suncus murinus.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaldehyde; Alcohol Deterrents; Animals; Antiemetics; Baclofen; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Disulfiram; Dose-Response Relationship, Drug; Ethanol; Female; GABA Antagonists; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Male; Piperidines; Serotonin Antagonists; Serotonin Receptor Agonists; Shrews; Tiopronin; Tropisetron; Vagotomy; Vomiting

1997
Inhibition of cisplatin-induced emesis in ferrets by the non-NMDA receptor antagonists NBQX and CNQX.
    Neuroscience letters, 1992, Mar-30, Volume: 137, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisplatin; Exploratory Behavior; Ferrets; Imidazoles; Male; Ondansetron; Quinoxalines; Receptors, Amino Acid; Receptors, Cell Surface; Serotonin Antagonists; Vomiting

1992
Preliminary evidence for the involvement of the putative 5-HT4 receptor in zacopride- and copper sulphate-induced vomiting in the ferret.
    European journal of pharmacology, 1991, Nov-12, Volume: 204, Issue:3

    Topics: Analysis of Variance; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Copper; Copper Sulfate; Female; Ferrets; Granisetron; Imidazoles; Indazoles; Indoles; Loperamide; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting

1991
Serotonin antagonists: a new class of antiemetic agents.
    Journal of the National Cancer Institute, 1991, May-01, Volume: 83, Issue:9

    Topics: Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Granisetron; Humans; Imidazoles; Indazoles; Indoles; Metoclopramide; Ondansetron; Quinolizines; Receptors, Serotonin; Serotonin Antagonists; Tropanes; Tropisetron; Vomiting

1991
Emesis and defecations induced by the 5-hydroxytryptamine (5-HT3) receptor antagonist zacopride in the ferret.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Administration, Oral; Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Defecation; Dose-Response Relationship, Drug; Ferrets; Granisetron; Indazoles; Injections, Intravenous; Male; Metoclopramide; Pyrazoles; Serotonin; Serotonin Antagonists; Vagotomy; Vomiting

1990
Effects of zacopride and BMY25801 (batanopride) on radiation-induced emesis and locomotor behavior in the ferret.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Animals; Antiemetics; Behavior, Animal; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Dose-Response Relationship, Radiation; Ferrets; Gait; Injections, Intraperitoneal; Male; Metoclopramide; Radiation Injuries, Experimental; Vagotomy; Vomiting

1990
Comparison of the 5-HT3 receptor antagonist properties of ICS 205-930, GR38032F and zacopride.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Carbachol; Cisplatin; Guinea Pigs; Heart Rate; Imidazoles; In Vitro Techniques; Indoles; Male; Ondansetron; Receptors, Serotonin; Serotonin Antagonists; Tropisetron; Vomiting

1989
The antiemetic profile of zacopride.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:2

    Topics: Animals; Antiemetics; Antineoplastic Agents; Apomorphine; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Copper; Copper Sulfate; Dogs; Female; Histamine Antagonists; Male; Peptide YY; Peptides; Pilocarpine; Protoveratrines; Vomiting

1989
Blockade of 5-hydroxytryptamine3 receptors prevents cisplatin-induced but not motion- or xylazine-induced emesis in the cat.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:1

    Topics: Animals; Antiemetics; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cats; Cisplatin; Indoles; Motion Sickness; Receptors, Serotonin; Serotonin Antagonists; Thiazines; Tropanes; Tropisetron; Vomiting; Xylazine

1989